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Desisobutyryl-ciclesonide
Catalog No. A19718 Desisobutyryl-ciclesonide is the active metabolite of Ciclesonide. Desisobutyryl-ciclesonide has affinity for the glucocorticoid receptor. 了解更多 -
Fluorescein di(β-D-galactopyranoside)
Catalog No. A19707 β-galactosidase fluorogenic substrateFluorescein di(β-D-galactopyranoside) is a fluorogenic substrate for β-galactosidase (λex=485 nm, λem=535 nm). 了解更多 -
Oxyphenisatin acetate
Catalog No. A19700 Oxyphenisatin acetate, the pro-drug of oxyphenisatin, is used to be a laxative. 了解更多 -
Fmoc-Ser(O-α-D-GalNAc(OAc)3)-OH
Catalog No. A19684 Fmoc-Ser(O-α-D-GalNAc(OAc)3)-OH is a drug for cancer. 了解更多 -
Aticaprant
Catalog No. A19664 kappa opioid receptor antagonistAticaprant (CERC-501) is a potent and centrally-penetrant kappa opioid receptor antagonist with a Ki of 0.807 nM. 了解更多 -
Melinamide
Catalog No. A19631 cholesterol absorption inhibitorMelinamide, an amide derivative of an unsaturated long-chain fatty acid, is an inhibitor of cholesterol absorption with an IC50 of 20.9 μM. 了解更多 -
PDE5-IN-2
Catalog No. A19625 PDE5 inhibitorPDE5-IN-2 is a potent, highly selective, and orally active PDE5 inhibitor, with an IC50 of 0.31 nM, less potently inhibits PDE2A, PDE10A, PDE4D2, and PDE6C, with IC50s of 106, 46, 43, 1.2 nM, respectively. Anti-pulmonary arterial hypertension activity. 了解更多 -
KP-457
Catalog No. A19622 ADAM17 inhibitorKP-457 is a selective a disintegrin and metalloproteinase 17 (ADAM17) inhibitor, with higher selectivity for ADAM17 than for other MMPs and ADAM10, and IC50s are 11.1 nM (ADAM17), 748 nM (ADAM10), 717 nM (MMP2), 9760 nM (MMP3), 2200 nM (MMP8), 5410 nM (MMP9), 930 nM (MMP13), 2140 nM (MMP14), and 7100 nM (MMP17), respectively. 了解更多 -
HIV-1 integrase inhibitor 4
Catalog No. A19617 INST inhibitorHIV-1 integrase inhibitor 4 is a HIV-1 integrase strand transfer (INST) inhibitor with an IC50 of 3.7 nM. 了解更多 -
ReN-1869 hydrochloride
Catalog No. A19610 histamine H1 receptor antagonistReN 1869 hydrochloride is a novel, selective histamine H1 receptor antagonist, which demonstrates affinity to the histamine H1 receptor (guinea pig brain) with Ki of 0.19±0.04 μM and the non-selective ?? site (guinea pig brain) with Ki of 0.45 μM. 了解更多 -
DS-1040 Tosylate
Catalog No. A19600 TAFIa inhibitorDS-1040 Tosylate is an inhibitor of the activated thrombin-activatable fibrinolysis inhibitor (TAFIa), used for the treatment of acute ischemic stroke (AIS). 了解更多 -
4-(6-Bromo-2-benzothiazolyl)benzenamine
Catalog No. A19574 β-amyloid PET tracer4-(6-Bromo-2-benzothiazolyl)benzenamine is a β-amyloid PET (positron emission tomography) tracer that can be used in the diagnosis of neurological diseases, such as Alzheimer's and Down's syndrome. 了解更多 -
Antibacterial compound 2
Catalog No. A19573 Antibacterial compound 2 is a useful antibacterial agent extracted from patent US5652238, compound example 9. 了解更多 -
GlyRS-IN-1
Catalog No. A19543 GlyRS inhibitorGlyRS-IN-1 is a glycyl-tRNA synthase (GlyRS) inhibitor extracted from patent WO 2017066459 A1. GlyRS-IN-1 can also inhibit the growth of bacteria. 了解更多 -
RIG-1 modulator 1
Catalog No. A19536 RIG-1 modulator 1 is an anti-viral compound which can be useful for the treatment of viral infections including influenza virus, HBV, HCV and HIV extracted from patent WO 2015172099 A1. 了解更多 -
Pralsetinib
Catalog No. A19526 -
JFD00244
Catalog No. A19517 -
Ipsalazide
Catalog No. A19511 sulfasalazine analogIpsalazide is a novel sulfasalazine analog designed to release 5-aminosalicylic acid and a nontoxic carrier molecule in the gastrointestinal tract. 了解更多 -
Avapritinib
Catalog No. A19505 KIT and PDGFRA inhibitorAvapritinib (BLU-285) is a highly potent, selective, and orally bioavailable KIT and PDGFRA activation loop mutant kinases inhibitor with IC50s of 0.27 and 0.24 nM for KIT D816V and PDGFRA D842V, respectively. 了解更多 -
IDH1 Inhibitor 3
Catalog No. A19502 IDH1 inhibitorIDH1 Inhibitor 3 (compound 6f) is a mutant isocitric dehydrogenase 1 (IDH1) inhibitor, with an IC50 of 45 nM for IDH1R132H. 了解更多 -
Octaaminocryptand 1
Catalog No. A19497 -
DS28120313
Catalog No. A19481 hepcidin production inhibitorDS28120313 (compound 32) is an orally hepcidin production inhibitor with an IC50 of 0.093 μM. 了解更多 -
Apararenone
Catalog No. A19480 mineralocorticoid receptor antagonistApararenone (MT-3995) is a novel non-steroidal mineralocorticoid receptor antagonists under development for the treatment of diabetic nephropathies and non-alcoholic steatohepatitis. 了解更多 -
3-Methyltoxoflavin
Catalog No. A19466 PDI inhibitor3-Methyltoxoflavin is a potent Protein disulfide isomerase (PDI) inhibitor, with an IC50 of 170 nM. 了解更多 -
Arrhythmias-Targeting Compound 1
Catalog No. A19464 Arrhythmias-Targeting Compound 1 is used in the research of arrhythmias, extracted from patent WO 2001028992 A2. 了解更多 -
BI-3663
Catalog No. A19455 BI-3663 is a highly selective PTK2/FAK PROTAC, with cereblon ligands to hijack E3 ligases for PTK2 degradation. BI-3663 inhibits PTK2 with an IC50 of 18 nM. BI-3663 is a PROTAC that composes of BI-4464 (HY-124625) linked to Pomalidomide (HY-10984) with a linker. Anti-cancer activity. 了解更多 -
Lith-O-Asp
Catalog No. A19397 ST inhibitorLith-O-Asp is a sialytransferase (ST) inhibitor, with IC50s of 12-37 μM. 了解更多 -
AcLys-PABC-VC-Aur0101
Catalog No. A19371 drug-linker conjugate for ADCAcLys-PABC-VC-Aur0101 is a drug-linker conjugate for ADC (anti-CXCR4 ADC) with potent antitumor activity by using Aur0101 (an auristatin microtubule inhibitor), linked via the cleavable linker AcLys-PABC-VC. 了解更多 -
β-Apo-13-carotenone
Catalog No. A19360 antagonist of RXRαβ-Apo-13-carotenone (D'Orenone) is a naturally occurring β-apocarotenoid functioned as an antagonist of RXRα. 了解更多 -
Lanicemine
Catalog No. A19339 NMDA channel blockerLanicemine (AZD6765) is a low-trapping NMDA channel blocker with a binding (Ki) of 0.56-2.1?μM. 了解更多 -
(+)-JQ1 PA
Catalog No. A19328 BET bromodomain inhibitor(+)-JQ1 PA is a clickable JQ1 for building PROTACs, which acts as a BET bromodomain inhibitor. 了解更多 -
SAHA chloroalkane T1
Catalog No. A19324 SAHA chloroalkane T1 is a chloroalkane capture tag by tethering Vorinostat (SAHA) and a chloroalkane tag T1. 了解更多
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