“Lurasidone HCl”的搜索结果

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  1. Lurasidone (SM13496)

    Catalog No. A11214
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    Dopamine D2 抑制剂
    Lurasidone (SM-13496)是dopamine D2和5-HT7的拮抗剂,IC50 值分别为 1.68 和 0.495 nM。Lurasidone (SM-13496) 也是 5-HT1A 受体的部分激动剂。 了解更多
  2. Fexofenadine HCl

    Catalog No. A11859
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    COX 抑制剂/histamine H1 receptor 激动剂
    Fexofenadine Hydrochloride是一种抗组胺药,可抑制Cox-1,Cox-2,并且是组胺H1受体激动剂,IC50为246 nM。 了解更多
  3. Edivoxetine HCl

    Catalog No. A13865
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    norepinephrine reuptake 抑制剂
    Edivoxetine HCl是一种选择性去甲肾上腺素再摄取抑制剂。 了解更多
  4. Antazoline HCl

    Catalog No. A16411
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    Histamine H1 receptor 抑制剂
    Antazoline HCl是第一代抗组胺药,可与组胺H1受体结合并阻断内源性组胺的作用。 了解更多
  5. Atomoxetine HCl

    Catalog No. A13424
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    norepinephrine (NE) transporter 抑制剂
    Atomoxetine HCl是SLC6A2的一种竞争性特异性抑制剂,同时在大鼠下丘脑突触体中显示出微弱的ST和DAT抑制作用。 了解更多
  6. Levomilnacipran HCl

    Catalog No. A14391
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    serotonin/NE reuptake 抑制剂
    Levomilnacipran HCl是一种选择性的5-羟色胺和去甲肾上腺素再摄取抑制剂。 了解更多
  7. GBR-12935 2HCl

    Catalog No. A11937
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    DAT and SLC6A2 抑制剂
    GBR-12935 dihydrochloride是一种有效的选择性多巴胺再摄取抑制剂。 了解更多
  8. Vanoxerine 2HCl (GBR-12909)

    Catalog No. A10725
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    dopamine re-uptake 抑制剂
    Vanoxerine 2HCl (GBR-12909)是哌嗪衍生物,是一种有效的、选择性的多巴胺摄取(dopamine uptake)抑制剂。 了解更多
  9. Nefazodone hydrochloride

    Catalog No. A17622
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    5-HT2 receptors inhibitor
    Nefazodone HCl is an inhibitor of 5-HT2 receptors, SERT, NET, and hERG K+ channels used to treat mood disorders. It decreases immobility time in the forced swim test. 了解更多
  10. Promazine hydrochloride

    Catalog No. A17638
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    D2DR inhibitor
    Promazine Hydrochloride is a phenothiazine compound and D2DR inhibitor. Promazine Hydrochloride has been employed in studies investigating dopamine-stimulated glycosylation of brain proteins in vitro. It has actions similar to chlorpromazine but with less antipsychotic activity. 了解更多
  11. Asenapine HCl

    Catalog No. A15002
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    adrenergic receptor/5-HT receptor 抑制剂
    Asenapine hydrochloride抑制肾上腺素能受体(α1,α2A,α2B,α2C)的Ki为0.25-1.2 nM,还抑制5-HT受体(1A,1B,2A,2B,2C,5A,6、7),Ki为0.03- 4.0 nM。 了解更多
  12. Phenoxybenzamine hydrochloride

    Catalog No. A10719
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    α-adrenergic (AR) 拮抗剂/CaM 抑制剂
    Phenoxybenzamine hydrochloride是一种细胞可渗透的,非特异性的,不可逆的α-肾上腺素(AR)拮抗剂,也可作为CaM抑制剂。 了解更多

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