“leukotriene receptor”的搜索结果
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sigma-1 receptors modulator
E1R is a novel positive allosteric modulator of sigma-1 receptors.
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mGlu4 receptors modulator
VU 0364770是mGlu4受体的正变构调节剂,在表达mGlu4的HEK 293细胞中EC50值为290 nM。
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mGlu4 receptors modulator
VU 0361737是mGluR-4的选择性正变构调节剂(人和大鼠受体的EC50值分别为240和110 nM)。
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A3 adenosine receptor allosteric modulator
LUF6000 is an allosteric modulator of the human A3 adenosine receptor (AR).
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mGlu4 receptor modulator
TCN238 is a positive allosteric mGlu4 receptor modulator with an EC50 of 1 μM.
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endothelin receptor modulator
Endothelin Mordulator 1 is a endothelin receptor modulator, used for the research of endothelin-mediated disorders.
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mGlu4 receptor modulator
Lu AF21934 is a selective and brain-penetrant mGlu4 receptor positive allosteric modulator with an IC50 of 500 nM for human mGlu4.
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GLP-1R modulator
NNC0640 is a negative allosteric modulator of glucagon-like peptide-1 receptor (GLP-1R).
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GLP-1R modulator
VU0453379 is a CNS-penetrant glucagon-like peptide 1 receptor (GLP-1R) positive allosteric modulator (PAM) with an EC50 of 1.3 μM.
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mGlu5 modulator
VU0652835 is a metabotropic glutamate receptor subtype 5 (mGlu5) negative allosteric modulator with an IC50 of 81 nM.
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CXCR4 receptor modulator
NSC-23026是CXCR4受体调节剂。
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S1P1 receptor modulator
Ponesimod是一种口服活性,选择性鞘氨醇-1-磷酸受体1(S1P1)免疫调节剂,EC50为5.7 nM。
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mGlu2 receptor modulator
CBiPES HCl是mGluR-2的选择性正变构调节剂,IC50值为98.2 nM。
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5-HT3 Receptor Modulator
PU 02是5-HT3受体的负变构调节剂。
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5-HT Receptor modulator
Vortioxetine (Lu AA21004) hydrobromide是一种口服多峰血清素能药物,可抑制5-HT(1A),5-HT(1B),5-HT(3A),5-HT(7)和SERT,IC50为15 nM,33 nM,3.7 nM,19 nM和1.6 nM。
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