“betaine hydrochloride”的搜索结果

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  1. Tebanicline hydrochloride

    Catalog No. A21918
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    nAChR modulator
    Tebanicline hydrochloride (ABT594 hydrochloride) is a nAChR modulator with potent, orally effective analgesic activity. 了解更多
  2. Gaboxadol hydrochloride

    Catalog No. A21730
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    GABAA receptors agonist
    Gaboxadol hydrochloride (Lu 02-030 hydrochloride) is a selective agonist at GABAA receptors that contain α4-δ subunits, and has anxiolytic and sedative effects. 了解更多
  3. Varenicline Hydrochloride

    Catalog No. A21539
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    α4β2 nAChR partial agonist
    Varenicline Hydrochloride (CP 526555 hydrochloride) is a high affinity, selective α4β2 nicotine acetylcholine receptor (nAChR) partial agonist and full α7 nAChR agonist. 了解更多
  4. SDZ 220-581 hydrochloride, SDZ220-581, SDZ-220-581

    Catalog No. A21897
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    NMDA receptor antagonist
    SDZ 220-581 hydrochloride is an orally active, potent, competitive NMDA receptor antagonist with pKi value of 7.7. 了解更多
  5. LY2365109 hydrochloride

    Catalog No. A21779
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    GlyT1 inhibitor
    LY2365109 hydrochloride is a potent and selective GlyT1 inhibitor, with an IC50 of 15.8 nM for glycine uptake in cells over-expressing hGlyT1a. 了解更多
  6. mAChR-IN-1 hydrochloride

    Catalog No. A21398
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    mAChR antagonist
    mAChR-IN-1 hydrochloride is a potent muscarinic cholinergic receptor (mAChR) antagonist, with an IC50 of 17 nM. 了解更多
  7. CP-409092 hydrochloride

    Catalog No. A21397
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    GABAA receptor partial agonist
    CP-409092 hydrochloride is a partial agonist of GABAA receptor, with anti-anxiety activity. 了解更多
  8. KN-92 hydrochloride

    Catalog No. A15138
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    CaMK-II 抑制剂
    KN-92 hydrochloride是KN-93的阴性对照。 了解更多
  9. EVP-6124 hydrochloride

    Catalog No. A15087
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    nAChR 抑制剂
    EVP-6124 hydrochloride是一种新型的α7神经元烟碱型乙酰胆碱受体(nAChRs)的部分激动剂。EVP-6124对α7nAChRs具有选择性,并且不激活或抑制异源α4β2nAChRs。 了解更多
  10. Cevimeline hydrochloride

    Catalog No. A18092
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    mAChR agonist
    Cevimeline (Evoxac) Hcl is a parasympathomimetic and muscarinic agonist, with particular effect on M3 receptors; used in the treatment of dry mouth associated with sjogren's syndrome. 了解更多
  11. Mecamylamine Hydrochloride

    Catalog No. A17884
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    nAChR antagonist
    Mecamylamine hydrochloride is a nAChR antagonist previously used to treat hypertension. It displays a wide variety of activities, including reducing depression-like behaviors in subjects with Tourette's syndrome and improving rates of smoking cessation. 了解更多
  12. Pitofenone Hydrochloride

    Catalog No. A17053
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    Antispasmodic Agent
    Pitofenone Hydrochloride是抗痉化合物。它是乙酰胆碱酯酶活性的有效抑制剂。 了解更多
  13. Acotiamide hydrochloride trihydrate

    Catalog No. A15782
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    AChE 抑制剂
    Acotiamide hydrochloride trihydrate是一种在日本获准用于治疗餐后饱胀,上腹胀气和功能性消化不良引起的早饱的药物。 了解更多
  14. Cevimeline hydrochloride hemihydrate

    Catalog No. A15042
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    M1 激动剂
    Cevimeline hydrochloride hemihydrate是一种新型毒蕈碱受体激动剂,是干燥综合征干燥症的候选治疗药物。 了解更多
  15. Phenoxybenzamine hydrochloride

    Catalog No. A10719
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    α-adrenergic (AR) 拮抗剂/CaM 抑制剂
    Phenoxybenzamine hydrochloride是一种细胞可渗透的,非特异性的,不可逆的α-肾上腺素(AR)拮抗剂,也可作为CaM抑制剂。 了解更多
  16. Gabapentin Hydrochloride

    Catalog No. A10414
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    Gabapentin Hydrochloride是一种加巴类似物。 了解更多
  17. GW791343 trihydrochloride

    Catalog No. A21204
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    P2X7 allosteric modulator
    GW791343 3Hcl is a P2X7 allosteric modulator; exhibits species-specific activity and acts as a negative allosteric modulator of human P2X7 (pIC50 = 6.9 - 7.2). 了解更多
  18. GTS-21 (DMBX-A)

    Catalog No. A15950
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    nAChR 激动剂
    GTS-21 dihydrochloride (DMBX-A)是一种选择性的α7烟碱乙酰胆碱受体激动剂,最近已被确定为一种有希望的炎症治疗方法。 了解更多
  19. Fexofenadine HCl

    Catalog No. A11859
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    COX 抑制剂/histamine H1 receptor 激动剂
    Fexofenadine Hydrochloride是一种抗组胺药,可抑制Cox-1,Cox-2,并且是组胺H1受体激动剂,IC50为246 nM。 了解更多
  20. Adiphenine HCl

    Catalog No. A11716
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    AChR抑制剂
    Adiphenine Hydrochloride是烟碱受体抑制剂,IC50为15μM,用作解痉药物。 了解更多
  21. Dimebon 2HCl

    Catalog No. A10312
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    Neuroprotectant
    Dimebon dihydrochloride是一种非选择性的抗组胺药,具有增强认知能力。 了解更多
  22. ARL-15896

    Catalog No. A13858
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    NMDA receptor ion channel 拮抗剂
    ARL-15896是新型的N-甲基-D-天冬氨酸受体离子通道拮抗剂。 了解更多
  23. Deoxyvasicine HCl

    Catalog No. A13925
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    AChE 抑制剂
    Desoxypeganine hydrochloride是一种AChE(乙酰胆碱酯酶)抑制剂,已用于治疗阿尔茨海默氏痴呆症。 了解更多
  24. Ticlopidine HCl

    Catalog No. A11690
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    Ticlopidine是一种二磷酸腺苷(ADP)受体抑制剂。它通过阻断ADP受体来改变血小板膜的功能,从而抑制血小板聚集。这防止了糖蛋白IIb/IIIa的构象变化,从而使血小板与血纤蛋白原结合。 了解更多
  25. Prasugrel Hydrochloride

    Catalog No. A16144
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    P2Y12 拮抗剂
    Prasugrel Hydrochloride是噻吩并吡啶ADP受体(P2Y12)拮抗剂,用于减少血栓性心血管事件。 了解更多
  26. Etifoxine hydrochloride

    Catalog No. A15084
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    Anxiolytic anticonvulsant
    Etifoxine hydrochloride是培养的神经元中GABAA受体功能的增强剂。 了解更多
  27. A 438079 hydrochloride

    Catalog No. A14983
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    P2X7 receptor 拮抗剂
    A 438079 hydrochloride是一种竞争性P2X7受体拮抗剂(抑制人重组P2X7细胞系中Ca2+流入的pIC50 = 6.9)。 了解更多
  28. Donepezil hydrochloride

    Catalog No. A10330
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    cholinesterase 抑制剂
    Donepezil hydrochloride是一种中枢可逆的乙酰胆碱酯酶抑制剂。 了解更多
  29. Biperiden HCl

    Catalog No. A10147
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    Muscarinic receptor antagonist
    Biperiden HCl是毒蕈碱受体拮抗剂,对M1亚型表现出一定的选择性。 了解更多
  30. SKF 89976A HCl

    Catalog No. A10849
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    GABA uptake 抑制剂
    SKF 89976A HCl是一种有效的GABA吸收抑制剂,hGAT-1,rGAT-2,hGAT-3和hBGT-1的IC50分别为0.13、550、944和7210μM。 了解更多
  31. Tacrine HCl Hydrate

    Catalog No. A16970
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    AChE and BChE 抑制剂
    Tacrine hydrochloride hydrate是乙酰(AChE)和丁酰胆碱酯酶(BChE)的抑制剂,IC50分别为31 nM和25.6 nM。 了解更多
  32. Tiagabine hydrochloride

    Catalog No. A16135
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    GABA reuptake 抑制剂
    Tiagabine hydrochloride是一种抗惊厥药。该药物还用于治疗惊恐症,还有其他一些抗惊厥药。 了解更多
  33. Guvacine hydrochloride

    Catalog No. A13613
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    GABA uptake 抑制剂
    Guvacine hydrochloride可抑制GABA的摄取(hGABA T-1,rGABA T-2,hGABA T-3和hBGT-1的IC50值分别为14、58、119和1870 uM)。 了解更多
  34. Memantine hydrochloride

    Catalog No. A11708
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    NMDA receptor 拮抗剂
    Memantine hydrochloride是nmda受体的拮抗剂,与离子通道位点结合。它还是CYP2B6和CYP2D6抑制剂,作用于重组CYP2B6和CYP2D6,Ki分别为0.51 nM和94.9 μM。它被用于治疗帕金森综合征。 了解更多

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