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￥ 0.00 “AZ 960”的搜索结果
42 个项目
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PF-04620110
Catalog No. A11526 -
JNJ 1661010
Catalog No. A12420 -
Leptomycin B
Catalog No. A20985 nuclear export receptor CRM1 inhibitorLeptomycin B (CI 940; LMB) is a potent inhibitor of the nuclear export of proteins. Leptomycin B inactivates CRM1/exportin 1 by covalent modification at a cysteine residue. Leptomycin B is a potent antifungal antibiotic blocking the eukaryotic cell cycle. 了解更多 -
PAT-1251 Hydrochloride
Catalog No. A21969 LOXL2 inhibitorPAT-1251 Hydrochloride is a potent, selective and oral lysyl oxidase-like 2 (LOXL2) inhibitor, with IC50s of 0.71 and 1.17 μM for hLOXL2 and hLOXL3, respectively, and also potently inhibits mouse, rat, and dog LOXL2 (IC50s, 0.10, 0.12, and 0.16 μM, respectively). 了解更多 -
FAAH inhibitor 1
Catalog No. A21841 FAAH inhibitorFAAH inhibitor 1 (Benzothiazole analog 3) is a potent fatty acid amide hydrolase (FAAH) inhibitor with an IC50 of 18??8 nM. 了解更多 -
Brofaromine
Catalog No. A21777 MAO inhibitorBrofaromine (CGP 11305A) is a monoamine oxidase (MAO) inhibitor with IC50 of 0.2?μM for MAO-A. 了解更多 -
BMS-654457
Catalog No. A21704 Factor XIa (FXIa) inhibitorBMS-654457 is a small-molecule, reversible inhibitor of factor XIa (FXIa), binding with human and rabbit FXIa with Kis of 0.2 and 0.42 nM, respectively. 了解更多 -
Saterinone hydrochloride
Catalog No. A21402 PDE3 inhibitorSaterinone hydrochloride is a phosphodiesterase III (PDE III) inhibitor. 了解更多 -
Lazabemide
Catalog No. A21270 MAO-B inhibitorLazabemide(Ro 19-6327) is selective, reversible monoamine oxidase B (MAO-B) inhibitor (IC50 values are 0.03 and > 100 μM for MAO-B and MAO-A respectively). 了解更多 -
Isocarboxazid
Catalog No. A17887 monoamine oxidase inhibitorIsocarboxazid is a non-selective and irreversible inhibitor of monoamine oxidase, with an IC50 of 4.8 μM for rat brain monoamine oxidase in vitro. 了解更多 -
Retaspimycin
Catalog No. A15221 Hsp90 inhibitorRetaspimycin is a potent and water-soluble inhibitor of Hsp90, with EC50s of 119 nM for both Hsp90 and Grp9. 了解更多 -
CYP17-IN-1
Catalog No. A12622 CYP17 inhibitorCYP17-IN-1 (compound 9c) is a potent and orally active CYP17 inhibitor against rat and human CYP17 with IC50s of 15.8 and 20.1 nM. 了解更多 -
IDH1 Inhibitor 2
Catalog No. A18420 IDH1 inhibitorDH1 Inhibitor 2 is a potent IDH1 inhibitor via a direct covalent modification of His315, with an IC50 of 110 nM. 了解更多 -
Iproniazid phosphate
Catalog No. A18135 MAO inhibitorIproniazid phosphate is an irreversible inhibitor of monoamine oxidase types A and B that is used as an antidepressive agent. It has also been used as an antitubercular agent, but its use is limited by its toxicity. 了解更多 -
Iproniazid
Catalog No. A17445 MAO inhibitorIproniazid is a non-selective, irreversible monoamine oxidase (MAO) inhibitor (MAOI) that is used as an antidepressive agent. 了解更多 -
Ethoxzolamide
Catalog No. A17359 Carbonic anhydrase inhibitorEthoxzolamide is a carbonic anhydrase inhibitor with Ki of 1 nM. 了解更多 -
Sulfaphenazole
Catalog No. A17283 CYP2C9 inhibitorSulfaphenazole is a specific inhibitor of CYP2C9 which blocks atherogenic and pro-inflammatory effects of linoleic acid (increase in oxidative stress and activation of AP-1) mediated by CYP2C9. 了解更多 -
Fomepizole
Catalog No. A16164 -
Gedunin
Catalog No. A16034 -
Acetazolamide
Catalog No. A15859 Carbonic Anhydrase 抑制剂Acetazolamide是一种有效的碳酸酐酶（CA）抑制剂，在临床实践中通常用作迅速降低眼内压（IOP）的直接且容易获得的选择。 了解更多 -
AZD7687
Catalog No. A15012 -
Azathramycin
Catalog No. A15010 -
AZD4017
Catalog No. A13542 -
Pralatrexate
Catalog No. A11522 -
Talarozole R enantiomer
Catalog No. A13113 Cytochrome P450 抑制剂Talarozole R enantiomer 通过阻断细胞色素P450酶同工酶CYP26（一种视黄酸羟化酶）来抑制视黄酸的代谢。 了解更多 -
LY 2183240
Catalog No. A11960 FAAH 抑制剂LY 2183240既可作为内源性大麻素再摄取的有效抑制剂，IC50为270 pM，又可作为脂肪酸酰胺水解酶（FAAH）的抑制剂，IC50为12.4 nM，而脂肪酸酰胺水解酶是负责降解花生四烯酸的主要酶。 了解更多 -
Cobicistat (GS-9350)
Catalog No. A11277 CYP3A 抑制剂Cobicistat (GS-9350)是有效，选择性的细胞色素酶P450 3A (CYP3A)抑制剂，包括重要的cyp3a4亚型。它还抑制肠道转运蛋白，增加几种hiv药物的整体吸收，包括atazanavir、darunavir和tenofovir alafenamide延胡索酸盐。 了解更多 -
Ketoconazole
Catalog No. A10498 -
Brinzolamide
Catalog No. A11765 -
Posaconazole
Catalog No. A10744 CYP3A4 抑制剂Posaconazole主要是CYP3A4的抑制剂，但不抑制其他CYP酶的活性。也是甾醇C14+脱甲基酶抑制剂的抑制剂，IC50为0.25μM。泊沙康唑的终末消除半衰期中位数为15-35小时。 了解更多 -
Voriconazole (Vfend)
Catalog No. A10978 -
Cilostazol
Catalog No. A10217
42 个项目
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- Cytochrome P450 (9)
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- HSP (3)
- Factor Xa (2)
- MAO (7)
- DHFR (1)
- Dehydrogenases (3)
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- FAAH (3)
- CETP (1)
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- Fatty acid synthase (FASN) (1)
- Lactate dehydrogenase A (LDHA) (1)
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