“glucagon receptor”的搜索结果

产品 1 到 50 共 51个

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  1. Anisodamine

    Catalog No. A18215
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    alpha-1 adrenergic receptors / mAChRs inhibitor
    Anisodamine is an inhibitor of alpha-1 adrenergic receptors and mAChRs isolated from Chinese solanacea plant. 了解更多
  2. Urapidil

    Catalog No. A17074
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    α1 adrenoreceptor 拮抗剂
    Urapidil是一种α1肾上腺素受体拮抗剂和5-HT1A受体激动剂。 了解更多
  3. Vilanterol

    Catalog No. A13125
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    ultra-long-acting β? adrenoreceptor 激动剂
    Vilanterol是一种新的选择性β2-AR激动剂,PEC50值为10.37±0.05。 了解更多
  4. Acebutolol HCl

    Catalog No. A16387
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    β-adrenergic receptors 拮抗剂
    Acebutolol HCl是一种β-肾上腺素能受体拮抗剂,用于治疗高血压,心绞痛和心律不齐。 了解更多
  5. Cimaterol

    Catalog No. A13401
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    β-adrenergic receptors 激动剂
    Cimaterol是β的有效激动剂;肾上腺素能受体(人β的pEC50 = 8.13、8.78和6.62;1β,2β和3β)。 了解更多
  6. BRL 37344 Na Salt

    Catalog No. A13676
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    β3-adrenergic receptors 激动剂
    BRL 37344 Na Salt是具有脂解活性的β3-AR(β3-肾上腺素能受体)选择性激动剂。 了解更多
  7. Labetalol HCl

    Catalog No. A14239
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    alpha1/beta adrenergic receptors 拮抗剂
    Labetalol HCl是选择性α1-肾上腺素能受体和非选择性β-肾上腺素能受体的双重拮抗剂。 了解更多
  8. Bisoprolol

    Catalog No. A13406
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    Bisoprolol是心脏选择性β1-adrenergic receptor阻滞剂,用于阻止心肌梗死、心力衰竭、心绞痛和轻中度高血压。 了解更多
  9. Asenapine

    Catalog No. A18010
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    adrenergic receptor inhibitor
    Asenapine(Org 5222) inhibits adrenergic receptor (α1, α2A, α2B, α2C) with Ki of 0.25-1.2 nM and also inhibits 5-HT receptor (1A, 1B, 2A, 2B, 2C, 5A, 6, 7) with Ki of 0.03-4.0 nM. 了解更多
  10. Atenolol

    Catalog No. A21962
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    β1 receptor antagonist
    Atenolol is a selective β1 receptor antagonist. 了解更多
  11. Norepinephrine hydrochloride

    Catalog No. A21605
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    β1-selective adrenergic receptor agonist
    Norepinephrine hydrochloride (Levarterenol hydrochloride; L-Noradrenaline hydrochloride) is a β1-selective adrenergic receptor agonist with EC50 of 5.37 μM. 了解更多
  12. β3-AR agonist 1

    Catalog No. A12777
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    β3-adrenergic receptor agonist
    β3-AR agonist 1 (compound 15) is a highly potent, selective, and orally available β3-adrenergic receptor (β3-AR) agonist (EC50=18 nM), being inactive to β1-, β2-, and α1A-AR (β1/β3, β2/β3, and α1A/β3>556-fold). 了解更多
  13. Norepinephrine

    Catalog No. A11306
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    β1-selective adrenergic receptor agonist
    Norepinephrine (Levarterenol; L-Noradrenaline) is a β1-selective adrenergic receptor agonist with EC50 of 5.37 μM. 了解更多
  14. OPC-28326

    Catalog No. A12762
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    α2-adrenergic receptor angatonist
    OPC-28326 is a selective peripheral vasodilator and an angatonist of α2-adrenergic receptor, with Ki of 2040, 285, and 55?nM for α2A-, α2B- and α2C-adrenoceptors, respectively. 了解更多
  15. BI-167107

    Catalog No. A18687
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    β2 adrenergic receptor agonist
    BI-167107 is a high affinity, full agonist that binds to the β2 adrenergic receptor (β2AR) with a dissociation constant Kd of 84 pM. 了解更多
  16. Tulobuterol hydrochloride

    Catalog No. A18226
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    β2-adrenergic receptor agonist
    Tulobuterol Hydrochloride is a long-acting beta2-adrenergic receptor agonist. 了解更多
  17. Metipranolol hydrochloride

    Catalog No. A18064
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    β-adrenergic receptor antagonist
    Metipranolol (hydrochloride) is a non-selective β-adrenergic receptor (β-AR) antagonist. Formulations containing metipranolol have been used in the treatment of elevated IOP in patients with ocular hypertension or glaucoma. 了解更多
  18. Brimonidine

    Catalog No. A17899
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    α2-adrenergic receptor agonist
    Brimonidine (UK 14304) is a full α2-adrenergic receptor (α2-AR) agonist. 了解更多
  19. Doxazosin

    Catalog No. A17779
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    α-1 adrenergic receptor blocker
    Doxazosin is an α-1 adrenergic receptor blocker that inhibits the binding of norepinephrine, which is released from sympathetic nerve terminals, to the α-1 receptors on the membrane of vascular smooth muscle cells. Blockages of the alpha-1 adrenergic action on the vascular smooth muscles lead to a decrease in vascular resistance and antihypertensive activity. 了解更多
  20. Nifenalol HCl

    Catalog No. A17246
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    beta-adrenergic receptor antagonist
    Nifenalol, also known as INPEA, is a new beta-adrenergic receptor antagonist. 了解更多
  21. Asenapine HCl

    Catalog No. A15002
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    adrenergic receptor/5-HT receptor 抑制剂
    Asenapine hydrochloride抑制肾上腺素能受体(α1,α2A,α2B,α2C)的Ki为0.25-1.2 nM,还抑制5-HT受体(1A,1B,2A,2B,2C,5A,6、7),Ki为0.03- 4.0 nM。 了解更多
  22. AGN 192836

    Catalog No. A13013
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    α2 adrenergic agonist
    AGN 192836 is a potent and selective α2 adrenergic agonist with EC50s of 8.7, 41 and 6.6 nM for α2A, α2B and α2C receptor, respectively. 了解更多
  23. Clorprenaline HCl

    Catalog No. A16465
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    β2-adrenergic receptor 激动剂
    Clorprenaline HCl是一种β2受体激动剂,具有显着的支气管扩张作用。 了解更多
  24. Brimonidine Tartrate

    Catalog No. A15033
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    α-adrenergic receptor 激动剂
    Brimonidine Tartrate是一种高度选择性的α-肾上腺素能受体激动剂,对α2A肾上腺素能受体的EC50为0.45 nM。 了解更多
  25. Vilanterol trifenatate

    Catalog No. A15998
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    β2-adrenergic receptor 激动剂
    Vilanterol trifenatate是一种长效的β-2激动剂药物,于2013年5月与葛兰素氟替卡松合用,获葛兰素史克(Brax Elmitta)出售为Breo Ellipta,用于治疗慢性阻塞性肺疾病(COPD)。 了解更多
  26. ICI-118551

    Catalog No. A15878
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    β2 adrenergic receptor 拮抗剂
    ICI-118551是选择性的β2肾上腺素能受体(肾上腺素受体)拮抗剂。 了解更多
  27. Tamsulosin hydrochloride

    Catalog No. A14936
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    α1 receptor 拮抗剂
    Tamsulosin hydrochloride是一种选择性的α1受体拮抗剂,是用于良性前列腺增生的药物。 了解更多
  28. Xylazine HCl

    Catalog No. A13434
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    Adrenergic Receptor 激动剂
    Xylazine hydrochloride是α2A-AR、α2B-AR和α2C-AR的活化剂。 了解更多
  29. Tulobuterol

    Catalog No. A13432
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    Adrenergic Receptor 激动剂
    Tulobuterol是β-肾上腺素能受体激动剂,在结构上与特布他林有关。 了解更多
  30. Rauwolscine

    Catalog No. A13426
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    α2-adrenergic receptor 拮抗剂
    Rauwolscine是一种天然生物碱,具有选择性和可逆性α2肾上腺素能受体拮抗剂(Ki = 12 nM)。 了解更多
  31. NAN-190 hydrobromide

    Catalog No. A13417
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    5-HT1A receptor 拮抗剂
    NAN-190 hydrobromide是一种广泛用于科学研究的药物和研究化学品。以前认为它是一种选择性的5-HT1A受体拮抗剂,但后来的发现表明它也能有效地阻断α2肾上腺素能受体。 了解更多
  32. Idazoxan Hydrochloride

    Catalog No. A13409
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    α2- adrenoceptor 拮抗剂 / I2 imidazoline receptor 激动剂
    Idazoxan hydrochloride 是α2-AR肾上腺素受体拮抗剂和潜在I2咪唑啉受体激动剂。还显示I1咪唑啉受体拮抗剂活性。(I1、I2和α的公钥基础设施值分别为5.90、7.22、8.01、7.43和7.7)。 了解更多
  33. HEAT hydrochloride (BE 2254)

    Catalog No. A13408
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    Adrenergic α1 Receptor 拮抗剂
    HEAT hydrochloride (BE 2254)是一种选择性很强的α1-肾上腺素受体拮抗剂,是3-[125I]-衍生物的前体。肾上腺素受体或肾上腺素能受体是参与多种交感神经系统过程的G蛋白偶联受体。 了解更多
  34. Celiprolol HCl

    Catalog No. A13623
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    adrenergic receptor 拮抗剂
    Celiprolol HCl是一种b1肾上腺素能受体拮抗剂和b2肾上腺素能受体局部激动剂,在体外显示其ED50值为40-50 uM可使人的动脉和静脉松弛。 了解更多
  35. Medetomidine HCl

    Catalog No. A13775
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    adrenergic alpha-2 receptor 激动剂
    Medetomidine Hydrochloride是一种肾上腺素α2-受体激动剂,Ki为1.08 nM,比作用于α1-adrenoceptor选择性高1620倍。由于其镇痛和镇静作用而被用于兽医学。 了解更多
  36. Atipamezole HCl

    Catalog No. A13902
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    α2 adrenergic receptor 拮抗剂
    Atipamezole hydrochloride是一种选择性α2肾上腺素受体拮抗剂(α2A、α2B、α2C、α1A和α1B受体的Ki值分别为1.1、1.0、0.89、1300和6500nm)。已经被证明是大脑的渗透剂。 了解更多
  37. Nebivolol

    Catalog No. A13738
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    Beta-1 adrenergic receptor blocker
    Nebivolol是一种选择性抑制β-1肾上腺素能受体,IC50为0.8 nM。 了解更多
  38. Pindolol

    Catalog No. A13422
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    Beta adrenergic receptor blocker
    Pindolol是一种非选择性β阻断剂,具有部分β肾上腺素能受体激动剂活性。 了解更多
  39. ICI 118,551 hydrochloride

    Catalog No. A13225
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    β2 adrenergic 拮抗剂
    ICI 118,551 hydrochloride是选择性的β2 adrenergic receptor 拮抗剂,结合 β2,β1 和 β3 肾上腺素能受体的Ki 值分别为 0.7,49.5 和 611 nM。 了解更多
  40. Tetrahydrozoline Hydrochloride

    Catalog No. A13080
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    Adrenergic Receptor 激动剂
    Tetrahydrozoline Hydrochloride是一种引起结膜血管收缩的α激动剂。 了解更多
  41. Mirabegron

    Catalog No. A12861
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    β3 adrenergic receptor activator
    Mirabegron是一种选择性的beta3-adrenoceptor(β3肾上腺素受体)激动剂,EC50为22.4 nM。是有效的膀胱松弛药和糖尿病药物。 了解更多
  42. Salmeterol

    Catalog No. A11788
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    beta2-adrenergic receptor 激动剂
    Salmeterol是一种长效β2-肾上腺素能受体激动剂。 了解更多
  43. Carvedilol

    Catalog No. A11843
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    β2-adrenergic receptor
    Carvedilol是具有抗氧化特性的β1和β2肾上腺素能受体(AR)激动剂。 了解更多
  44. Detomidine hydrochloride

    Catalog No. A10298
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    Adrenergic Receptor 激动剂
    Detomidine hydrochloride是具有镇痛作用的镇静剂。α2-肾上腺素能激动剂产生剂量依赖性的镇静和镇痛作用,并通过激活α2儿茶酚胺受体介导,从而引起负反馈反应,从而减少兴奋性神经递质的产生。 了解更多
  45. Metoprolol tartrate

    Catalog No. A11713
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    Beta1 receptor blocker
    Metoprolol tartrate是一种选择性β1受体阻滞剂,用于治疗多种心血管系统疾病,尤其是高血压。 了解更多
  46. Apalutamide (ARN-509)

    Catalog No. A11923
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    Androgen Receptor 抑制剂
    Apalutamide (ARN-509)是一种具有潜在抗肿瘤活性的雄激素受体拮抗剂,IC50 为 16 nM。ARN-509与靶组织中的AR结合,从而阻止了雄激素诱导的受体激活,并促进了无法转运至细胞核的无活性复合物的形成。这防止了AR应答基因的结合和转录。 了解更多
  47. Phenylephrine HCl

    Catalog No. A11666
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    α1-adrenergic receptor 激动剂
    Phenylephrine HCl是一种选择性的α1肾上腺素能受体激动剂,主要用作减充血剂,扩张瞳孔和增加血压的药物。 了解更多
  48. Bisoprolol fumarate

    Catalog No. A10149
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    β1 adrenergic receptor blocker
    Bisoprolol fumarate是一种属于β受体阻滞剂的药物,β受体阻滞剂是一类主要用于心血管疾病的药物。更具体地说,它是一种选择性的β1肾上腺素能受体阻滞剂。 了解更多
  49. Naftopidil 2HCl

    Catalog No. A10619
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    5-HT1A and α1-adrenergic receptor 拮抗剂
    Naftopidil 2HCl是选择性5-HT1A和α1-肾上腺素能受体拮抗剂,IC50分别为0.1μM和0.2μM。 了解更多
  50. Salbutamol sulfate (Albuterol)

    Catalog No. A10819
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    Adrenergic Receptor 激动剂
    Salbutamol sulfate (Albuterol)是一种短效β2肾上腺素能受体激动剂。 了解更多

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