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  1. AZD3839 free base

    Catalog No. A21606
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    BACE1 inhibitor
    AZD3839 (free base) is a potent and selective BACE1 inhibitor with IC50 of 23.6 uM, about 14-fold selectivity over BACE2, also a β-secretase enzyme inhibitor. 了解更多
  2. Lanabecestat

    Catalog No. A12282
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    BACE1 inhibitor
    Lanabecestat (AZD3293) is a potent, highly permeable, orally active and blood-brain barrier penetrating BACE1 inhibitor with a Ki of 0.4 nM. 了解更多
  3. AZD7986

    Catalog No. A17095
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    DPPI 抑制剂
    AZD7986,也称为INS 1007,是第二代可逆共价,有效和选择性DPP1抑制剂,潜在地可用于治疗慢性阻塞性肺疾病(COPD),其预测的人PK特性适用于每日一次人类给药。 了解更多
  4. Alvelestat

    Catalog No. A12779
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    neutrophil elastase 抑制剂
    Avelestat,也称为AZD9668,是可口服的,高度选择性neutrophil elastase (NE)抑制剂,IC50和Ki分别为12 nM和9.4 nM,其选择性超过其他丝氨酸蛋白酶至少600倍。 了解更多
  5. AZD3839

    Catalog No. A12825
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    BACE1 抑制剂
    AZD3839是人类BACE1的有效选择性抑制剂,Ki为26.1 nM。 了解更多

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