“ab fubinaca”的搜索结果

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  1. Fludarabine Phosphate (Fludara)

    Catalog No. A10395
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    Fludarabine Phosphate (Fludara)是一种用于治疗血液恶性肿瘤(血细胞癌,如白血病和淋巴瘤)的化疗药物。氟达拉滨通过干扰核糖核苷酸还原酶和dna聚合酶来抑制DNA合成。它对分裂细胞和静止细胞都有活性。 了解更多
  2. Fludarabine (Fludara)

    Catalog No. A10396
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    STAT 抑制剂
    Fludarabine或fludarabine(fludara)是一种用于治疗血液恶性肿瘤(血细胞癌,如白血病和淋巴瘤)的化疗药物。Fludarabine通过干扰核糖核苷酸还原酶和DNA聚合酶来抑制DNA合成。它对分裂细胞和静止细胞都有活性。 了解更多
  3. 1,2,3,4,5,6-Hexabromocyclohexane

    Catalog No. A15361
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    JAK2 抑制剂
    1,2,3,4,5,6-Hexabromocyclohexane是一种有效且特异性的JAK2自磷酸化抑制剂。 了解更多
  4. Napabucasin

    Catalog No. A13474
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    STAT 抑制剂
    Napabucasin是一种口服小分子药物,它可以阻止癌症干细胞(CSC)自我更新,并诱导CSC和非干细胞中的细胞死亡。 了解更多
  5. Avitinib (AC0010)

    Catalog No. A16826
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    irreversible EGFR 抑制剂
    Avitinib (AC0010)是一种基于吡咯并嘧啶的不可逆EGFR抑制剂,对EGFR L858R/T790M双重突变具有突变选择性,IC50值为0.18 nM,效力比野生型EGFR(IC50值为7.68 nM)高近43倍。它具有可比的抗肿瘤活性和耐受的毒性。 了解更多
  6. Abrocitinib (PF-04965842)

    Catalog No. A18318
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    JAK1 抑制剂
    Abrocitinib (PF-04965842) is a potent, orally active and selective JAK1 inhibitor, with IC50s of 29 and 803 nM for JAK1 and JAK2, respectively. Abrocitinib (PF-04965842) exhibits less active effect on TYK2 (IC50, 1.253 μM), and inhibits phosphorylation of STAT1, STAT3 and STAT5 after stimulation. Effective in autoimmune disease. 了解更多
  7. Upadacitinib (ABT-494)

    Catalog No. A18316
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    JAK-1 抑制剂
    Upadacitinib (ABT-494) is a potent and selective Janus kinase (JAK) 1 inhibitor being developed for the treatment of several autoimmune disorders with an IC50 of 43 nM. IC50 & Target: IC50: 43 nM (JAK1), 200 nM (JAK2) 了解更多
  8. Tofacitinib

    Catalog No. A17252
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    JAK3/2/1 inhibitor
    Tofacitinib is an orally available JAK3/2/1 inhibitor with IC50s of 1, 20, and 112 nM, respectively. 了解更多
  9. GDC-0339

    Catalog No. A20920
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    Pim kinase inhibitor
    GDC-0339 is a potent, orally bioavailable and well tolerated pan-Pim kinase inhibitor, with Kis of 0.03 nM, 0.1 nM and 0.02 nM for Pim1, Pim2 and Pim3, respectively. GDC-0339 is discovered as a potential treatment of multiple myeloma. 了解更多
  10. HS-10296 hydrochloride

    Catalog No. A21661
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    EGFR/T790M inhibitor
    HS-10296 hydrochloride is an orally available and third-Generation inhibitor of epidermal growth factor receptor (EGFR)-activating mutations and T790M-resistant mutation with limited activity against wild-type EGFR. 了解更多

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