“glucagon receptor”的搜索结果

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  1. Edicotinib

    Catalog No. A13008
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    CSF-1 receptor inhibitor
    Edicotinib is a selective and orally available colony-stimulating factor-1 (CSF-1) receptor inhibitor, and has entered phase IIA clinical trial to study rheumatoid arthritis (RA) despite disease. 了解更多
  2. JTE-952

    Catalog No. A18391
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    CSF-1R 抑制剂
    TE-952 is a potent, oral active and selective Type II inhibitor of colony stimulating factor-1 receptor (CSF-1R or cFMS, type III receptor tyrosine kinase), with IC50 values of 13 nM and 261 nM for CSF1R and TrkA , respectively. Effective against a mouse collagen-induced model of arthritis. 了解更多
  3. FGFR1/DDR2 inhibitor 1

    Catalog No. A18716
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    FGFR1/DDR2 inhibitor
    FGFR1/DDR2 inhibitor 1 is an inhibitor of fibroblast growth factor receptor 1 (FGFR1) and discoindin domain receptor 2 (DDR2), with IC50 values of 31.1 nM, 108.4 nM and 3.2 nM for FGFR1, KG-1, and DDR2, respectively. 了解更多
  4. ALW-II-41-27

    Catalog No. A12493
    Eph receptor 抑制剂
    ALW-II-41-27是新型的Eph受体酪氨酸激酶抑制剂。 了解更多
  5. Dovitinib lactate

    Catalog No. A21851
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    FGFR3 inhibitor
    Dovitinib(CHIR-258; TKI258) lactate is a potent inhibitor of fibroblast growth factor receptor 3 (FGFR3) with an IC50 of 5 nM. 了解更多
  6. HS-10296 hydrochloride

    Catalog No. A21661
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    EGFR/T790M inhibitor
    HS-10296 hydrochloride is an orally available and third-Generation inhibitor of epidermal growth factor receptor (EGFR)-activating mutations and T790M-resistant mutation with limited activity against wild-type EGFR. 了解更多
  7. TAS-115

    Catalog No. A21533
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    VEGFR/c-Met/HGFR inhibitor
    TAS-115 is a potent VEGFR and hepatocyte growth factor receptor (c-Met/HGFR)-targeted kinase inhibitor with IC50s of 30 and 32 nM for rVEGFR2 and rMET, respectively. 了解更多
  8. Indirubin Derivative E804

    Catalog No. A21052
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    IGF1R inhibitor
    E 804 is a potent inhibitor of Insulin-like Growth Factor 1 Receptor (IGF1R), with an IC50 of 0.65 μM for IGF1R. 了解更多
  9. EGFR-IN-3

    Catalog No. A15847
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    EGFR inhibitor
    EGFR-IN-3 is an epidermal growth factor receptor (EGFR) inhibitor. 了解更多
  10. GENZ-882706

    Catalog No. A12484
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    CSF-1R Inhibitor
    GENZ-882706 is a potent colony stimulating factor-1 receptor (CSF-1R) Inhibitor extracted from patent WO 2017015267A1. 了解更多
  11. CHMFL-EGFR-202

    Catalog No. A12524
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    EGFR inhibitor
    CHMFL-EGFR-202 is a potent, irreversible inhibitor of epidermal growth factor receptor (EGFR) mutant kinase, with IC50s of 5.3 nM and 8.3 nM for drug-resistant mutant EGFR T790M and WT EGFR kinases, respectively. 了解更多
  12. FLT3-IN-4

    Catalog No. A18509
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    FLT3 inhibitor
    FLT3-IN-4 is a potent and orally effective Fms-like tyrosine receptor kinase 3 (FLT3; IC50=7 nM) inhibitor for treating acute myelogenous leukemia. 了解更多
  13. c-Fms-IN-8

    Catalog No. A18879
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    CSF-1R, c-FMS Type II inhibitor
    c-Fms-IN-8 (compound 4a) is a colony stimulating factor-1 receptor (CSF-1R, c-FMS) Type II inhibitor, with an IC50 of 9.1 nM. 了解更多
  14. WRG-28

    Catalog No. A18832
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    DDR2 inhibitor
    WRG-28 is a novel, potent and selective, allosteric inhibitor of discoidin domain receptor 2 (ddr2). 了解更多
  15. DBPR112

    Catalog No. A18857
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    EGFR 抑制剂
    DBPR112 is an orally active Furanopyrimidine-Based Epidermal Growth Factor Receptor inhibitor with IC50s of 15 nM and 48 nM for EGFRWT and EGFRL858R/T790M, respectively. 了解更多
    • 最新产品

    AG1295

    Catalog No. A17227
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    PDGFR 抑制剂
    AG1295 is a PDGF receptor specific inhibitor. 了解更多
  16. AG 555

    Catalog No. A18337
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    EGFR 抑制剂
    AG555 is a potent epidermal growth factor receptor (EGFR) kinase inhibitor. 了解更多
  17. LDC1267

    Catalog No. A13003
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    TAM Receptor 抑制剂
    LDC1267是一种高选择性TAM(Tyro3,Axl和Mer)激酶抑制剂,对于Tyro3,Axl和Mer的IC50分别小于5 nM/8 nM/29 nM。 了解更多
  18. EGFR Inhibitor

    Catalog No. A13673
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    EGFR 抑制剂
    EGFR inhibitor是一种可透过细胞的4,6-二取代嘧啶化合物,可选择性抑制EGFR激酶,在体外的IC50值为21 nM,可阻断细胞中的受体自身磷酸化。 了解更多
  19. DDR1-IN-1

    Catalog No. A13985
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    DDR1 receptor 抑制剂
    DDR1-IN-1是一种有效的选择性DDR1受体酪氨酸激酶抑制剂,IC50/EC50为105 nM/87 nM,对DDR2的效力低4倍(IC50 = 413 nM)。 了解更多

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