“ADM Hydrochloride”的搜索结果

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  1. Amsacrine hydrochloride

    Catalog No. A17707
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    antineoplastic agent
    Amsacrine hydrochloride (m-AMSA hydrochloride; acridinyl anisidide hydrochloride) is an inhibitor of topoisomerase II, and acts as an antineoplastic agent which can intercalates into the DNA of tumor cells. 了解更多
  2. Niraparib hydrochloride

    Catalog No. A18018
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    PARP1 and PARP2 inhibitor
    Niraparib hydrochloride (MK-4827 hydrochloride) is a highly potent and orally bioavailable PARP1 and PARP2 inhibitor with IC50s of 3.8 and 2.1 nM, respectively. 了解更多
  3. Resminostat hydrochloride

    Catalog No. A15220
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    HDAC 抑制剂
    Resminostat hydrochloride是HDAC1/3/6的有效抑制剂(IC50 = 43-72 nM);对HDAC8的效力较低,IC50为877 nM。 了解更多
  4. Givinostat hydrochloride

    Catalog No. A21487
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    HDAC inhibitor
    Givinostat hydrochloride (ITF-2357 hydrochloride) is a HDAC inhibitor with an IC50 of 198 and 157 nM for HDAC1 and HDAC3, respectively. 了解更多
  5. Pirarubicin Hydrochloride

    Catalog No. A18037
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    topoisomerase II inhibitor
    Pirarubicin Hydrochloride is an anthracycline antibiotics, acts as a topoisomerase II inhibitor, and is a widely used for treatment of various cancers, in particular, solid tumors. 了解更多
  6. Voreloxin Hydrochloride

    Catalog No. A15280
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    Topoisomerase 抑制剂
    Voreloxin hydrochloride是一种小分子,是具有抗肿瘤活性的萘啶类似物;Topo II抑制剂。 了解更多
  7. SRT 1720 Hydrochloride

    Catalog No. A21143
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    SIRT1 activator of
    SRT 1720 Hydrochloride is a selective activator of SIRT1 with an EC50 of 0.10 μM, and shows less potent activities on SIRT2 and SIRT3. 了解更多
  8. PJ 34 hydrochloride

    Catalog No. A12665
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    PARP 抑制剂
    PJ 34 hydrochloride是聚(ADP-核糖)聚合酶(PARP)(EC50 = 20 nM)的有效抑制剂。 了解更多
  9. Bleomycin hydrochloride

    Catalog No. A12773
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  10. Mitoxantrone Hydrochloride

    Catalog No. A10596
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    Mitoxantrone Dihydrochloride是一种抗病毒,抗菌,抗原生动物,免疫调节和抗肿瘤细胞抑制性蒽醌衍生物。 了解更多
  11. Epirubicin HCl

    Catalog No. A10345
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    Topoisomerase II 抑制剂
    Epirubicin HCl是一种可透过细胞的蒽环类抗肿瘤抗生素。它用于抑制拓扑异构酶II和DNA解旋酶活性。 了解更多
  12. PIK-75 hydrochloride

    Catalog No. A10729
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    PI3K 抑制剂
    PIK-75是一种p110α抑制剂,IC50值为5.8nM。在p110γ和p110β的效果较差,IC50值为0.076 ?M和1.3 ?M。 了解更多
  13. Veliparib dihydrochloride

    Catalog No. A21356
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    PARP inhibitor
    Veliparib dihydrochloride is a potent PARP inhibitor, inhibiting PARP1 and PARP2 with Kis of 5.2 and 2.9 nM, respectively. 了解更多
  14. Hoechst 33258 trihydrochloride

    Catalog No. A15106
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    Hoechst 33258 trihydrochloride是用于DNA定量的细胞染料 了解更多
  15. Nolatrexed Dihydrochloride

    Catalog No. A13261
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    Thymidylate synthase 抑制剂
    Nolatrexed Dihydrochloride是一种抗叶酸胸苷酸合酶抑制剂。 了解更多
  16. TAS-102

    Catalog No. A15533
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    Trifluridine-tipiracil hydrochloride mixture
    TAS-102是一种生物利用的联合剂,由细胞毒性嘧啶类似物三氟吡啶(5-三氟-2α-脱氧胸苷或TFT)和胸苷磷酸化酶抑制剂(TPI)替吡西酯盐酸盐组成,摩尔比为1.0:0.5(TFT :TPI),具有潜在的抗肿瘤活性。 了解更多
  17. Sarafloxacin HCl

    Catalog No. A11659
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    Topoisomerase 抑制剂
    Sarafloxacin hydrochloride是氟喹诺酮类抗菌剂。抑制细菌DNA促旋酶(拓扑异构酶)。 了解更多
  18. Bendamustine HCl (SDX-105)

    Catalog No. A10124
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    Bendamustine Hydrochloride (SDX-105)是一种小分子双功能DNA烷基化剂,结合了氮芥菜碱功能和嘌呤类似物结构。苯达莫司汀具有致密的破坏DNA的功能,使其与用作抗增殖剂的其他化合物区分开来,这些功能被认为可通过多种不同途径(包括凋亡和有丝分裂灾难)促进细胞死亡。 了解更多
  19. Lincomycin hydrochloride (U-10149A)

    Catalog No. A10532
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    Lincomycin hydrochloride是Lincomycin的一水盐,是从林肯链霉菌中分离的林肯酰胺抗生素,据报道其抑制细菌蛋白质合成并依赖于浓度。 了解更多

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