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THIQ

Catalog No. A12860
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THIQ是一种有效的选择性黑皮质素4（MC4）受体激动剂（人MC4，MC3和MC1受体的IC50值分别为1.2、761和2067 nM）。了解更多

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MK-3697

Catalog No. A12633
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OX2 拮抗剂

MK-3697是一种高效的，口服生物利用的选择性orexin 2受体拮抗剂，Ki值为0.95nM。了解更多

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ESI-09

Catalog No. A14233
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EPAC1/EPAC2 抑制剂

ESI-09是一种直接由cAMP（EPAC）抑制剂激活的特异性交换蛋白，对于EPAC1和EPAC2，IC50为3.2 uM和1.4 uM。了解更多

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DL-AP3

Catalog No. A15378
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mGluR1 拮抗剂

DL-AP3是D-AP3和L-AP3的外消旋制剂，是磷酸丝氨酸磷酸酶的抑制剂和代谢型谷氨酸受体（mGluR）的拮抗剂，阻断了由mGluR介导的磷酸肌醇转换。了解更多

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SKI-II

Catalog No. A15988
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SphK 抑制剂

SKI-II是鞘氨醇激酶的选择性非脂质抑制剂（IC50 = 0.5 uM）。了解更多

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(1R,2S)-VU0155041

Catalog No. A21933
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partial mGluR4 agonist

(1R,2S)-VU0155041, Cis regioisomer of VU0155041, is a partial mGluR4 agonist with an EC50 of 2.35 μM. 了解更多

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MRT-83

Catalog No. A21020
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Smo antagonist

MRT-83 is a potent antagonist of Smo, with an IC50 in the nanomolar range. MRT-83 also blocks Hedgehog (Hh) signaling. 了解更多

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