“Acetyl glycitin”的搜索结果

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  1. Tubacin

    Catalog No. A10954
    HDAC6 抑制剂
    Tubacin (tubulin acetylation inducer)是一种高效且选择性强,可逆,可透过细胞的HDAC6抑制剂,IC50为4 nM。 了解更多
  2. CI994 (Tacedinaline)

    Catalog No. A11964
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    HDAC 抑制剂
    CI994 (Tacedinaline)是一种组蛋白脱乙酰基酶(HDAC)抑制剂,可在活细胞中诱导组蛋白超乙酰化。 了解更多
  3. Splitomicin

    Catalog No. A14221
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    NAD(+)-dependent histone deacetylase Sir2p 抑制剂
    Splitomicin是一种选择性的NAD(+)-依赖性组蛋白脱乙酰基酶Sir2p抑制剂,IC50为60 uM,在基于细胞的测定中显示出更高的活性。 了解更多
  4. TC-H 106

    Catalog No. A15357
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    HDAC 抑制剂
    TC-H 106是一种慢速,紧密结合的I类HDAC(组蛋白脱乙酰基酶)抑制剂。 了解更多
  5. M344

    Catalog No. A11355
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    HDAC 抑制剂
    M344是HDAC的有效抑制剂,IC50为100 nM,能够诱导细胞分化。 了解更多
  6. CM-675

    Catalog No. A18741
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    PDE5/HDAC-1 inhibitor
    CM-675 is a dual phosphodiesterase 5 (PDE5) and class I histone deacetylases-selective inhibitor, with IC50 values of 114 nM and 673 nM for PDE5 and HDAC1, respectively. CM-675 has potential to treat Alzheimer??s disease. 了解更多
  7. Ac-Lys-AMC

    Catalog No. A18461
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    fluorescent substrate for HDAC
    Ac-Lys-AMC (Hexanamide), also termed MAL, is a fluorescent substrate for histone deacetylase HDACs. 了解更多
  8. SW-100

    Catalog No. A18947
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    HDAC6 inhibitor
    SW-100, a selective histone deacetylase 6 (HDAC6) inhibitor with an IC50 of 2.3 nM, shows at least 1000-fold selectivity for HDAC6 relative to all other HDAC isozymes. 了解更多
  9. CHDI-390576

    Catalog No. A18899
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    HDAC inhibitor
    CHDI-390576, a potent, cell permeable and CNS penetrant class IIa histonedeacetylase (HDAC) inhibitor with IC50s of 54 nM, 60 nM, 31 nM, 50 nM for class IIa HDAC4, HDAC5, HDAC7, HDAC9, respectively, shows >500-fold selectivity over class I HDACs (1, 2, 3) and ~150-fold selectivity over HDAC8 and the class IIb HDAC6 isoform. 了解更多
  10. ACY-775

    Catalog No. A12456
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    HDAC6 inhibitor
    ACY-775 is a potent and selective inhibitor of the of histone deacetylase 6 (HDAC6) with an IC50 of 7.5?nM. 了解更多
  11. Remetinostat

    Catalog No. A12149
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    HDAC inhibitor
    Remetinostat (SHP-141) is a hydroxamic acid-based inhibitor of histone deacetylase enzymes (HDAC) which is under development for the treatment of cutaneous T-cell lymphoma. 了解更多
  12. HDACs/mTOR Inhibitor 1

    Catalog No. A13462
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    HDACs/mTOR Inhibitor 1
    HDACs/mTOR Inhibitor 1 is a dual Histone Deacetylases (HDACs) and mammalian target of Rapamycin (mTOR) target inhibitor for treating hematologic malignancies. 了解更多
  13. Nanatinostat

    Catalog No. A21625
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    HDAC inhibitor
    Nanatinostat (CHR-3996) is a potent, class I selective and orally active histone deacetylase (HDAC) inhibitor with an IC50 of 8 nM. 了解更多
  14. HDAC-IN-5

    Catalog No. A20972
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    HDAC inhibitor
    HDAC-IN-5 is a histone deacetylase (HDAC) inhibitor. 了解更多
  15. HDAC-IN-3

    Catalog No. A20785
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    HDAC inhibitor
    HDAC-IN-3 is a histone deacetylase (HDAC) inhibitor, extracted from patent WO/2008040934 A1. 了解更多

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