“ADM Hydrochloride”的搜索结果

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  1. Phenformin hydrochloride

    Catalog No. A10717
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    Phenformin hydrochloride是双胍类药物中苯乙双胍的盐酸盐,具有抗糖尿病活性。 了解更多
  2. CAL-130 Hydrochloride

    Catalog No. A15031
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    PI3K 抑制剂
    CAL-130 Hydrochloride是一种新型的磷酸肌醇3激酶(PI3K)抑制剂。据报道,PI3Kδ/γ的联合抑制可作为T细胞急性淋巴细胞白血病(T-ALL)的疗法。 了解更多
  3. AT7867 2HCl

    Catalog No. A15006
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    Akt 抑制剂
    AT7867 dihydrochloride是一种有效的ATP竞争性Akt1/2/3和p70S6K/PKA抑制剂,IC50分别为32 nM/17 nM/47 nM和85 nM/20 nM,在AGC激酶家族之外几乎没有活性。 了解更多
  4. CHIR-99021 monohydrochloride

    Catalog No. A21430
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    GSK-3α/β inhibitor
    CHIR-99021 monohydrochloride (CT99021 monohydrochloride) is a GSK-3α/β inhibitor with IC50 of 10 nM/6.7 nM; > 500-fold selectivity for GSK-3 versus its closest homologs CDC2 and ERK2, as well as other protein kinases. 了解更多
  5. CHIR-99021 trihydrochloride

    Catalog No. A21436
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    GSK-3α/β inhibitor
    CHIR-99021 trihydrochloride (CT99021 trihydrochloride) is a GSK-3α/β inhibitor with IC50 of 10 nM/6.7 nM. 了解更多
  6. Ipatasertib dihydrochloride

    Catalog No. A21734
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    pan-Akt inhibitor
    Ipatasertib dihydrochloride (GDC-0068 dihydrochloride) is a highly selective pan-Akt inhibitor targeting Akt1/2/3 with IC50 of 5/18/8 nM, 620-fold selectivity over PKA. 了解更多
  7. PIK-75 hydrochloride

    Catalog No. A10729
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    PI3K 抑制剂
    PIK-75是一种p110α抑制剂,IC50值为5.8nM。在p110γ和p110β的效果较差,IC50值为0.076 ?M和1.3 ?M。 了解更多
  8. PI-103 Hydrochloride

    Catalog No. A15212
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    PI3K 抑制剂
    PI-103 Hydrochloride是对重组PI3K亚型p110alpha(IC50 = 2 nM),p110beta(IC50 = 3 nM),p110delta(IC50 = 3 nM)和p110gamma(IC50 = 15 nM)具有低IC50值的有效抑制剂,对mTOR的效力较低/DNA-PK,IC50为30 nM/23 nM。 了解更多
  9. MELK-8a hydrochloride

    Catalog No. A21751
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    MELK inhibitor
    MELK-8a hydrochloride is a novel maternal embryonic leucine zipper kinase (MELK) inhibitor with an IC50 of 2 nM. 了解更多
  10. NVP-BKM120 Hydrochloride

    Catalog No. A15195
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    PI3K 抑制剂?
    NVP-BKM120 Hydrochloride是p110α/β/δ/γ的选择性PI3K抑制剂,IC50分别为52 nM/166 nM/116 nM/262 nM。对VPS34,mTOR,DNA-PK的效力降低,对PI4Kβ几乎没有活性。 了解更多
  11. JNJ-47117096 hydrochloride

    Catalog No. A21542
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    MELK inhibitor
    JNJ-47117096 hydrochloride is potent and selective MELK inhibitor, with an IC50 of 23 nM, also effectively inhibits Flt3, with an IC50 of 18 nM. 了解更多
  12. Alpelisib hydrochloride

    Catalog No. A21794
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    PI3Kα inhibitor
    Alpelisib hydrochloride (BYL-719 hydrochloride) is a potent, orally active, and selective PI3Kα inhibitor with IC50s of 5 nM, 250 nM, 290 nM and 1200 nM for p110α, p110γ, p110δ, and p110β, respectively. 了解更多
  13. TGR-1202 hydrochloride (Umbralisib HCl)

    Catalog No. A16278
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    PI3Kδ 抑制剂
    TGR-1202 hydrochloride是一种口服的下一代PI3Kδ抑制剂,在基于酶和细胞的测定中抑制PI3Kδ活性,IC50和EC50值分别为22.2和24.3 nM。 了解更多

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