“ADM Hydrochloride”的搜索结果

产品 1 到 50 共 68个

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  1. Clomipramine HCl

    Catalog No. A10231
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    5-HT Receptor 激动剂
    Clomipramine HCl是下列转运蛋白的阻滞剂:5-羟色胺转运蛋白 (SERT)(Ki = 0.14 nM),去甲肾上腺素转运蛋白(NET)(Ki = 54 nM),多巴胺转运蛋白(DAT)(Ki = 3,020 nM),甘氨酸转运蛋白(GlyT/LeuT)。 了解更多
  2. Dobutamine hydrochloride

    Catalog No. A10325
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    Adrenoceptors 激动剂
    Dobutamine hydrochloride是一种直接作用剂,其主要活性来自刺激心脏的β1肾上腺素能受体,增加收缩力和心输出量。 了解更多
  3. Oxymetazoline hydrochloride

    Catalog No. A10686
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    alpha-1 adrenergic 激动剂
    Oxymetazoline是一种选择性的α-1激动剂和部分α-2激动剂局部减充血剂,以盐酸羟甲唑啉的形式使用。 了解更多
  4. Lidocaine hydrochloride

    Catalog No. A16132
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    Histamine H1-receptor 激动剂
    Lidocaine hydrochloride是用作抗心律不齐药物的局部麻醉药和心脏抑制剂。 了解更多
  5. Rimonabant hydrochloride

    Catalog No. A11548
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    CB1 receptor inverse 激动剂
    Rimonabant hydrochloride是CB1受体反向激动剂。 了解更多
  6. BRL 52537 HCl

    Catalog No. A11210
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    Opioid Receptors 激动剂
    BRL 52537 hydrochloride是一种高度选择性和有效的κ阿片类激动剂(Ki = 0.24 nM)。比吗啡强25倍。 了解更多
  7. Rotigotine HCl

    Catalog No. A11118
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    Dopamine Receptor 激动剂
    Rotigotine hydrochloride是一种多巴胺D2和D3受体激动剂。D2和D3的Ki值分别为13和0.71 nM。 了解更多
  8. Phenylephrine HCl

    Catalog No. A11666
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    α1-adrenergic receptor 激动剂
    Phenylephrine HCl是一种选择性的α1肾上腺素能受体激动剂,主要用作减充血剂,扩张瞳孔和增加血压的药物。 了解更多
  9. Siramesine Hydrochloride

    Catalog No. A12479
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    Sigma-2 receptor 激动剂
    Siramesine Hydrochloride是一种选择性sigma-2受体激动剂,已被证明可触发癌细胞的细胞死亡并在体内表现出强大的抗癌活性。 了解更多
  10. Guanfacine hydrochloride

    Catalog No. A15098
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    α2A-adrenoceptor 激动剂
    Guanfacine hydrochloride是一种抗高血压药,是一种选择性的α2A肾上腺素受体激动剂,Kd为31 nM,选择性是α2B肾上腺素受体的60倍。 了解更多
  11. Pitolisant hydrochloride

    Catalog No. A15213
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    Nonimidazole inverse 激动剂
    Pitolisant hydrochloride是一种在重组人H3受体(Ki = 0.16 nM)处新颖,有效且选择性的壬二唑反向激动剂。 了解更多
  12. rac-Rotigotine Hydrochloride

    Catalog No. A15217
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    D2 receptor 激动剂
    rac-Rotigotine Hydrochloride是D-2受体的高效效价和选择性激动剂,Ki为0.69 nM。 了解更多
  13. Pioglitazone hydrochloride

    Catalog No. A16670
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    PPARγ agonist
    Pioglitazone hydrochloride is a potent and selective PPARγ agonist with EC50s of 0.93 and 0.99 μM for human and mouse PPARγ, respectively. 了解更多
  14. Dexmedetomidine HCl

    Catalog No. A11846
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    alpha2-adrenoceptor 激动剂
    Dexmedetomidine hydrochloride是美托咪啶的活性异构体,它充当有效的,高度选择性的α2-AR(α2-肾上腺素受体)激动剂。 了解更多
  15. Xylazine HCl

    Catalog No. A13434
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    Adrenergic Receptor 激动剂
    Xylazine hydrochloride是α2A-AR、α2B-AR和α2C-AR的活化剂。 了解更多
  16. SKF38393 HCl

    Catalog No. A15839
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    Dopamine Receptor 激动剂?
    SKF38393 HCl是D1激动剂,IC50为110 nM。 了解更多
  17. Xylometazoline HCl

    Catalog No. A17251
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    α-adrenoceptor agonist
    Xylometazoline hydrochloride is an α-adrenoceptor agonist commonly used as nasal decongestant. 了解更多
  18. Ractopamine HCl

    Catalog No. A17372
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    beta-Adrenergic agonist
    Ractopamine HCl is a beta-Adrenergic agonist. It acts by being a full agonist at the TAAR1. 了解更多
  19. Tetrahydrozoline Hydrochloride

    Catalog No. A13080
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    Adrenergic Receptor 激动剂
    Tetrahydrozoline Hydrochloride是一种引起结膜血管收缩的α激动剂。 了解更多
  20. CGS 21680 HCl

    Catalog No. A16441
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    Adenosine A2 receptor 激动剂
    CGS 21680 HCl是腺苷A2受体激动剂,IC50为22 nM,比A1受体高140倍。 了解更多
  21. MCOPPB 3HCl

    Catalog No. A10561
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    NOP receptor 激动剂
    MCOPPB 3HCl是一种用作伤害感受器受体的有效和选择性激动剂的化合物,pKi为10.07。 了解更多
  22. Pramipexole dihydrochloride monohyrate

    Catalog No. A10747
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    Dopamine Receptor 激动剂
    Pramipexole dihydrochloride monohyrate是非麦角灵类的多巴胺激动剂,适用于治疗早期帕金森氏病(PD)和不安腿综合征(RLS)。 了解更多
  23. (+) PD 128907

    Catalog No. A14376
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    Dopamine receptor 激动剂
    (+)-PD 128907 hydrochloride是一种有效的D3DR(多巴胺受体)激动剂(Ki = 2.3 nM)。 了解更多
  24. Medetomidine HCl

    Catalog No. A13775
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    adrenergic alpha-2 receptor 激动剂
    Medetomidine Hydrochloride是一种肾上腺素α2-受体激动剂,Ki为1.08 nM,比作用于α1-adrenoceptor选择性高1620倍。由于其镇痛和镇静作用而被用于兽医学。 了解更多
  25. Dexpramipexole dihydrochloride

    Catalog No. A15066
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    dopamine 激动剂
    Dexpramipexole dihydrochloride是一种神经保护剂和弱非麦角灵多巴胺激动剂。 了解更多
  26. Inolitazone dihydrochloride

    Catalog No. A15129
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    PPARγ 激动剂
    Inolitazone dihydrochloride是一种新型的高亲和力PPARγ激动剂,可激活PPARγ,其EC50约为罗格列酮的EC50,对RIE细胞无影响。 了解更多
  27. GTS-21 (DMBX-A)

    Catalog No. A15950
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    nAChR 激动剂
    GTS-21 dihydrochloride (DMBX-A)是一种选择性的α7烟碱乙酰胆碱受体激动剂,最近已被确定为一种有希望的炎症治疗方法。 了解更多
  28. ZK-756326 dihydrochloride

    Catalog No. A16363
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    CCR8 激动剂
    ZK-756326是有效的,选择性的非肽CCR8趋化因子受体激动剂。ZK 756326抑制了CCR8配体I-309(CCL1)的结合,IC(50)值为1.8μM。 了解更多
  29. Buspirone HCl

    Catalog No. A15687
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    5HT(1A) receptor 激动剂
    Buspirone hydrochloride是一种具有5-D(2)多巴胺能作用的血清素能(5HT(1A)受体激动剂)抗焦虑药,用于焦虑症。 了解更多
  30. KAG-308

    Catalog No. A18389
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    EP4 激动剂
    KAG-308, a newly-identified EP4-selective agonist shows efficacy for treating ulcerative colitis and can bring about lower risk of colorectal carcinogenesis by oral administration. 了解更多
  31. Lesopitron dihydrochloride

    Catalog No. A12950
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    5-HT1A receptor agonist
    Lesopitron dihydrochloride is a full and selective 5-HT1A receptor agonist with IC50 of 125 nM in rat hippocampal membranes. 了解更多
  32. diABZI STING agonist-1 trihydrochloride

    Catalog No. A21694
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    STING receptor agonist
    diABZI STING agonist-1 (trihydrochloride) is a selective stimulator of interferon genes (STING) receptor agonist, with an EC50s of 130 for human PBMCs. 了解更多
  33. TLR7/8 agonist 1 dihydrochloride

    Catalog No. A21700
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    TLR7/8 agonist
    TLR7/8 agonist 1 dihydrochloride is a toll-like receptor (TLR7)/TLR8 dual-agonistic imidazoquinoline. 了解更多
  34. MCOPPB triHydrochloride

    Catalog No. A21722
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    nociceptin receptor agonist
    MCOPPB 3Hcl is a nociceptin receptor agonist with pKi of 10.07; weaker activity at other opioid receptors. 了解更多
  35. Ro 10-5824 dihydrochloride

    Catalog No. A21986
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    dopamine D4 receptor partial agonist
    Ro 10-5824 dihydrochloride is a selective dopamine D4 receptor partial agonist, with Ki of 5.2 nM. 了解更多
  36. Detomidine hydrochloride

    Catalog No. A10298
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    Adrenergic Receptor 激动剂
    Detomidine hydrochloride是具有镇痛作用的镇静剂。α2-肾上腺素能激动剂产生剂量依赖性的镇静和镇痛作用,并通过激活α2儿茶酚胺受体介导,从而引起负反馈反应,从而减少兴奋性神经递质的产生。 了解更多
  37. Clonidine hydrochloride

    Catalog No. A10232
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    Alpha adrenergic 激动剂
    Clonidine hydrochloride被归类为中枢作用的α肾上腺素能激动剂。Clonidine主要作为咪唑啉受体激动剂。 了解更多
  38. Nalfurafine hydrochloride

    Catalog No. A12579
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    opioid κ-selective 激动剂
    Nalfurafine hydrochloride是一种κ-opioid激动剂。 了解更多
  39. ent Naxagolide Hydrochloride

    Catalog No. A13089
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    dopamine D2-receptor 激动剂
    ent Naxagolide Hydrochloride是一种多巴胺D2受体激动剂,用于治疗锥体外系疾病。该化合物是抗帕金森病药物。 了解更多
  40. Nalmefene hydrochloride

    Catalog No. A13843
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    dopamine receptor 激动剂
    Nalmefene hydrochloride是opioid receptor拮抗剂。 了解更多
  41. Idazoxan Hydrochloride

    Catalog No. A13409
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    α2- adrenoceptor 拮抗剂 / I2 imidazoline receptor 激动剂
    Idazoxan hydrochloride 是α2-AR肾上腺素受体拮抗剂和潜在I2咪唑啉受体激动剂。还显示I1咪唑啉受体拮抗剂活性。(I1、I2和α的公钥基础设施值分别为5.90、7.22、8.01、7.43和7.7)。 了解更多
  42. Cevimeline hydrochloride hemihydrate

    Catalog No. A15042
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    M1 激动剂
    Cevimeline hydrochloride hemihydrate是一种新型毒蕈碱受体激动剂,是干燥综合征干燥症的候选治疗药物。 了解更多
  43. Cevimeline hydrochloride

    Catalog No. A18092
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    mAChR agonist
    Cevimeline (Evoxac) Hcl is a parasympathomimetic and muscarinic agonist, with particular effect on M3 receptors; used in the treatment of dry mouth associated with sjogren's syndrome. 了解更多
  44. Tulobuterol hydrochloride

    Catalog No. A18226
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    β2-adrenergic receptor agonist
    Tulobuterol Hydrochloride is a long-acting beta2-adrenergic receptor agonist. 了解更多
  45. CYT-1010 hydrochloride

    Catalog No. A21348
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    mu-opioid receptor agonist
    CYT-1010 hydrochloride is a mu-opioid receptor agonist extracted from patent WO2013173730A2, with EC50s of 13.1 nM and 0.0053 nM on beta-arrestin recruitment and inhibition of cAMP production, respectively. 了解更多
  46. LY 344864 hydrochloride

    Catalog No. A21748
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    5-HT1F agonist
    LY 344864 hydrochloride is a selective 5-HT1F agonist with a Ki of 6 nM. 了解更多
  47. lorcaserin hydrochloride (APD-356)

    Catalog No. A12598
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    serotonin 2C receptor 激动剂
    lorcaserin hydrochloride (APD-356)是血清素2C受体激动剂,可指示与减少热量饮食和增加体育锻炼以减轻慢性体重成人管理。 了解更多
  48. Moxonidine Hydrochloride

    Catalog No. A13416
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    imidazoline receptor 1 激动剂
    Moxonidine Hydrochloride (BDF5895)是咪唑啉1型受体(I1-R)选择性激动剂,为降压剂。 了解更多
  49. UNC 9994 hydrochloride

    Catalog No. A16087
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    dopamine D2 receptor 激动剂
    UNC 9994 hydrochloride,独特的,β-arrestin偏向的功能选择性多巴胺D2受体(D2R)激动剂(Ki值为30 nM;在ε-arrestin-2募集试验中EC50值为50 nM),在体内具有抗精神病活性。UNC9994在野生型小鼠中显着抑制了PCP诱导的超运动,而在Δr-arrestin-2基因敲除小鼠中这种作用被完全消除。 了解更多
  50. SRI-011381 hydrochloride

    Catalog No. A16210
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    TGF-beta 激动剂
    SRI-011381 hydrochloride是一种TGF-β信号传导激动剂。 了解更多

产品 1 到 50 共 68个

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