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AZD5153 6-Hydroxy-2-naphthoic acid

Catalog No. A21852
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BET/BRD4 bromodomain inhibitor

AZD5153 6-Hydroxy-2-naphthoic acid is the 6-Hydroxy-2-naphthoic acid of AZD5153. AZD5153 is a potent, selective, and orally available BET/BRD4 bromodomain inhibitor; disrupts BRD4 with an IC50 of 1.7 nM. 了解更多

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MS417

Catalog No. A19433
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BRD4 inhibitor

MS417 is a BET-specific BRD4 inhibitor, binds to BRD4-BD1 and BRD4-BD2 with IC50s of 30, 46 nM and Kds of 36.1, 25.4 nM, respectively, with weak selectivity at CBP BRD (IC50, 32.7 μM). 了解更多

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GNE-049

Catalog No. A20206
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CBP inhibitor

GNE-049 is a highly potent and selective CBP inhibitor with an IC50 of 1.1 nM in TR-FRET assay. GNE-049 also inhibits BRET and BRD4(1) with IC50s of 12 nM and 4200 nM, respectively. 了解更多

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GW841819X

Catalog No. A16367
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BET 抑制剂

GW841819X是(+)-JQ1的类似物，是BET溴结构域的新型抑制剂。GW841819X是单个对映异构体，但在苯并二氮杂3.环3的4位具有不确定的手性。了解更多

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Anacardic Acid

Catalog No. A14226
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KAT5 (Tip60), p300/PCAF 抑制剂

Anacardic Acid是p300和p300/CBP相关因子组蛋白乙酰转移酶的有效抑制剂。了解更多

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MS436

Catalog No. A13749
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BRD4 抑制剂

MS436是用于BRD4溴结构域的重氮基小分子抑制剂，Ki值为30-50 nM。了解更多

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OTX015

Catalog No. A13890
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BET 抑制剂

OTX015是口服可生物利用的BRD2，BRD3和BRD4的小分子抑制剂（EC50s = 10-19 nM）。了解更多

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