“jwh 250”的搜索结果

24 个项目

每页

设置降序顺序
  1. Cariprazine

    Catalog No. A21202
    Quick View
    D3 receptor and D2 receptor partial agonist
    Cariprazine is a novel antipsychotic drug candidate that exhibits high affinity for the D3 (Ki=0.085 nM) and D2 (Ki=0.49 nM) receptors, and moderate affinity for the 5-HT1A receptor (Ki=2.6 nM). 了解更多
  2. Taranabant ((1R,2R)stereoisomer)

    Catalog No. A21705
    Quick View
    CB1 receptor inverse agonist
    Taranabant (1R,2R)stereoisomer is the R-enantiomer of Taranabant. Taranabant is a highly potent and selective cannabinoid 1 (CB1) receptor inverse agonist. 了解更多
  3. (1R,2R)-2-PCCA(hydrochloride)

    Catalog No. A21655
    Quick View
    GPR88 receptor agonist
    (1R,2R)-2-PCCA hydrochloride is a diastereomer of 2-PCCA, and acts as a potent GPR88 receptor agonist, with an EC50 of 3 nM in cell-free assay, and 603 nM in cell assay. 了解更多
  4. LY2812223

    Catalog No. A21100
    Quick View
    mGlu2 receptor agonist
    LY2812223 is a highly potent, functionally selective mGlu2 receptor agonist with mGlu2 binding affinity for mGlu2 and mGlu3 (Ki=144 nM and 156 nM, respectively). 了解更多
  5. Lesopitron dihydrochloride

    Catalog No. A12950
    Quick View
    5-HT1A receptor agonist
    Lesopitron dihydrochloride is a full and selective 5-HT1A receptor agonist with IC50 of 125 nM in rat hippocampal membranes. 了解更多
  6. Tasimelteon

    Catalog No. A17351
    Quick View
    MT1 and MT2 receptor agonist
    Tasimelteon is a melatonin MT1 and MT2 receptor agonist. 了解更多
  7. Albiglutide

    Catalog No. A16823
    Quick View
    GLP-1 激动剂
    Albiglutide是一种胰高血糖素样肽1激动剂(GLP-1激动剂)。 了解更多
  8. LY2979165

    Catalog No. A11487
    Quick View
    mGlu2 激动剂
    LY2979165是mglu2激动剂。 了解更多
  9. S 32212 HCl

    Catalog No. A13501
    Quick View
    5-HT2C 激动剂
    S 32212 HCl是5-HT2C受体的反向激动剂(人5-HT2C INI受体的pKi = 8.18)。 了解更多
  10. Ibotenic Acid

    Catalog No. A14006
    Quick View
    NMDA& mGlu receptor 激动剂
    Ibotenic Acid是最初从鹅膏菌属物种中分离出来的一种神经兴奋性氨基酸,它起着NMDA和代谢型谷氨酸受体激动剂的作用。 了解更多
  11. Linaclotide

    Catalog No. A13834
    Quick View
    Guanylate cyclase C 激动剂
    Linaclotide是鸟苷酸环化酶2C的肽激动剂。 了解更多
  12. CYM 5442 HCl

    Catalog No. A13637
    Quick View
    EDG-1 (S1P1) 激动剂
    CYM 5442 HCl是一种有效的体外选择性EDG-1(S1P1)激动剂(EC50 = 1.35 nM)。 了解更多
  13. Immethridine hydrobromide

    Catalog No. A13641
    Quick View
    histamine H3 receptor 激动剂
    Immethridine hydrobromide是一种强而高选择性的组胺H3受体激动剂(pEC50 = 9.74),其选择性是H4受体的300倍(pKi值分别为9.07和6.61)。 了解更多
  14. lorcaserin hydrochloride (APD-356)

    Catalog No. A12598
    Quick View
    serotonin 2C receptor 激动剂
    lorcaserin hydrochloride (APD-356)是血清素2C受体激动剂,可指示与减少热量饮食和增加体育锻炼以减轻慢性体重成人管理。 了解更多
  15. Arformoterol tartrate

    Catalog No. A12795
    Quick View
    beta2-adrenergic 激动剂
    Arformoterol tartrate是β2-肾上腺素能激动剂。 了解更多
  16. WIN 55,212-2 mesylate

    Catalog No. A11932
    Quick View
    CB receptor 激动剂
    WIN 55,212-2 mesylate是一种有效的cannabinoid receptor激动剂,在神经性疼痛的大鼠模型中具有有效的镇痛作用。它通过受体介导的信号激活p42和p44 MAP激酶。 了解更多
  17. Moxonidine HCl

    Catalog No. A11741
    Quick View
    imidazoline receptor 1 激动剂
    Moxonidine HCl是咪唑啉受体亚型1(I1)的选择性激动剂。Moxonidine引起交感神经系统活动的减少,因此导致血压的降低。 了解更多
  18. Synephrine (Oxedrine)

    Catalog No. A10882
    Quick View
    Adrenergic Receptor 激动剂
    Synephrine (Oxedrine)是一种通常用于减肥的胺化合物。 了解更多
  19. Buspirone HCl

    Catalog No. A15687
    Quick View
    5HT(1A) receptor 激动剂
    Buspirone hydrochloride是一种具有5-D(2)多巴胺能作用的血清素能(5HT(1A)受体激动剂)抗焦虑药,用于焦虑症。 了解更多
  20. Nalmefene hydrochloride

    Catalog No. A13843
    Quick View
    dopamine receptor 激动剂
    Nalmefene hydrochloride是opioid receptor拮抗剂。 了解更多
  21. Oxymetazoline hydrochloride

    Catalog No. A10686
    Quick View
    alpha-1 adrenergic 激动剂
    Oxymetazoline是一种选择性的α-1激动剂和部分α-2激动剂局部减充血剂,以盐酸羟甲唑啉的形式使用。 了解更多
  22. Adrenalone HCl

    Catalog No. A11807
    Quick View
    adrenergic 激动剂
    Adrenalone HCl是一种肾上腺素能激动剂,用作局部血管收缩药和止血药,主要作用于α-1肾上腺素能受体。 了解更多
  23. Carvedilol

    Catalog No. A11843
    Quick View
    β2-adrenergic receptor
    Carvedilol是具有抗氧化特性的β1和β2肾上腺素能受体(AR)激动剂。 了解更多
  24. Aripiprazole (Abilify)

    Catalog No. A11801
    Quick View
    5-HT1A receptor 激动剂
    Aripiprazole (Abilify)是人5-HT1A受体部分激动剂,Ki为4.2 nM。 了解更多

24 个项目

每页

设置降序顺序
Rewards