“angiotensin receptors”的搜索结果

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  1. BRL 52537 HCl

    Catalog No. A11210
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    Opioid Receptors 激动剂
    BRL 52537 hydrochloride是一种高度选择性和有效的κ阿片类激动剂(Ki = 0.24 nM)。比吗啡强25倍。 了解更多
  2. BRL 37344 Na Salt

    Catalog No. A13676
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    β3-adrenergic receptors 激动剂
    BRL 37344 Na Salt是具有脂解活性的β3-AR(β3-肾上腺素能受体)选择性激动剂。 了解更多
  3. Cimaterol

    Catalog No. A13401
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    β-adrenergic receptors 激动剂
    Cimaterol是β的有效激动剂;肾上腺素能受体(人β的pEC50 = 8.13、8.78和6.62;1β,2β和3β)。 了解更多
  4. CP-809101

    Catalog No. A12481
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    5-HT2C receptor agonist
    CP-809101 is a potent and selective 5-HT2C receptor agonist with pEC50 of 9.96/7.19/6.81 for human 5-HT2C/5-HT2B/5-HT2A receptors respectively. 了解更多
  5. AB-MECA

    Catalog No. A12189
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    A3 adenosine receptor agonist
    AB-MECA is a high affinity A3 adenosine receptor agonist, has high affinity for recombinant A1 and A3 receptors. 了解更多
  6. L-APB

    Catalog No. A21872
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    mGluRs M3 agonist
    L-APB is a potent and specific agonist for the group III mGluRs, with EC50s of 0.13, 0.29, 1.0, 249 μM for mGlu4, mGlu8, mGlu6 and mGlu7 receptors, respectively. 了解更多
  7. Eglumegad

    Catalog No. A21005
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    group II (mGlu2/3) receptor agonist
    Eglumegad (LY354740) is a highly potent and selective group II (mGlu2/3) receptor agonist with IC50s of 5 and 24 nM on transfected human mGlu2 and mGlu3 receptors, respectively. 了解更多
  8. Cariprazine

    Catalog No. A21202
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    D3 receptor and D2 receptor partial agonist
    Cariprazine is a novel antipsychotic drug candidate that exhibits high affinity for the D3 (Ki=0.085 nM) and D2 (Ki=0.49 nM) receptors, and moderate affinity for the 5-HT1A receptor (Ki=2.6 nM). 了解更多
  9. Donitriptan

    Catalog No. A13145
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    5-HT1B/1D receptors agonist
    Donitriptan is a potent, high efficacy agonist at 5-HT1B/1D receptors with pKis of 9.4 and 9.3, respectively. 了解更多
  10. Carbetocin

    Catalog No. A18080
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    peripheral oxytocin receptors agonist
    Carbetocin (Lonactene; Duratocin) is an obstetric drug used to control postpartum hemorrhage and bleeding after giving birth; an agonist at peripheral oxytocin receptors. 了解更多
  11. RU 24969

    Catalog No. A20857
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    5-HT1A/5-HT1B receptors agonist
    RU 24969 is a selective agonist at the 5-HT1A and 5-HT1B receptors. 了解更多
  12. O-Phospho-L-serine

    Catalog No. A21159
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    group III mGluR receptors agonist
    O-Phospho-L-serine is the immediate precursor to L-serine in the serine synthesis pathway, and an agonist at the group III mGluR receptors (mGluR4, mGluR6, mGluR7, and mGluR8); O-Phospho-L-serine also acts as a weak antagonist for mGluR1 and a potent antagonist for mGluR2. 了解更多
  13. DPI-3290

    Catalog No. A13699
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    opioid receptors agonist
    DPI-3290 (Org 41793) is a potent and specific opioid receptors agonist with Ki values of 0.18 nM, 0.46 nM, and 0.62 nM for δ-, μ-, and κ-opioid receptors, respectively. 了解更多
  14. PSN632408

    Catalog No. A20902
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    GPR119 receptors agonist
    PSN632408 is an optimized agonist of GPR119 receptors that shows similar potency to OEA at both recombinant mouse and human GPR119 receptors, exhibiting EC50 values of 5.6 and 7.9 uM, respectively. 了解更多

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