Cannabinoid Receptors

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  1. Taranabant ((1R,2R)stereoisomer)

    Catalog No. A21705
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    CB1 receptor inverse agonist
    Taranabant (1R,2R)stereoisomer is the R-enantiomer of Taranabant. Taranabant is a highly potent and selective cannabinoid 1 (CB1) receptor inverse agonist. 了解更多
  2. Taranabant

    Catalog No. A11578
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    CB1 receptor inverse agonist
    Taranabant is a highly potent and selective cannabinoid 1 (CB1) receptor inverse agonist that inhibits the binding and functional activity of various agonists, with a binding Ki of 0.13 nM for the human CB1R in vitro. 了解更多
  3. CB2R-IN-1

    Catalog No. A12306
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    cannabinoid CB2 receptor inverse agonist
    CB2R-IN-1 is a potent cannabinoid CB2 receptor inverse agonist with a Ki of 0.9 nM. 了解更多
  4. SR 144528

    Catalog No. A12376
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    CB2 inverse 激动剂
    SR 144528是一种选择性的外周大麻素受体反向激动剂,对大鼠脾脏和人重组CB2受体的Ki值为0.6 nM,对大鼠脑和人重组CB1受体的Ki值为400 nM。 了解更多
  5. VCE-004.8

    Catalog No. A18549
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    PPARγ and CB2 receptor dual agonist
    VCE-004.8, a semi-synthetic multitarget cannabinoquinoid, is a specific PPARγ and CB2 receptor dual agonist with potent anti-inflammatory activity. 了解更多
  6. Rimonabant hydrochloride

    Catalog No. A11548
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    CB1 receptor inverse 激动剂
    Rimonabant hydrochloride是CB1受体反向激动剂。 了解更多
  7. AM1241

    Catalog No. A16397
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    CB2 receptor 激动剂
    AM1241是选择性的大麻素CB2受体激动剂,Ki为3.4 nM,相对于CB1受体具有82倍的选择性。 了解更多
  8. Bay 59-3074

    Catalog No. A16328
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    CB1/CB2 receptor 激动剂
    Bay 59-3074是一种新型的选择性CB1/CB2受体部分激动剂,对人CB1和CB2受体的Ki值分别为48.3和45.5 nM。 了解更多
  9. Tedalinab

    Catalog No. A14189
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    CB2 receptor 激动剂
    Tedalinab (GRC-10693)是开发用于治疗骨关节炎和神经性疼痛的药物,它可作为有效的选择性大麻素CB2受体激动剂。与相关的CB1受体相比,它对CB2的选择性为4700x,具有很高的口服生物利用度,并在早期临床试验中显示出令人鼓舞的安全性结果以及有效的镇痛和抗炎作用。 了解更多
  10. GW842166X

    Catalog No. A11253
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    CB2 receptor 激动剂
    GW842166X是一种选择性的非大麻类CB2受体激动剂,EC50为63 nM,对CB1受体没有显著的活性。 了解更多
  11. MDA 19

    Catalog No. A11939
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    CB2 激动剂
    MDA 19是CB2的有效选择性激动剂,对精神活性CB1受体具有合理的选择性。 了解更多
  12. WIN 55,212-2 mesylate

    Catalog No. A11932
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    CB receptor 激动剂
    WIN 55,212-2 mesylate是一种有效的cannabinoid receptor激动剂,在神经性疼痛的大鼠模型中具有有效的镇痛作用。它通过受体介导的信号激活p42和p44 MAP激酶。 了解更多

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