5-HT Receptors

产品 51 到 72 共 72个

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  1. Lu AE58054 (Idalopirdine)

    Catalog No. A12521
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    5-HT6R 拮抗剂
    Lu AE58054是有效的选择性5-HT6受体拮抗剂。 了解更多
  2. Blonanserin

    Catalog No. A11824
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    D2/5-HT2 receptor 拮抗剂
    Blonanserin是D2/5-HT2受体拮抗剂。 了解更多
  3. PRX-08066

    Catalog No. A13267
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    5-HT2B receptor 拮抗剂
    PRX-08066是一种新型的5-HT受体2B(5-HT2BR)拮抗剂,IC50为3.4 nM,,可减轻单芥子碱诱导的大鼠肺动脉高压和右室肥大。 了解更多
  4. Tandospirone

    Catalog No. A13293
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    5-HT Receptor 拮抗剂
    Tandospirone是5HT1A受体的部分激动剂。它以剂量依赖性方式显着降低氟哌啶醇诱导的运动迟缓。 了解更多
  5. SB-742457

    Catalog No. A14092
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    5-HT6 receptor 拮抗剂
    SB-742457是一种选择性的5-HT6受体拮抗剂,具有认知,记忆和增强学习的作用。 了解更多
  6. SB 399885 HCl

    Catalog No. A14102
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    5-HT6 拮抗剂
    SB 399885 hydrochloride是一种有效的,脑渗透剂和口服活性的SR-6拮抗剂。它对SR-6的选择性比其他血清素受体高200倍(对于人类重组,天然大鼠和天然人类SR-6受体,pKi值分别为9.11、8.81和9.02)。 了解更多
  7. Cyclobenzaprine HCl

    Catalog No. A14255
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    5-HT2 receptor 拮抗剂
    Cyclobenzaprine HCl是一种肌肉松弛剂,可阻止疼痛感。 了解更多
  8. LuAE58054

    Catalog No. A14356
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    5-HT6 receptor 拮抗剂
    LuAE58054是一种有效且选择性的5-HT6受体拮抗剂,Ki 为 0.83 nM。由伦德贝克(Lundbeck)开发,作为增强疗法,用于治疗与阿尔茨海默氏病和精神分裂症相关的认知缺陷。 了解更多
  9. Tropisetron HCL

    Catalog No. A14375
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    5-HT3 receptor 拮抗剂
    Tropisetron HCL是选择性的5-HT3受体拮抗剂和α7烟碱样受体激动剂,对5-HT3受体的IC50为70.1±0.9 nM。 了解更多
  10. NAN-190 hydrobromide

    Catalog No. A13417
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    5-HT1A receptor 拮抗剂
    NAN-190 hydrobromide是一种广泛用于科学研究的药物和研究化学品。以前认为它是一种选择性的5-HT1A受体拮抗剂,但后来的发现表明它也能有效地阻断α2肾上腺素能受体。 了解更多
  11. Clozapine N-oxide

    Catalog No. A15048
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    5-HT1C receptor 拮抗剂
    Clozapine N-oxide是氯氮平的主要代谢产物,在体外可降低SR-2A(5-HT2血清素受体)密度。 了解更多
  12. Ziprasidone

    Catalog No. A15286
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    5-HT/dopamine receptor 拮抗剂
    Ziprasidone是5-HT(5-羟色胺)和多巴胺受体拮抗剂的组合,具有抗精神病活性。 了解更多
  13. Alosetron Hydrochloride

    Catalog No. A14989
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    5HT3-receptor 拮抗剂
    Alosetron Hydrochloride是一种5-羟色胺5HT3受体拮抗剂,可用于治疗肠易激综合症。 了解更多
  14. Cyproheptadine hydrochloride

    Catalog No. A16169
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    serotonin/histamine2 拮抗剂
    Cyproheptadine hydrochloride是抗组胺药,是5-羟色胺和组胺的拮抗剂。 了解更多
  15. Azasetron HCl

    Catalog No. A16417
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    5-HT3 receptor 拮抗剂
    Azasetron HCl是一种选择性的5-HT3受体拮抗剂,IC50为0.33 nM,用于治疗癌症化学疗法引起的恶心和呕吐。 了解更多
  16. LY 334370 hydrochloride

    Catalog No. A17027
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    5-HT1F 激动剂
    LY 334370 hydrochloride是一种选择性的5-HT1F受体激动剂(Ki值为1.87、16.4,> 100 (IC50))。CAS:199673-74-0(LY 334370盐酸盐);182563-08-2(LY 334370游离碱) 了解更多
  17. Volinanserin

    Catalog No. A17115
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    5-HT2A receptor 拮抗剂
    Volananserin是高度选择性的5-HT2A受体拮抗剂。 了解更多
  18. Dolasetron

    Catalog No. A17595
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    5-HT3 receptor antagonist
    Dolasetron is a serotonin 5-HT3 receptor antagonist used to treat nausea and vomiting following chemotherapy. Its main effect is to reduce the activity of the vagus nerve, which is a nerve that activates the vomiting center in the medulla oblongata. It does not have much antiemetic effect when symptoms are due to motion sickness. 了解更多
  19. Dolasetron Mesylate

    Catalog No. A17729
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    5-HT3 receptor antagonist
    Dolasetron mesylate is a selective 5-HT3 receptor antagonist. 了解更多
  20. Alprenolol hydrochloride

    Catalog No. A17781
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    5-HT1A receptor antagonist
    Alprenolol (hydrochloride) is a non-selective beta blocker as well as 5-HT1A receptor antagonist. 了解更多
  21. Pizotifen

    Catalog No. A18107
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    5-HT receptor antagonist
    Pizotifen is a serotonin antagonist which acts mainly at the 5-HT1, 5-HT2A, and 5HT2C receptors with some antihistamine activity. 了解更多
  22. Alosetron (Hydrochloride(1:X))

    Catalog No. A11309
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    Serotonin 5HT3-receptor antagonist
    Alosetron Hydrochloride(1:X) (GR 68755 Hydrochloride(1:X)) is a Serotonin 5HT3-receptor antagonist that is used in treatment of irritable bowel syndrome. 了解更多

产品 51 到 72 共 72个

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