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  1. Naringenin

    Catalog No. A10625
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    Naringenin是一种黄烷酮,是一种类黄酮,被认为具有抗氧化剂,自由基清除剂,消炎,碳水化合物代谢促进剂和免疫系统调节剂等对人体健康的生物活性。 了解更多
  2. Itraconazole (Sporanox)

    Catalog No. A10489
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    Itraconazole (Sporanox)是CYP3A4相对有效的抑制剂,IC50为6.1nM,用作三唑类抗真菌剂。 了解更多
  3. ABT

    Catalog No. A13361
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    Cytochrome P450 抑制剂
    ABT (1-Aminobenzotriazole)是(CYP)细胞色素P-450和氯过氧化物酶的自杀底物。 了解更多
  4. Azathramycin

    Catalog No. A15010
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    CYP3A4 抑制剂
    Azathramycin是一种抗生素。阿奇霉素与细菌核糖体的50S亚基结合,从而抑制mRNA的翻译。 了解更多
  5. Cobicistat (GS-9350)

    Catalog No. A11277
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    CYP3A 抑制剂
    Cobicistat (GS-9350)是有效,选择性的细胞色素酶P450 3A (CYP3A)抑制剂,包括重要的cyp3a4亚型。它还抑制肠道转运蛋白,增加几种hiv药物的整体吸收,包括atazanavir、darunavir和tenofovir alafenamide延胡索酸盐。 了解更多
  6. Deferasirox

    Catalog No. A10293
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    Iron chelator
    Deferasirox是一种铁螯合剂,也是细胞色素P450 3A4诱导剂,细胞色素P450 2C8抑制剂和细胞色素P450 1A2抑制剂。 了解更多
  7. Bergaptol

    Catalog No. A12303
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    CYP3A4 enzyme inhibitor
    Bergaptol is a hydroxylated psoralen that acts as a potent inhibitors of debenzylation activity of CYP3A4 enzyme with an IC50 value of 24.92 uM. Recent studies suggest that it may have antiproliferative and anticancer properties. 了解更多

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