微信关注
China
Total item
Cart Subtotal
￥ 0.00 “receptor”的搜索结果
-
CIQ
Catalog No. A15523 -
SB-505124 HCl
Catalog No. A15232 -
BRL 37344 Na Salt
Catalog No. A13676 -
Labetalol HCl
Catalog No. A14239 alpha1/beta adrenergic receptors 拮抗剂Labetalol HCl是选择性α1-肾上腺素能受体和非选择性β-肾上腺素能受体的双重拮抗剂。 了解更多 -
NVP-AAM077 Tetrasodium Hydrate (PEAQX)
Catalog No. A14071 -
CVT 6883
Catalog No. A13745 -
2-Hydroxysaclofen
Catalog No. A13696 -
VU 0361737
Catalog No. A12467 mGlu4 receptors modulatorVU 0361737是mGluR-4的选择性正变构调节剂（人和大鼠受体的EC50值分别为240和110 nM）。 了解更多 -
Bisoprolol
Catalog No. A13406 Bisoprolol是心脏选择性β1-adrenergic receptor阻滞剂，用于阻止心肌梗死、心力衰竭、心绞痛和轻中度高血压。 了解更多 -
LY 255283
Catalog No. A13090 -
Oxybutynin
Catalog No. A10684 Oxybutynin (Ditropan)是一种抗胆碱能药物，是一种竞争性的muscarinic acetylcholine receptorM1，M2，和M3拮抗剂，用于缓解尿道和膀胱疾病。 了解更多 -
Ondansetron HCl (GR 38032F)
Catalog No. A10674 5-HT Receptors 拮抗剂Ondansetron HCl (GR 38032F)是5-羟色胺5-HT3受体拮抗剂，主要用作止吐药，通常在化疗后用于治疗恶心和呕吐。 了解更多 -
Anamorelin
Catalog No. A12346 Anamorelin是一种新型 ghrelin receptor激动剂，FLIPR 检测中，EC50 为 0.74 nM，用于治疗与恶病质/厌食症相关的非小肺癌。 了解更多 -
Chlormezanone (Trancopal)
Catalog No. A10201 Chlormezanone (Trancopal)是一种非苯二氮卓类药物，用于治疗焦虑症。已经建议将其用于治疗肌肉痉挛。氯甲酮与中央苯并二氮杂receptor受体结合，后者与GABA受体发生变构作用。这增强了抑制性神经递质GABA的作用，增强了对网状激活系统的抑制作用，并阻断了在刺激网状通路后发生的皮质和边缘觉醒。 了解更多 -
Calcitriol (Rocaltrol)
Catalog No. A10173 Calcitriol (Rocaltrol)作为vitamin D的激素活性形式，是一种非选择性vitamin D receptor的激活剂，对vitamin D receptor的结合亲和力(IC50=0.4 nM)。 了解更多 -
BRL 52537 HCl
Catalog No. A11210 Opioid Receptors 激动剂BRL 52537 hydrochloride是一种高度选择性和有效的κ阿片类激动剂（Ki = 0.24 nM）。比吗啡强25倍。 了解更多 -
GW3965 HCl
Catalog No. A11204 -
A2A receptor antagonist 1
Catalog No. A12567 adenosine A2A/A1 receptor antagonistA2A receptor antagonist 1 (CPI-444 analog) is an antagonist of both adenosine A2A receptor and A1 receptor with Kis of 4 and 264 nM, respectively. 了解更多 -
Sigma-1 receptor antagonist 2
Catalog No. A18504 sigma 1 receptor antagonistSigma-1 receptor antagonist 2 is a potent and selective sigma 1 receptor (??1 R) antagonist with Kis of 3.88 and 1288 nM for ??1 and ??2 receptor, respectively. 了解更多 -
S1p receptor agonist 1
Catalog No. A20461 S1P receptor agonistS1p receptor agonist 1 is an S1P receptor agonist extracted from patent WO 2015039587 A1, compound example 2. 了解更多 -
Sigma-2 receptor antagonist 1
Catalog No. A20310 sigma-2 (??-2) receptor antagonistSigma-2 receptor antagonist 1 is a sigma-2 (??-2) receptor antagonist. 了解更多 -
Interferon receptor inducer-1
Catalog No. A19877 IFN receptor inducerInterferon receptor inducer-1 (compound 6) is an interferon (IFN) receptor inducer. Used accordingly in the treatment of a disorder in which the induction of interferon is involved. 了解更多 -
Y1 receptor antagonist 1
Catalog No. A19763 neuropeptide Y1 receptor antagonistY1 receptor antagonist 1 (H 409-22 isomer) is a neuropeptide Y1 receptor antagonist. 了解更多 -
Glucagon receptor antagonists-1
Catalog No. A11428 glucagon receptor antagonistGlucagon receptor antagonists-1 is a highly potent glucagon receptor antagonist. 了解更多 -
Glucocorticoid receptor agonist
Catalog No. A11431 Glucocorticoid receptor agonistGlucocorticoid receptor agonist is a potent Glucocorticoid receptor agonist. 了解更多 -
Sigma-1 receptor antagonist 3
Catalog No. A18501 Sigma-1 receptor antagonistSigma-1 receptor antagonist 3 (compound135) is a potent and selective Sigma-1 (??1) receptor antagonist with a Ki of 1.14 nM. 了解更多 -
H4 Receptor antagonist 1
Catalog No. A18929 histamine H4 receptor inverse agonistH4 Receptor antagonist 1 is a potent and selective histamine H4 receptor inverse agonist, with an IC50 of 19 nM. 了解更多 -
Glucagon receptor antagonists-3
Catalog No. A11430 Glucagon receptor antagonistGlucagon receptor antagonists-3 is a highly potent glucagon receptor antagonist. 了解更多 -
Glucagon receptor antagonists-2
Catalog No. A11429 Glucagon receptor antagonistGlucagon receptor antagonists-2 is a highly potent glucagon receptor antagonist. 了解更多 -
GLP-1 receptor agonist 1
Catalog No. A19885 GLP-1 receptor agonistGLP-1 receptor agonist 1 is a glucagon-like peptide-1 (GLP-1) receptor agonist extracted from patent WO2018056453A1, Compound 67. 了解更多 -
GLP-1 receptor agonist 2
Catalog No. A19722 GLP-1R agonistGLP-1 receptor agonist 2 is a glucagon-like peptide-1 receptor (GLP-1R) agonist. 了解更多 -
Orexin 2 Receptor Agonist
Catalog No. A15982 -
Calcium-Sensing Receptor Antagonists I
Catalog No. A15034 Calcium-Sensing Receptor 拮抗剂Calcium-Sensing Receptor Antagonists I 是钙敏感甲状旁腺激素受体的拮抗剂。 了解更多 -
TGR5-Receptor-Agonist
Catalog No. A13732 TGR5(GPCR19) 激动剂TGR5 Receptor Agonist是一种有效的TGR5（GPCR19）激动剂，在U2-OS细胞分析（pEC50 = 6.8）和黑素细胞（pEC50 = 7.5）中显示出增强的效力。 了解更多 -
Toll-Like Receptor 7 Ligand II
Catalog No. A12683 TLR7 LigandToll-Like Receptor 7 Ligand II是一种细胞可渗透的羟基腺嘌呤化合物，可作为强效且高度特异性的TLR7（toll样受体7）激动剂，对TLR2/3/5/8/9没有任何可检测的活性。它在刺激体外培养物中产生TLR7依赖性细胞因子方面比R848效力高10倍。 了解更多 -
ML-335
Catalog No. A22244 OPRM1(μ-opioid receptor)-OPRD1(δ-opioid receptor) heterodimerization agonistML335 (CYM 51010, CID-23723457) is an agonist for OPRM1(μ-opioid receptor)-OPRD1(δ-opioid receptor) heterodimerization with EC50 of 403 nM demonstrating selectivity over the individual OPRM1 and OPRD1 receptors and the serotonin HT5A receptor with EC50 of 14.9 μM, 1.1 μM, and >40 μM, respectively. 了解更多 -
AMPA Receptor Modulator-1
Catalog No. A19659 TARP γ-8 negative modulatorAMPA Receptor Modulator-1 is a potent, oral active and selective AMPAR regulatory protein TARP γ-8 negative modulator with a pIC50 of 9.7, more selective over GluA1/γ-2 (pIC50=5). 了解更多 -
Pardoprunox hydrochloride
Catalog No. A21624 partial dopamine D2 and D3 receptor agonistPardoprunox hydrochloride is a novel partial dopamine D2 and D3 receptor agonist and serotonin 5-HT1A receptor agonist, D2 (pKi = 8.1) and D3 receptor (pKi = 8.6) partial agonist and 5-HT1A receptor (pKi = 8.5) full agonist. 了解更多 -
Tonapofylline
Catalog No. A21328 adenosine A1 receptor antagonistTonapofylline (BG 9928) is an orally active and selective adenosine A1 receptor antagonist with a Ki of 7.4 nM for human adenosine A1 receptor (hA1), which displays 915-fold selectivity versus human adenosine A2A receptor and 12-fold selectivity versus human adenosine A2B receptor and is used in development for the treatment of heart failure. 了解更多 -
NRA-0160
Catalog No. A20128 Dopamine D4 receptor antagonistNRA-0160 is a selective dopamine D4 receptor antagonist, with a Ki value of 0.48 nM and with negligible affinity for dopamine D2 receptor (Ki: >10000 nM), D3 receptor (Ki: 39 nM), rat 5-HT2A receptor (Ki: 180 nM) and rat α1 adrenoceptor (Ki: 237 nM). 了解更多 -
Toll-like receptor modulator
Catalog No. A15264 Toll-like receptor modulator是一类在先天免疫系统中起关键作用的蛋白质。是一类在先天免疫系统中起关键作用的蛋白质。 了解更多 -
Thrombin Receptor Activator for Peptide 5 (TRAP-5)
Catalog No. A14885 Thrombin Receptor Activator for Peptide 5 (TRAP-5)是一种G蛋白偶联受体，参与调节血栓形成反应。 了解更多 -
Epidermal Growth Factor Receptor Peptide (985-996)
Catalog No. A14877 Epidermal Growth Factor Receptor Peptide (985-996)存在于细胞表面，并通过其特定配体（包括表皮生长因子和转化生长因子）的结合而被激活。 了解更多 -
Betahistine EP Impurity C
Catalog No. A22638 histamine H1 receptor agonist and H3 receptor antagonistBetahistine EP Impurity C (NSC19005) is an impurity of Betahistine. Betahistine is a potent, orally active and well-tolerated histamine H1 receptor agonist and H3 receptor antagonist used for the study of rheumatoid arthritis (RA). 了解更多 -
PF-06291874
Catalog No. A20635 glucagon receptor antagonistPF-06291874 (Glucagon receptor antagonists-4) is a highly potent and orally active glucagon receptor antagonist. It displays low in vivo clearance in both rats and dogs. 了解更多 -
Cipralisant
Catalog No. A20061 histamine H3 receptor antagonistCipralisant is a potent and selective histamine H3 receptor antagonist in vivo, and an agonist in vitro, with a pKi of 9.9 for histamine H3 receptor and a Ki of 0.47 nM for rat histamine H3 receptor; Cipralisant has entered in clinical trials for the treatment of attention-deficit hyperactivity disorder. 了解更多
联系我们
United StatesAdooq Bioscience
Toll Free: (866) 930-6790
Fax: +1-323-606-8156
Email: sales@adooq.com
Not your Region? View all Distributors
FILTER BY:
购物选项
- 分类
-
- Epigenetics (2)
- Apoptosis (9)
- Protein Tyrosine Kinases (21)
- Angiogenesis (15)
- JAK / Stat (7)
- Cell Cycle (1)
- Cytoskeleton (2)
- Cell Metabolism (31)
- Autophagy Signaling (11)
- Immunology & Inflammation (31)
- GPCR / G Protein (493)
- TGF-β / Smad (6)
- Neuronal Signaling (101)
- Proteases (2)
- Microbiology (4)
- Membrane Transporters/Ion Channels (26)
- Endocrinology / Hormones (88)
- PROTACs (5)
- Others (12)
- Natural Products (2)
- Ready to Use Solution (71)
- Products On Sale (131)
- Recombinant Proteins (100)
- Neurotrophins (7)
- Growth Factors (16)
- Hormones (1)
- Monoclonal Antibodies (27)
- Natural Proteins (1)
- Viral Antigens (5)
- CD Antigens (3)
- Cytokines (78)
- Enzymes (42)
- COVID-19 Related Products (1)
- 作用机制
-
- Inhibitor (抑制剂) (109)
- Agonist (激动剂) (292)
- Antagonist (拮抗剂) (471)
- Activator (激活剂) (2)
- Modulator (调节剂) (55)
- Blocker (阻断剂) (13)
- Degrader (降解剂) (7)
- Potentiator (增强剂) (2)
- 靶点
-
- A1 adenosine receptor (1)
- A3 adenosine receptor (1)
- Aurora A (1)
- Aurora B (1)
- Aurora C (1)
- COX-1 (1)
- COX-2 (1)
- CSF1R (1)
- CXCL8 (1)
- CXCR1 (1)
- CXCR2 (1)
- CXCR4 (2)
- Ecdysone receptor (1)
- Histamine H1 receptor (1)
ADOOQ 产品质量保证
We promise all products to perform as described.