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￥ 0.00 “kinase inhibitor”的搜索结果
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PDE-9 inhibitor
Catalog No. A11532 -
MMP3 inhibitor 1
Catalog No. A13185 MMP-3 inhibitorMMP3 inhibitor 1 is a potent and highly selective MMP-3 inhibitor with an IC50 of 1 nM. 了解更多 -
Top1 inhibitor 1
Catalog No. A13304 human topoisomerase I (Top1) inhibitorTop1 inhibitor 1 (compound 28) is a potent human topoisomerase I (Top1) inhibitor with an IC50 value of 29 nM. 了解更多 -
HPGDS inhibitor 2
Catalog No. A18390 H-PGDS 抑制剂HPGDS inhibitor 2 is a highly potent and selective hematopoietic prostaglandin D synthase (H-PGDS) inhibitor with an IC50 of 9.9 nM. 了解更多 -
IDH1 Inhibitor 2
Catalog No. A18420 IDH1 inhibitorDH1 Inhibitor 2 is a potent IDH1 inhibitor via a direct covalent modification of His315, with an IC50 of 110 nM. 了解更多 -
KRAS G12C inhibitor 17
Catalog No. A18441 KRAS G12C inhibitorKRAS G12C inhibitor 17 is a potent KRAS G12C inhibitor extracted from patent WO2019110751A1, compound 82, has an IC50 of 5 nM. 了解更多 -
KRAS G12C inhibitor 16
Catalog No. A18444 KRAS G12C inhibitorKRAS G12C inhibitor 16 is a potent KRAS G12C inhibitor extracted from patent WO2019110751A1, compound 39, has an IC50 of 97 nM. 了解更多 -
KRAS G12C inhibitor 15
Catalog No. A18447 KRAS G12C inhibitorKRAS G12C inhibitor 15 is a potent KRAS G12C inhibitor extracted from patent WO2019110751A1, compound 22, has an IC50 of 5 nM. 了解更多 -
PARP14 inhibitor H10
Catalog No. A18616 PARP14 抑制剂PARP14 inhibitor H10, compound H 10, is a selective inhibitor against PARP14 (IC50=490 nM), over other PARPs (??24 fold over PARP1). PARP14 inhibitor H10 induces caspase-3/7-mediated cell apoptosis. 了解更多 -
BRD4 Inhibitor-10
Catalog No. A18679 BRD4-BD1 inhibitorBRD4 Inhibitor-10 is a potent BRD4-BD1 inhibitor extracted from patent WO2015022332A1, Compound II-25, has an IC50 of 8 nM. 了解更多 -
KRAS G12C inhibitor 5
Catalog No. A18840 KRas G12C inhibitorKRAS G12C inhibitor 5 is a KRas G12C inhibitor extracted from patent WO2017201161A1, Compound example 147. 了解更多 -
Tuberculosis inhibitor 1
Catalog No. A18906 trypanosoma brucei growth inhibitorTuberculosis inhibitor 1 is a potent and non-cytotoxic trypanosoma brucei growth inhibitor with an EC50 of 5 nM. 了解更多 -
CA inhibitor 1
Catalog No. A18928 HIV capsid inhibitorCA inhibitor 1 (GS-6207 analog) is a potent HIV capsid inhibitor for HIV inhibition. 了解更多 -
NaV1.7 inhibitor-1
Catalog No. A18933 NaV 1.7 inhibitorNaV1.7 inhibitor-1 is an efficacious voltage-gated sodium channel (NaV) 1.7 inhibitor with an IC50 of 0.6 nM for hNaV1.7, exhibits 80-fold selectivity versus hNaV1.5. 了解更多 -
PKC-theta inhibitor 1
Catalog No. A18966 PKCθ inhibitorPKC-theta inhibitor 1 is the PKCθ inhibitor with an Ki value of 6 nM, inhibits IL-2 production in vivo with an IC50 of 0.19 μM. 了解更多 -
KRAS G12C inhibitor 13
Catalog No. A19041 KRAS G12C inhibitorKRAS G12C inhibitor 13 is a KRAS G12C inhibitor extracted from patent WO2018143315A1, compound 30. 了解更多 -
Syncytial Virus Inhibitor-1
Catalog No. A19053 RSV fusion inhibitorSyncytial Virus Inhibitor-1 is a potent, orally bioavailable respiratory syncytial virus (RSV) fusion inhibitor with EC50s of 0.002 μM, 0.004 μM, and 0.002 μM for RSV Long, RSV A2, and RSV B strains, respectively. 了解更多 -
TDP1 Inhibitor-1
Catalog No. A19072 TDP1 inhibitorTDP1 Inhibitor-1 is a potent Tyrosyl-DNA Phosphodiesterase 1 (TDP1) inhibitor with an IC50 of 7 μM. 了解更多 -
FadD32 Inhibitor-1
Catalog No. A19086 FadD32 inhibitorFadD32 Inhibitor-1 is a potent FadD32 inhibitor with anti-tubercular activity. 了解更多 -
LIN28 inhibitor LI71
Catalog No. A19107 LIN28 inhibitorLIN28 inhibitor LI71 is a potent and cell-permeable LIN28 inhibitor, which abolishes LIN28-mediated oligouridylation with an IC50 of 7 uM. 了解更多 -
HIV-1 inhibitor-3
Catalog No. A19110 HIV infection inhibitorHIV-1 inhibitor-3 is a HIV infection inhibitor extracted from patent US2018360927. 了解更多 -
EMT inhibitor-2
Catalog No. A18568 EMT inhibitorEMT inhibitor-2 inhibits epithelial-mesenchymal transition (EMT) induced by substances such as IL-1β and TGF-β released from the immunocytes. EMT inhibitor-2 inhibits CYP3A4 testosteron and CYP2C9 with IC50s of 49.72 and 5.54 μM, respectively. 了解更多 -
FGFR1/DDR2 inhibitor 1
Catalog No. A18716 FGFR1/DDR2 inhibitorFGFR1/DDR2 inhibitor 1 is an inhibitor of fibroblast growth factor receptor 1 (FGFR1) and discoindin domain receptor 2 (DDR2), with IC50 values of 31.1 nM, 108.4 nM and 3.2 nM for FGFR1, KG-1, and DDR2, respectively. 了解更多 -
RAD51 Inhibitor B02
Catalog No. A18334 RAD51 inhibitorAD51 Inhibitor B02 (B02) is an inhibitor of human RAD51 with an IC50 of 27.4 μM. 了解更多 -
TC-S 7010 (Aurora A Inhibitor I)
Catalog No. A10100 Aurora A 抑制剂TC-S 7010 (Aurora A Inhibitor I)是Aurora A激酶（AurA）的有效和选择性抑制剂，IC50值为3.4 nM（Aurora A），对Aurora B具有极高的选择性1000倍； 用于研究Aurora A激酶的细胞作用的有用工具化合物。 了解更多 -
Ehp inhibitor 2
Catalog No. A22325 Eph family tyrosine kinase inhibitorEhp inhibitor 2 is a Eph family tyrosine kinase inhibitor. 了解更多 -
Raf inhibitor 2
Catalog No. A22641 raf kinase inhibitorRaf inhibitor 2 is a potent raf kinase (IC50<1.0 μM) inhibitor, compound 32, extracted from patent EP1003721B1. Raf inhibitor 2 can be used for cancer research. 了解更多 -
ROCK inhibitor
Catalog No. A15225 ROCK 抑制剂ROCK inhibitor是人类ROCK-1和ROCK-2同工酶的高效抑制剂，IC50值分别为0.6和1.1 nM。 了解更多 -
IRAK inhibitor 3
Catalog No. A11457 IL-1 receptor-associated kinase (IRAK) kinase modulatorIRAK inhibitor 3 is an interleukin-1 (IL-I) receptor-associated kinase (IRAK) kinase modulator extracted from patent WO2008030579 A2. 了解更多 -
cGMP Dependent Kinase Inhibitor Peptid
Catalog No. A16052 PKG/PKA 抑制剂cGMP Dependent Kinase Inhibitor Peptid是一种特定的cGKI（环GMP依赖性蛋白激酶）抑制剂。数据表明，它不阻断完整组蛋白的环状GMP依赖性蛋白激酶磷酸化，已被用于研究恶性疟原虫。 了解更多 -
FB23 inhibitor
Catalog No. A22571 FB23 is a potent and selective inhibitor of N6-methyladenosine (m6A) demethylase FTO (fat mass and obesity associated protein). 了解更多 -
EMT inhibitor-1
Catalog No. A20427 EMT inhibitor-1 is an inhibitor of of Hippo, TGF-β, and Wnt signaling pathways with antitumor activities. 了解更多 -
Glutaminyl Cyclase Inhibitor 3
Catalog No. A20399 GC inhibitorGlutaminyl Cyclase Inhibitor 3 (compound 212 ), a designed anti-Alzheimer??s compound, is a potent human Glutaminyl Cyclase (GC) inhibitor, with an IC50 of 4.5 nM. 了解更多 -
MAT2A inhibitor 1
Catalog No. A20226 MATA2 inhibitorsMAT2A inhibitor 1 is a methionine adenosyltransferase 2A (MATA2) inhibitor with an IC50 less than l00 nM. 了解更多 -
IK1 inhibitor PA-6
Catalog No. A20216 IK1 inhibitorIK1 inhibitor PA-6 (PA-6), a pentamidine analogue, is a selective and potent IK1 (KIR2.x ion-channel-carried inward rectifier current) inhibitor, with IC50 values of 12-15 nM for human and mouse KIR2.x currents. 了解更多 -
ATX inhibitor 1
Catalog No. A20142 ATX inhibitorATX inhibitor 1 is a potent ATX (IC50=1.23 nM, FS-3 and 2.18 nM, bis-pNPP) inhibitor. 了解更多 -
IDH1 Inhibitor 1
Catalog No. A20065 IDH1 inhibitorIDH1 Inhibitor 1 is a potent, orally bioavailable, brain-penetrant and selective mutant IDH1 inhibitor with IC50s of 0.021 μM, 0.045 μM, and 2.52 μM for IDH1R132H, IDH1R132C, and IDH1WT, respectively. Anticancer activity. 了解更多 -
Endothelial lipase inhibitor-1
Catalog No. A20064 endothelial lipase inhibitorEndothelial lipase inhibitor-1 is a potent endothelial lipase inhibitor with an IC50 of 49 nM. 了解更多 -
PI3K/mTOR Inhibitor-1
Catalog No. A20055 PI3K/mTOR inhibitorPI3K/mTOR Inhibitor-1 is a potent, orally bioavailable dual PI3K/mTOR inhibitor with IC50s of 20/376/204/46 nM and 186 nM for PI3Kα/PI3Kβ/PI3Kγ/PI3Kδ and mTOR, respectively. Antitumor activity. 了解更多 -
SOCE inhibitor 1
Catalog No. A20041 SOCE inhibitorSOCE inhibitor 1 is a store-operated calcium entry (SOCE) inhibitor with an IC50 of 4.4 μM. 了解更多 -
Eg5 Inhibitor V, trans-24
Catalog No. A20019 kinesin Eg5 inhibitorEg5 Inhibitor V, trans-24 is a potent and specific kinesin Eg5 inhibitor with an IC50 of 0.65 μM, and can be used in the research of cancer. 了解更多 -
sPLA2-X Inhibitor 31
Catalog No. A20018 sPLA2-X inhibitorsPLA2-X Inhibitor 31 is a selective secreted phospholipase A2 type X (sPLA2-X) inhibitor with IC50s of 26 nM, 310 nM, and 2230 nM for sPLA2-X, sPLA2-IIa, and sPLA2-V, respectively. 了解更多 -
ATM Inhibitor-1
Catalog No. A19931 ATM inhibitorATM Inhibitor-1 is a highly potent, selective and orally active ATM inhibitor, with an IC50 of 0.7 nM. 了解更多 -
ATR inhibitor 1
Catalog No. A19874 ATR inhibitorATR inhibitor 1 is a ATR inhibitor extracted from patent WO2015187451A1, compound I-l, has a Ki value below 1 ?μ. 了解更多 -
AMPD2 inhibitor 1
Catalog No. A19839 AMPD2 inhibitorAMPD2 inhibitor 1 is an adenosine monophosphate deaminase 2 (AMPD2) inhibitor, used in the research of sugar craving, salt craving, umami craving, and addictions including drug, tobacco, nicotine and alcohol addictions. 了解更多 -
Glutaminyl Cyclase Inhibitor 2
Catalog No. A19713 glutaminyl cyclase inhibitorGlutaminyl Cyclase Inhibitor 2 is a glutaminyl cyclase inhibitor with an IC50 of 1.23 μM. 了解更多 -
CDK4/6/1 Inhibitor
Catalog No. A19641 CDK4/6 inhibitorCDK4/6/1 Inhibitor is a CDK4/6 inhibitor with IC50s of 3 and 1 nM, respectively. 了解更多 -
CHK1 inhibitor
Catalog No. A19623 -
PI3Kγ inhibitor 2
Catalog No. A19606 PI3Kγ inhibitorPI3Kγ inhibitor 2 (Compound 16) is an orally bioavailable, CNS-penetrant, isoform selective PI3Kγ inhibitor with a Ki of 4 nM. 了解更多
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