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Gemilukast
Catalog No. A21021 CysLT1/CysLT2 antagonistGemilukast is an orally active and potent dual cysteinyl leukotriene 1 and 2 receptors (CysLT1 and CysLT2) antagonist, with IC50s of 1.7, 25 nM for human CysLT1 and CysLT2, respectively. 了解更多 -
Minodronic acid
Catalog No. A21975 purinergic P2X2/3 receptors antagonistMinodronic acid (YM-529) is an antagonist of purinergic P2X2/3 receptors involved in pain. 了解更多 -
Barnidipine
Catalog No. A21940 L-type calcium antagonistBarnidipine (Mepirodipine) is an L-type calcium antagonist (CaA) with high affinity for [3H] initrendipine binding sites (Ki=0.21 nmol/l), has selective action against CaA receptors. 了解更多 -
Naspm trihydrochloride
Catalog No. A21437 CP-AMPA receptors antagonistNaspm trihydrochloride (1-Naphthylacetyl spermine trihydrochloride), a synthetic analogue of Joro spider toxin, is a calcium permeable AMPA (CP-AMPA) receptors antagonist. 了解更多 -
JDTic dihydrochloride
Catalog No. A11469 KOR antagonistJDTic (dihydrochloride) is a potent antagonist of kappa-opioid receptors (KOR), blocking the κ-agonist U50, 488-induced antinociception. 了解更多 -
VPC 23019
Catalog No. A20102 S1P antagonistVPC 23019, an aryl amide-containing Sphingosine 1-phosphate (S1P) analog, is a competitive antagonist at the S1P1 and S1P3 receptors (pKi= 7.86 and 5.93, respectively) and an agonist at the S1P4 and S1P5 receptors (pEC50= 6.58 and 7.07, respectively). 了解更多 -
Urapidil
Catalog No. A17074 -
Proxyphylline
Catalog No. A16821 A1 adenosine receptors 拮抗剂Proxyphylline是茶碱的衍生物，由于其心血管特性而被用作支气管扩张剂。它与A2腺苷受体（对于血小板，Ki = 850μM）选择性拮抗A1腺苷受体（对于牛脑，Ki = 82 nM）。 了解更多 -
Acebutolol HCl
Catalog No. A16387 -
Ketanserin tartrate
Catalog No. A13664 5HT2A 拮抗剂Ketanserin tartrate是一种选择性的5-HT receptor拮抗剂。Ketanserin tartrate 也抑制 hERG 电流 (IhERG)，IC50 为 0.11 μM。 了解更多 -
Labetalol HCl
Catalog No. A14239 alpha1/beta adrenergic receptors 拮抗剂Labetalol HCl是选择性α1-肾上腺素能受体和非选择性β-肾上腺素能受体的双重拮抗剂。 了解更多 -
NVP-AAM077 Tetrasodium Hydrate (PEAQX)
Catalog No. A14071 -
CVT 6883
Catalog No. A13745 -
2-Hydroxysaclofen
Catalog No. A13696 -
LY 255283
Catalog No. A13090 -
Ondansetron HCl (GR 38032F)
Catalog No. A10674 5-HT Receptors 拮抗剂Ondansetron HCl (GR 38032F)是5-羟色胺5-HT3受体拮抗剂，主要用作止吐药，通常在化疗后用于治疗恶心和呕吐。 了解更多 -
A2A receptor antagonist 1
Catalog No. A12567 adenosine A2A/A1 receptor antagonistA2A receptor antagonist 1 (CPI-444 analog) is an antagonist of both adenosine A2A receptor and A1 receptor with Kis of 4 and 264 nM, respectively. 了解更多 -
Sigma-1 receptor antagonist 2
Catalog No. A18504 sigma 1 receptor antagonistSigma-1 receptor antagonist 2 is a potent and selective sigma 1 receptor (??1 R) antagonist with Kis of 3.88 and 1288 nM for ??1 and ??2 receptor, respectively. 了解更多 -
Glucagon receptor antagonists-1
Catalog No. A11428 glucagon receptor antagonistGlucagon receptor antagonists-1 is a highly potent glucagon receptor antagonist. 了解更多 -
Sigma-1 receptor antagonist 3
Catalog No. A18501 Sigma-1 receptor antagonistSigma-1 receptor antagonist 3 (compound135) is a potent and selective Sigma-1 (??1) receptor antagonist with a Ki of 1.14 nM. 了解更多 -
Glucagon receptor antagonists-3
Catalog No. A11430 Glucagon receptor antagonistGlucagon receptor antagonists-3 is a highly potent glucagon receptor antagonist. 了解更多 -
Glucagon receptor antagonists-2
Catalog No. A11429 Glucagon receptor antagonistGlucagon receptor antagonists-2 is a highly potent glucagon receptor antagonist. 了解更多 -
Calcium-Sensing Receptor Antagonists I
Catalog No. A15034 Calcium-Sensing Receptor 拮抗剂Calcium-Sensing Receptor Antagonists I 是钙敏感甲状旁腺激素受体的拮抗剂。 了解更多 -
Tonapofylline
Catalog No. A21328 adenosine A1 receptor antagonistTonapofylline (BG 9928) is an orally active and selective adenosine A1 receptor antagonist with a Ki of 7.4 nM for human adenosine A1 receptor (hA1), which displays 915-fold selectivity versus human adenosine A2A receptor and 12-fold selectivity versus human adenosine A2B receptor and is used in development for the treatment of heart failure. 了解更多 -
NRA-0160
Catalog No. A20128 Dopamine D4 receptor antagonistNRA-0160 is a selective dopamine D4 receptor antagonist, with a Ki value of 0.48 nM and with negligible affinity for dopamine D2 receptor (Ki: >10000 nM), D3 receptor (Ki: 39 nM), rat 5-HT2A receptor (Ki: 180 nM) and rat α1 adrenoceptor (Ki: 237 nM). 了解更多 -
CJ-42794
Catalog No. A21948 EP4 antagonistCJ-42794 is a selective prostaglandin E receptor subtype 4 (EP4) antagonist, inhibits [3H]-PGE2 binding to the human EP4 receptor with a mean pKi of 8.5, a binding affinity that was at least 200-fold more selective for the human EP4 receptor than other human EP receptor subtypes (EP1, EP2, and EP3). 了解更多 -
Risperidone hydrochloride
Catalog No. A21458 dopamine D2 receptor antagonistRisperidone hydrochloride is a serotonin 5-HT2 receptor blocker and a potent dopamine D2 receptor antagonist, with Kis of 0.16, 1.4 nM for 5-HT2 and D2 receptor, respectively. 了解更多 -
L-371,257
Catalog No. A21219 oxytocin receptor antagonistL-371,257 is an orally bioavailable, non-blood-brain barrier penetrant, selective and competitive antagonist of oxytocin receptor (pA2=8.4) with high affinity at both the oxytocin receptor (Ki=19 nM) and vasopressin V1a receptor (Ki=3.7 nM). 了解更多 -
Pipamperone
Catalog No. A12621 D2 receptor antagonistPipamperone (Floropipamide; McN-JR 3345; R 3345) is a high-affinity antagonist of 5-HT2A receptor (pKi=8.2) and D4 receptor (pKi=8.0) and a low-affinity antagonist of D2 receptor (pKi=6.7). 了解更多 -
Nemorexant
Catalog No. A12685 Orexin receptor antagonistNemorexant (ACT-541468) is a potent orexin receptor antagonist extracted from patent WO2015083094A1, compound example 7, has IC50s of 2 nM and 3 nM for Ox1 receptor and Ox2 receptor, respectively. 了解更多 -
JNJ-54175446
Catalog No. A18675 P2X7 receptor antagonistJNJ-54175446 is a potent and selective brain penetrant P2X7 receptor antagonist, with pIC50s of 8.46 and 8.81 for hP2X7 receptor and rP2X7 receptor, respectively. 了解更多 -
Seratrodast
Catalog No. A18134 thromboxane A2 (TXA2) receptor (TP receptor) antagonistSeratrodast is a thromboxane A2 (TXA2) receptor (TP receptor) antagonist used primarily in the treatment of asthma. 了解更多 -
AZD9496 maleate
Catalog No. A21726 estrogen receptor (ERα) antagonistAZD9496 maleate is a potent and selective estrogen receptor (ERα) antagonist with IC50 of 0.28 nM. AZD9496 maleate is an orally bioavailable selective oestrogen receptor degrader (SERD). 了解更多 -
Tarafenacin D-tartrate
Catalog No. A21477 M3 muscarinic receptor antagonistTarafenacin D-tartrate (SVT-40776 D-tartrate) is a highly selective M3 muscarinic receptor antagonist (Ki= 0.19 nM), ~200 fold selectivity over M2 receptor. 了解更多 -
JNJ-37822681 dihydrochloride
Catalog No. A21470 dopamine D2 receptor antagonistJNJ-37822681 dihydrochloride is a potent, specific, centrally active, fast-dissociating dopamine D2 receptor antagonist with a moderate binding affinity for the dopamine D2L receptor (Ki =158 nM), which has potential for the treatment of schizophrenia and bipolar disorder. 了解更多 -
Risperidone mesylate
Catalog No. A21463 dopamine D2 receptor antagonistRisperidone mesylate(R 64 766 mesylate) is a serotonin 5-HT2 receptor blocker(Ki= 0.16 nM) and a potent dopamine D2 receptor antagonist(Ki= 1.4 nM). 了解更多 -
Masupirdine mesylate
Catalog No. A21409 5-HT6 receptor antagonistMasupirdine mesylate (SUVN-502 mesylate) is a potent, selective, orally bioavailable, and brain penetrant 5-HT6 receptor antagonist (Ki of 2.04 nM for human 5-HT6 receptor). 了解更多 -
Zonampanel
Catalog No. A21199 glutamate receptor subtype antagonistZonampanel (YM 872) is a selective antagonist of the glutamate receptor subtype, α-amino-3-hydroxy-5-methylisoxazole-4-propionic acid (AMPA) receptor. 了解更多 -
Toreforant
Catalog No. A21058 histamine H4 receptor (H4R) antagonistToreforant is a potent and selective histamine H4 receptor (H4R) antagonist, with a Ki at the human receptor of 8.4 nM. 了解更多 -
Pexacerfont
Catalog No. A14105 CRF1 receptor antagonistPexacerfont is a selective corticotropin-releasing factor (CRF1) receptor antagonist with IC50 of 6.1??0.6 nM for human CRF1 receptor. 了解更多 -
LY-2940094
Catalog No. A19125 NOP receptor antagonistLY-2940094 is a potent, selective and orally available nociceptin receptor (NOP receptor) antagonist with high affinity (Ki=0.105 nM) and antagonist potency (Kb=0.166 nM). LY-2940094 reduces ethanol self-administration in animal models. 了解更多 -
Fimasartan
Catalog No. A17477 non-peptide angiotensin II receptor antagonistFimasartan is a non-peptide angiotensin II receptor antagonist (ARB) used for the treatment of hypertension and heart failure. Through oral administration, fimasartan blocks angiotensin II receptor type 1 (AT1 receptors), reducing pro-hypertensive actions of angiotensin II, such as systemic vasoconstriction and water retention by the kidneys. 了解更多 -
Decloxizine
Catalog No. A20964 histamine 1 receptor antagonistDecloxizine(UCB-1402; NSC289116) is a histamine 1 receptor antagonist. 了解更多 -
GSK189254A
Catalog No. A22005 histamine H3 receptor antagonistGSK189254A (GSK189254) is a novel, potent and selective histamine H3 receptor antagonist with pKi values of 9.59-9.90 and 8.51-9.17 for human and rat H3, respectively. 了解更多 -
Amisulpride hydrochloride
Catalog No. A21994 dopamine D2/D3 receptor antagonistAmisulpride hydrochloride is a dopamine D2/D3 receptor antagonist with Kis of 2.8 and 3.2 nM for human dopamine D2 and D3, respectively. 了解更多
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