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搜索结果：“AZ 960”

“AZ 960”的搜索结果

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Voriconazole (Vfend)

Catalog No. A10978
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CYP17 抑制剂

Voriconazole (Vfend)是一种三唑抗真菌剂，可以冻干粉的形式用于静脉输注溶液。了解更多

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Posaconazole

Catalog No. A10744
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CYP3A4 抑制剂

Posaconazole主要是CYP3A4的抑制剂，但不抑制其他CYP酶的活性。也是甾醇C14+脱甲基酶抑制剂的抑制剂，IC50为0.25μM。泊沙康唑的终末消除半衰期中位数为15-35小时。了解更多

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Ketoconazole

Catalog No. A10498
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P450 抑制剂

ketoconazole作为抗真菌药在结构上类似于咪唑，并干扰真菌细胞膜组成成分麦角甾醇以及某些酶的真菌合成。了解更多

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Cobicistat (GS-9350)

Catalog No. A11277
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CYP3A 抑制剂

Cobicistat (GS-9350)是有效，选择性的细胞色素酶P450 3A (CYP3A)抑制剂，包括重要的cyp3a4亚型。它还抑制肠道转运蛋白，增加几种hiv药物的整体吸收，包括atazanavir、darunavir和tenofovir alafenamide延胡索酸盐。了解更多

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Talarozole R enantiomer

Catalog No. A13113
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Cytochrome P450 抑制剂

Talarozole R enantiomer 通过阻断细胞色素P450酶同工酶CYP26（一种视黄酸羟化酶）来抑制视黄酸的代谢。了解更多

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ABT

Catalog No. A13361
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Cytochrome P450 抑制剂

ABT (1-Aminobenzotriazole)是（CYP）细胞色素P-450和氯过氧化物酶的自杀底物。了解更多

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Azathramycin

Catalog No. A15010
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CYP3A4 抑制剂

Azathramycin是一种抗生素。阿奇霉素与细菌核糖体的50S亚基结合，从而抑制mRNA的翻译。了解更多

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Sulfaphenazole

Catalog No. A17283
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CYP2C9 inhibitor

Sulfaphenazole is a specific inhibitor of CYP2C9 which blocks atherogenic and pro-inflammatory effects of linoleic acid (increase in oxidative stress and activation of AP-1) mediated by CYP2C9. 了解更多

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CYP17-IN-1

Catalog No. A12622
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CYP17 inhibitor

CYP17-IN-1 (compound 9c) is a potent and orally active CYP17 inhibitor against rat and human CYP17 with IC50s of 15.8 and 20.1 nM. 了解更多

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