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AZD-4635 (HTL1071)

Catalog No. A16820
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A2AR 拮抗剂

AZD-4635 (HTL1071)是一种口服A2AR拮抗剂，可与人A2AR结合，Ki为1.7 nM，选择性比其他腺苷受体高30倍。了解更多

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AZD-5069

Catalog No. A15941
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CXCR2 拮抗剂

AZD-5069是一种有效的选择性CXCR2拮抗剂，具有抑制COPD患者中性粒细胞向气管迁移的潜能。了解更多

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Glycine

Catalog No. A17936
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NMDA antagonist

AZD-4282, also known as aminoacetic acid and glycine, is a N-methyl-D-aspartate (NMDA) receptor antagonist potentially for the treatment of neuropathic pain. 了解更多

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AZD5582

Catalog No. A21735
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IAPs antagonist

AZD5582 is an antagonist of the inhibitor of apoptosis proteins (IAPs), which binds to the BIR3 domains cIAP1, cIAP2, and XIAP with IC50s of 15, 21, and 15 nM, respectively. 了解更多

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AZD9496 maleate

Catalog No. A21726
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estrogen receptor (ERα) antagonist

AZD9496 maleate is a potent and selective estrogen receptor (ERα) antagonist with IC50 of 0.28 nM. AZD9496 maleate is an orally bioavailable selective oestrogen receptor degrader (SERD). 了解更多

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AZD9496

Catalog No. A15822
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estrogen receptor downregulator and 拮抗剂

AZD9496是一种有效的生物选择性雌激素受体下调剂和拮抗剂。了解更多

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AZD1283

Catalog No. A15443
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P2Y12 receptor 拮抗剂

AZD1283是P2Y12受体的有效拮抗剂，EC50为3.0 ug/kg/min，TI> 10；结合IC50为11 nM。了解更多

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AZD1981

Catalog No. A13186
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CRTH2 receptor 拮抗剂

AZD1981作为疾病相关细胞系统的有效拮抗剂，可抑制DK-PGD2诱导的人嗜酸性粒细胞CD11b表达，IC50为10 nM。了解更多

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Ticagrelor (AZD6140)

Catalog No. A11238
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P2Y12 拮抗剂

Ticagrelor (AZD6140)是第一个可逆结合的口服P2Y（12）受体拮抗剂，可阻断ADP诱导的血小板聚集。了解更多

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