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40 个项目
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CFTRinh-172
Catalog No. A12897 CFTR 抑制剂CFTRinh-172是电压无关的选择性CFTR抑制剂。在2分钟内可逆地抑制CFTR短路电流的 Ki 值为300 nM。 了解更多 -
PF 3716556
Catalog No. A11408 -
MK-7145
Catalog No. A21030 -
Leptomycin B
Catalog No. A20985 nuclear export receptor CRM1 inhibitorLeptomycin B (CI 940; LMB) is a potent inhibitor of the nuclear export of proteins. Leptomycin B inactivates CRM1/exportin 1 by covalent modification at a cysteine residue. Leptomycin B is a potent antifungal antibiotic blocking the eukaryotic cell cycle. 了解更多 -
Ralfinamide mesylate
Catalog No. A22002 Na+ channel blockerRalfinamide mesylate (FCE-26742A mesylate) is an orally available Na+ channel blocker derived from α-aminoamide, with function of suppressing pain. 了解更多 -
Barnidipine
Catalog No. A21940 L-type calcium antagonistBarnidipine (Mepirodipine) is an L-type calcium antagonist (CaA) with high affinity for [3H] initrendipine binding sites (Ki=0.21 nmol/l), has selective action against CaA receptors. 了解更多 -
Capsazepine
Catalog No. A21208 TRPV1 receptorCapsazepine is a synthetic analogue of the sensory neurone excitotoxin, and an antagonist of TRPV1 receptor with an IC50 of 562 nM. 了解更多 -
PF-4778574
Catalog No. A21157 AMPA receptor positive allosteric modulatorPF-4778574 is a potent AMPA receptor positive allosteric modulator (PAM) that has been shown to enhance cognition in animal models. 了解更多 -
Ivacaftor benzenesulfonate
Catalog No. A15132 CFTR potentiatorIvacaftor benzenesulfonate is an orally bioavailable CFTR potentiator, used for cystic fibrosis treatment. 了解更多 -
Nav1.7-IN-3
Catalog No. A13626 voltage-gated sodium channel Nav1.7 inhibitorNav1.7-IN-3 is a selective, orally bioavailable voltage-gated sodium channel Nav1.7 inhibitor with an IC50 of 8 nM. Pain relief. Limited CNS penetration. 了解更多 -
P-gp inhibitor 1
Catalog No. A13384 P-gp inhibitorP-gp inhibitor 1 is a novel inhibitor reversing P-glycoprotein-mediated multidrug resistance. 了解更多 -
TRPC6-IN-1
Catalog No. A12309 TRPC6 inhibitorTRPC6-IN-1 is a Transient Receptor Potential Canonical 6 Channel (TRPC6) inhibitor, with an EC50 of 4.66 μM. 了解更多 -
Metaflumizone
Catalog No. A18830 Sodium channel blockerMetaflumizone is a semicarbazone insecticide, acts as a potent sodium channel blocker. 了解更多 -
Dapagliflozin impurity
Catalog No. A19103 SGLT2 抑制剂Dapagliflozin impurity is an enantiomer of Dapagliflozin which is a sodium-glucose transporter 2 inhibitor. 了解更多 -
Rebeprazole sodium
Catalog No. A16147 -
Esomeprazole sodium
Catalog No. A10365 -
Azaphen dihydrochloride monohydrate
Catalog No. A15009 -
Esomeprazole Magnesium trihydrate
Catalog No. A15082 Proton pump 抑制剂Esomeprazole Magnesium trihydrate 是质子泵抑制剂，可通过抑制胃壁细胞中的H+/K+ ATPase来减少酸的分泌。 了解更多 -
Cyclopiazonic Acid
Catalog No. A14002 SERCA 抑制剂Cyclopiazonic acid是SERCA（内质网Ca2+ -ATPase）的抑制剂，可诱导细胞内储存的Ca2+释放，而不会增加IP3水平。 了解更多 -
Cyclothiazide
Catalog No. A13700 AMPA desensitization 抑制剂Cyclothiazide是苯并噻二叠氮，可作为AMPA受体的增效剂，正向调节其对谷氨酸的响应（EC50 = 3.8 M）。 了解更多 -
GSK-2193874
Catalog No. A14201 -
Oxcarbazepine
Catalog No. A13943 -
Tenatoprazole
Catalog No. A14272 -
Omeprazole
Catalog No. A10672 -
Hydralazine hydrochloride
Catalog No. A10455 Hydralazine hydrochloride是肼屈嗪的盐酸盐(安普索林)，是一种直接作用的平滑肌松弛剂，IC50为1.9 mM。 了解更多 -
TAK-438 (vonoprazan)
Catalog No. A11239 -
Azelnidipine
Catalog No. A11219 calcium channel blockerAzelnidipine是一种钙阻断剂，可减轻肝纤维化并可能增加抗氧化防御能力。可以减轻肝纤维化并可能增加抗氧化防御能力。 了解更多 -
Amiloride HCl
Catalog No. A10064 Na+ channel blockerAmiloride HCl是一种Na+通道阻滞剂，还抑制TRPP3通道和Na+/H+交换剂（NHE）。 了解更多
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- 分类
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- ATPase (4)
- CFTR (2)
- Calcium Channels (5)
- Sodium Channels (7)
- Potassium Channels (3)
- SGLT (1)
- Monocarboxylate transporters (MCT) (1)
- AMPA receptor (2)
- P-gp (2)
- CRM1 (1)
- TRP Channel (2)
- TRPV (2)
- Serotonin Transporter (1)
- Proton Pump (4)
- Na+/H+ Exchanger (2)
- Monoamine Transporter (2)
- 作用机制
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- Inhibitor (抑制剂) (21)
- Antagonist (拮抗剂) (3)
- Modulator (调节剂) (1)
- Blocker (阻断剂) (6)
- Potentiator (增强剂) (1)
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