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Bergaptol

Catalog No. A12303
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CYP3A4 enzyme inhibitor

Bergaptol is a hydroxylated psoralen that acts as a potent inhibitors of debenzylation activity of CYP3A4 enzyme with an IC50 value of 24.92 uM. Recent studies suggest that it may have antiproliferative and anticancer properties. 了解更多

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Deferasirox

Catalog No. A10293
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Iron chelator

Deferasirox是一种铁螯合剂，也是细胞色素P450 3A4诱导剂，细胞色素P450 2C8抑制剂和细胞色素P450 1A2抑制剂。了解更多

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- Jamie L. Dombach, .et al. A small molecule that mitigates bacterial infection disrupts Gram-negative cell membranes and is inhibited by cholesterol and neutral lipids, PLoS Pathog, 2020, Dec; 16(12): e1009119 PMID: 33290418
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Cobicistat (GS-9350)

Catalog No. A11277
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CYP3A 抑制剂

Cobicistat (GS-9350)是有效，选择性的细胞色素酶P450 3A (CYP3A)抑制剂，包括重要的cyp3a4亚型。它还抑制肠道转运蛋白，增加几种hiv药物的整体吸收，包括atazanavir、darunavir和tenofovir alafenamide延胡索酸盐。了解更多

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Azathramycin

Catalog No. A15010
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CYP3A4 抑制剂

Azathramycin是一种抗生素。阿奇霉素与细菌核糖体的50S亚基结合，从而抑制mRNA的翻译。了解更多

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ABT

Catalog No. A13361
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Cytochrome P450 抑制剂

ABT (1-Aminobenzotriazole)是（CYP）细胞色素P-450和氯过氧化物酶的自杀底物。了解更多

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Itraconazole (Sporanox)

Catalog No. A10489
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Itraconazole (Sporanox)是CYP3A4相对有效的抑制剂，IC50为6.1nM，用作三唑类抗真菌剂。了解更多

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- Paul Mark Medina, .et al. Revealing the anticancer potential of candidate drugs in vivo using Caenorhabditis elegans mutant strains, Transl Oncol, 2021, Jan;14(1):100940 PMID: 33221682
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Naringenin

Catalog No. A10625
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Naringenin是一种黄烷酮，是一种类黄酮，被认为具有抗氧化剂，自由基清除剂，消炎，碳水化合物代谢促进剂和免疫系统调节剂等对人体健康的生物活性。了解更多

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