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￥ 0.00 CSF-1R
| Catalog No. | Inhibitor Name | CSF-1R | Other |
|---|---|---|---|
| A10025 | Linifanib | *** | VEGFR1/FLT1,FLT3,VEGFR2/KDR |
| A10679 | OSI-930 | ** | FLT1,KDR,LCK |
| A11959 | GW2580 | * | |
| A13772 | CEP-32496 | *** | c-Kit,RET,PDGFRβ |
| A15520 | Pexidartinib | ** | |
| A15540 | BLZ945 | **** | |
| A11472 | Ki 20227 | **** | VEGFR-2, PDGFRβ, c-Kit |
Notes:
1.Hover mouse over "" to view the IC50 value.(A few compounds have proven potency but without published IC50 data.)
2.For more details about the compound, click on the product name of your interest.
3.The higher the number of "" is, the more potent the inhibitor or activator is.
4."" refers to compounds which do inhibitory effects on the related isoform, but without specific value.
6 个项目
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Pazopanib (GW-786034)
Catalog No. A11518 VEGFR 抑制剂Pazopanib (GW-786034)是VEGFR-1，VEGFR-2，VEGFR-3，PDGFR-a/β和c-kit的有效且选择性的多靶点酪氨酸激酶抑制剂，可阻止肿瘤生长并抑制血管生成。 了解更多 -
Pexidartinib (PLX3397)
Catalog No. A15520 CSF1/Kit/FLT3 抑制剂Pexidartinib (PLX3397)是KIT，CSF1R和FLT3的小分子酪氨酸激酶（RTK）抑制剂，具有潜在的抗肿瘤活性。 了解更多 -
JTE-952
Catalog No. A18391 CSF-1R 抑制剂TE-952 is a potent, oral active and selective Type II inhibitor of colony stimulating factor-1 receptor (CSF-1R or cFMS, type III receptor tyrosine kinase), with IC50 values of 13 nM and 261 nM for CSF1R and TrkA , respectively. Effective against a mouse collagen-induced model of arthritis. 了解更多
6 个项目
每页