Pim

Catalog No.Inhibitor Name Pim1Pim2Pim3Other
A10838SGI-1776 free base
***
*
*
FLT3
A11945SMI-4a
**
A14275CX-6258 HCl
***
**
**
A13203AZD1208
****
***
****
A11967TCS PIM-1 4a
**
*
A12896CX-6258
***
**
**
A15368PIM-1 Inhibitor 2
*
A15369TCS PIM-1 1
*

Notes:
1.Hover mouse over " * " to view the IC50 value.(A few compounds have proven potency but without published IC50 data.)
2.For more details about the compound, click on the product name of your interest.
3.The higher the number of " * " is, the more potent the inhibitor or activator is.
4."" refers to compounds which do inhibitory effects on the related isoform, but without specific value.

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  1. CX-6258

    Catalog No. A12896
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    Pim 抑制剂
    CX-6258是一种有效,选择性和口服有效的pan-Pim激酶抑制剂。 了解更多
  2. CX-6258 hydrochloride hydrate

    Catalog No. A15055
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    Pim 抑制剂
    CX-6258 hydrochloride hydrate是一种有效的,口服有效的Pim 1/2/3激酶(IC50 = 5 nM/25 nM/16 nM)抑制剂,具有出色的生化效能和激酶选择性。 了解更多
  3. CX-6258 HCl

    Catalog No. A14275
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    Pan-PIM kinase 抑制剂
    CX-6258 HCl是一种有效的口服泛Pim激酶抑制剂,对Pim1,Pim2和Pim3的IC50为5 nM,25 nM和16 nM。 了解更多
  4. AZD1208

    Catalog No. A13203
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    pan-Pim kinase 抑制剂
    AZD1208是PIM激酶的小分子抑制剂,具有潜在的抗肿瘤活性。 了解更多
  5. LGB-321 HCl

    Catalog No. A14420
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    Pan-PIM kinase 抑制剂
    LGB-321 HCl是一种有效且选择性的PIM激酶竞争性小分子抑制剂(Pan-PIM激酶抑制剂)。 了解更多

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