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  1. Cariprazine
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    Cariprazine

    Catalog No. A21202
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    D3 receptor and D2 receptor partial agonist
    Cariprazine is a novel antipsychotic drug candidate that exhibits high affinity for the D3 (Ki=0.085 nM) and D2 (Ki=0.49 nM) receptors, and moderate affinity for the 5-HT1A receptor (Ki=2.6 nM). 了解更多
  2. Goserelin
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    Goserelin

    Catalog No. A21197
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    GnRH agonist
    Goserelin(ICI 118630) is an injectable gonadotropin releasing hormone superagonist (GnRH agonist). 了解更多
  3. GV-58
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    GV-58

    Catalog No. A21966
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    N- and P/Q-type Ca2+ channels agonist
    GV-58 is a potent, selective N- and P/Q-type Ca2+ channels agonist with EC50 of 7.21/8.81 uM for N-type/P-Q-type Ca2+ channel; 20-fold less potent CDK inhibitor activity. 了解更多
  4. Taranabant ((1R,2R)stereoisomer)
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    Taranabant ((1R,2R)stereoisomer)

    Catalog No. A21705
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    CB1 receptor inverse agonist
    Taranabant (1R,2R)stereoisomer is the R-enantiomer of Taranabant. Taranabant is a highly potent and selective cannabinoid 1 (CB1) receptor inverse agonist. 了解更多
  5. (1R,2R)-2-PCCA(hydrochloride)
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    (1R,2R)-2-PCCA(hydrochloride)

    Catalog No. A21655
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    GPR88 receptor agonist
    (1R,2R)-2-PCCA hydrochloride is a diastereomer of 2-PCCA, and acts as a potent GPR88 receptor agonist, with an EC50 of 3 nM in cell-free assay, and 603 nM in cell assay. 了解更多
  6. LY2812223
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    LY2812223

    Catalog No. A21100
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    mGlu2 receptor agonist
    LY2812223 is a highly potent, functionally selective mGlu2 receptor agonist with mGlu2 binding affinity for mGlu2 and mGlu3 (Ki=144 nM and 156 nM, respectively). 了解更多
  7. Lesopitron dihydrochloride
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    Lesopitron dihydrochloride

    Catalog No. A12950
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    5-HT1A receptor agonist
    Lesopitron dihydrochloride is a full and selective 5-HT1A receptor agonist with IC50 of 125 nM in rat hippocampal membranes. 了解更多
  8. BW 245C
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    BW 245C

    Catalog No. A13494
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    prostanoid DP-receptor (DP1) agonist
    BW 245C is a prostanoid DP-receptor (DP1) agonist, used to treat stroke. 了解更多
  9. GSK5182
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    GSK5182

    Catalog No. A19383
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    ERRγ agonist
    GSK5182 is a highly selective inverse agonist of estrogen-related receptor γ (ERRγ) with an IC50 of 79 nM and does not interact with other nuclear receptors, including ERRα or ERα. 了解更多
  10. Taltirelin
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    Taltirelin

    Catalog No. A18250
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    TRH-R agonist
    Taltirelin (TA0910) is a superagonist at thyrotropin-releasing hormone receptor (TRH-R) with an IC50 of 910 nM and EC50 of 36 nM for stimulating an increase in cytosolic Ca2+ concentration (Ca2+ release). 了解更多
  11. Tasimelteon
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    Tasimelteon

    Catalog No. A17351
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    MT1 and MT2 receptor agonist
    Tasimelteon is a melatonin MT1 and MT2 receptor agonist. 了解更多
  12. GSK4112
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    GSK4112

    Catalog No. A17135
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    Rev-Erbα 激动剂
    GSK4112是选择性的Rev-erbα激动剂,EC50值为250 nM。GSK4112是小分子化学探针, 用于核血红素受体REV-erbα的细胞生物学研究。 了解更多
  13. SR9238
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    SR9238

    Catalog No. A15763
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    LXR Inverse 激动剂
    SR9238是有效的选择性LXR反向激动剂（LXRβ和LXRα的IC50值分别为43和214 nM）。 了解更多
  14. Albiglutide
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    Albiglutide

    Catalog No. A16823
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    GLP-1 激动剂
    Albiglutide是一种胰高血糖素样肽1激动剂（GLP-1激动剂）。 了解更多
  15. LY2979165
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    LY2979165

    Catalog No. A11487
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    mGlu2 激动剂
    LY2979165是mglu2激动剂。 了解更多
  16. Resiquimod
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    Resiquimod

    Catalog No. A15890
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    TLR7/8 激动剂
    Resiquimod是一种免疫应答调节剂，可作为有效的TLR 7/8激动剂。阶段2。 了解更多
  17. TBPB
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    TBPB

    Catalog No. A14205
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    M1 mAChR 激动剂
    TBPB是一种变构M1 mAChR激动剂，EC50值为89 nM，可调节淀粉样蛋白加工并在大鼠中产生类抗精神病药活性。 了解更多
  18. SR9243
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    SR9243

    Catalog No. A15535
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    LXR 激动剂
    SR9243是有效的选择性LXR反向激动剂。SR9243通过抑制脂质产生和Warburg效应杀死癌细胞。它在多种类型的癌症中诱导细胞死亡，并且不会引起副作用，而这些副作用已使先前针对这些过程的尝试脱轨。 了解更多
  19. Muscimol hydrobromide
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    Muscimol hydrobromide

    Catalog No. A13459
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    GABA(A) receptor 激动剂
    Muscimol hydrobromide是抗抑郁药氟西汀的活性代谢产物，可抑制5-羟色胺的摄取，pKi值为7.35.1。诺氟西汀的S-对映体的5-羟色胺再摄取阻断效能比R-对映体高20倍（分别为pKis = 7.86与6.51）。 了解更多
  20. S 32212 HCl
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    S 32212 HCl

    Catalog No. A13501
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    5-HT2C 激动剂
    S 32212 HCl是5-HT2C受体的反向激动剂（人5-HT2C INI受体的pKi = 8.18）。 了解更多
  21. Ibotenic Acid
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    Ibotenic Acid

    Catalog No. A14006
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    NMDA& mGlu receptor 激动剂
    Ibotenic Acid是最初从鹅膏菌属物种中分离出来的一种神经兴奋性氨基酸，它起着NMDA和代谢型谷氨酸受体激动剂的作用。 了解更多
  22. Linaclotide
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    Linaclotide

    Catalog No. A13834
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    Guanylate cyclase C 激动剂
    Linaclotide是鸟苷酸环化酶2C的肽激动剂。 了解更多
  23. A-582941
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    A-582941

    Catalog No. A13539
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    α7 nAChR 激动剂
    A-582941是选择性的AChR a7部分激动剂。它对大鼠和人类a7受体均表现出高亲和力（Ki值分别为10.8和16.7 nM）。 了解更多
  24. CYM 5442 HCl
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    CYM 5442 HCl

    Catalog No. A13637
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    EDG-1 (S1P1) 激动剂
    CYM 5442 HCl是一种有效的体外选择性EDG-1（S1P1）激动剂（EC50 = 1.35 nM）。 了解更多
  25. Immethridine hydrobromide
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    Immethridine hydrobromide

    Catalog No. A13641
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    histamine H3 receptor 激动剂
    Immethridine hydrobromide是一种强而高选择性的组胺H3受体激动剂（pEC50 = 9.74），其选择性是H4受体的300倍（pKi值分别为9.07和6.61）。 了解更多
  26. AC-42
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    AC-42

    Catalog No. A13855
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    AC 42是一种变构激动剂。 了解更多
  27. APD668
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    APD668

    Catalog No. A14342
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    GPR119 激动剂
    APD668是有效的GPR119激动剂，hGPR119和ratGPR119的EC50分别为2.7 nM和33 nM。 了解更多
  28. AR-231453
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    AR-231453

    Catalog No. A13716
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    GPR119 激动剂
    AR-231453是GPR119的一种有效的，选择性的小分子药物，可增强葡萄糖依赖性胰岛素分泌和胰高血糖素样肽1（GLP-1）的释放。 了解更多
  29. MBX-2982
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    MBX-2982

    Catalog No. A12634
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    GPR119 激动剂
    MBX-2982是针对2型糖尿病的潜在一流疗法，其靶向G蛋白偶联受体119（GPR119），该受体与已知刺激葡萄糖依赖性胰岛素分泌的生物活性脂质相互作用。 了解更多
  30. lorcaserin hydrochloride (APD-356)
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    lorcaserin hydrochloride (APD-356)

    Catalog No. A12598
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    serotonin 2C receptor 激动剂
    lorcaserin hydrochloride (APD-356)是血清素2C受体激动剂，可指示与减少热量饮食和增加体育锻炼以减轻慢性体重成人管理。 了解更多
  31. Arformoterol tartrate
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    Arformoterol tartrate

    Catalog No. A12795
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    beta2-adrenergic 激动剂
    Arformoterol tartrate是β2-肾上腺素能激动剂。 了解更多
  32. WIN 55,212-2 mesylate
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    WIN 55,212-2 mesylate

    Catalog No. A11932
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    CB receptor 激动剂
    WIN 55,212-2 mesylate是一种有效的cannabinoid receptor激动剂，在神经性疼痛的大鼠模型中具有有效的镇痛作用。它通过受体介导的信号激活p42和p44 MAP激酶。 了解更多
  33. Moxonidine HCl
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    Moxonidine HCl

    Catalog No. A11741
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    imidazoline receptor 1 激动剂
    Moxonidine HCl是咪唑啉受体亚型1（I1）的选择性激动剂。Moxonidine引起交感神经系统活动的减少，因此导致血压的降低。 了解更多
  34. PNU 282987
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    PNU 282987

    Catalog No. A11233
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    α7 nAChR 激动剂
    PNU 282987 (PNU-282,987)可作为神经烟碱乙酰胆碱受体α7亚型的有效选择性激动剂。 了解更多
  35. GW4064
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    GW4064

    Catalog No. A11141
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    FXR 激动剂
    GW4064是选择性的非甾体类法尼醇X受体（FXR）激动剂（EC50 = 15 nM）。 了解更多
  36. Synephrine (Oxedrine)
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    Synephrine (Oxedrine)

    Catalog No. A10882
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    Adrenergic Receptor 激动剂
    Synephrine (Oxedrine)是一种通常用于减肥的胺化合物。 了解更多
  37. Beclometasone dipropionate
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    Beclometasone dipropionate

    Catalog No. A17254
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    glucocorticoid agonist
    Beclometasone dipropionate is a potent glucocorticoid agonist; it is a prodrug of the free form, beclometasone. 了解更多
  38. Clofibric Acid
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    Clofibric Acid

    Catalog No. A16463
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    PPARα 激动剂
    Clofibric Acid是PPARα激动剂和降血脂药。 了解更多
  39. Buspirone HCl
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    Buspirone HCl

    Catalog No. A15687
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    5HT(1A) receptor 激动剂
    Buspirone hydrochloride是一种具有5-D（2）多巴胺能作用的血清素能（5HT（1A）受体激动剂）抗焦虑药，用于焦虑症。 了解更多
  40. GTS-21 (DMBX-A)
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    GTS-21 (DMBX-A)

    Catalog No. A15950
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    nAChR 激动剂
    GTS-21 dihydrochloride (DMBX-A)是一种选择性的α7烟碱乙酰胆碱受体激动剂，最近已被确定为一种有希望的炎症治疗方法。 了解更多
  41. Nalmefene hydrochloride
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    Nalmefene hydrochloride

    Catalog No. A13843
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    dopamine receptor 激动剂
    Nalmefene hydrochloride是opioid receptor拮抗剂。 了解更多
  42. Diphenyleneiodonium chloride
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    Diphenyleneiodonium chloride

    Catalog No. A13359
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    GPR3 激动剂/NOS/ NADPH oxidases 抑制剂
    Diphenyleneiodonium是一种有效的不可逆的巨噬细胞抑制剂NOS2（iNOS）和内皮细胞NOS3（eNOS）抑制剂。 了解更多
  43. Oxymetazoline hydrochloride
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    Oxymetazoline hydrochloride

    Catalog No. A10686
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    alpha-1 adrenergic 激动剂
    Oxymetazoline是一种选择性的α-1激动剂和部分α-2激动剂局部减充血剂，以盐酸羟甲唑啉的形式使用。 了解更多
  44. NMDA
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    NMDA

    Catalog No. A12751
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    NMDA receptor 激动剂
    NMDA是一种原型NMDA受体激动剂。 了解更多
  45. Adrenalone HCl
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    Adrenalone HCl

    Catalog No. A11807
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    adrenergic 激动剂
    Adrenalone HCl是一种肾上腺素能激动剂，用作局部血管收缩药和止血药，主要作用于α-1肾上腺素能受体。 了解更多
  46. Carvedilol
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    Carvedilol

    Catalog No. A11843
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    β2-adrenergic receptor
    Carvedilol是具有抗氧化特性的β1和β2肾上腺素能受体（AR）激动剂。 了解更多
  47. Prednisone (Adasone)
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    Prednisone (Adasone)

    Catalog No. A10752
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    Glucocorticoid Receptor 激动剂
    Prednisone (Adasone)可降低粘膜TNF-a的产生，肠道通透性和NF-kB表达水平。 了解更多
  48. Aripiprazole (Abilify)
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    Aripiprazole (Abilify)

    Catalog No. A11801
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    5-HT1A receptor 激动剂
    Aripiprazole (Abilify)是人5-HT1A受体部分激动剂，Ki为4.2 nM。 了解更多
  49. pirinixic acid (WY 14643)
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    pirinixic acid (WY 14643)

    Catalog No. A12360
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    PPARα 激动剂
    pirinixic acid (WY 14643)是一种高效pparα激动剂。 了解更多
  50. Imiquimod (Aldara)
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    Imiquimod (Aldara)

    Catalog No. A10469
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    TLR7 激动剂
    Imiquimod (Aldara)是一种杂环咪唑并喹啉酰胺，用作免疫反应调节剂。 了解更多

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