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Cenicriviroc Mesylate
Catalog No. A17028 CCR2/5 receptors 抑制剂Cenicriviroc(TAK-652,TBR-652)是CCR2和CCR5受体的抑制剂，可使其充当防止病毒进入人细胞的进入抑制剂 了解更多 -
Urapidil
Catalog No. A17074 -
Proxyphylline
Catalog No. A16821 A1 adenosine receptors 拮抗剂Proxyphylline是茶碱的衍生物，由于其心血管特性而被用作支气管扩张剂。它与A2腺苷受体（对于血小板，Ki = 850μM）选择性拮抗A1腺苷受体（对于牛脑，Ki = 82 nM）。 了解更多 -
TIGIT Human
Catalog No. AP1720 T-Cell Immunoreceptor With Ig And ITIM Domains Human Recombinant 了解更多 -
Ro 25-6981 maleate
Catalog No. A13144 -
Vilanterol
Catalog No. A13125 ultra-long-acting β? adrenoreceptor 激动剂Vilanterol是一种新的选择性β2-AR激动剂，PEC50值为10.37±0.05。 了解更多 -
Acebutolol HCl
Catalog No. A16387 -
VU 0364770
Catalog No. A12139 mGlu4 receptors modulatorVU 0364770是mGlu4受体的正变构调节剂，在表达mGlu4的HEK 293细胞中EC50值为290 nM。 了解更多 -
RO 25-6981 maleate
Catalog No. A16083 NMDA receptors blockerRO 25-6981 maleate是含有NR2B亚基的NMDA受体的强效和选择性活性依赖性阻断剂。克隆的受体亚基组合NR1C/NR2B和NR1C/NR2A的IC50值分别为0.009和52 uM。 了解更多 -
Ketanserin tartrate
Catalog No. A13664 5HT2A 拮抗剂Ketanserin tartrate是一种选择性的5-HT receptor拮抗剂。Ketanserin tartrate 也抑制 hERG 电流 (IhERG)，IC50 为 0.11 μM。 了解更多 -
Imidafenacin
Catalog No. A15490 M3 receptors 抑制剂Imidafenacin是一种有效的选择性M3受体抑制剂，Kb为0.317 nM。对M2受体的效力较低（IC50 = 4.13 nM）。 了解更多 -
CIQ
Catalog No. A15523 -
SB-505124 HCl
Catalog No. A15232 -
BRL 37344 Na Salt
Catalog No. A13676 -
Labetalol HCl
Catalog No. A14239 alpha1/beta adrenergic receptors 拮抗剂Labetalol HCl是选择性α1-肾上腺素能受体和非选择性β-肾上腺素能受体的双重拮抗剂。 了解更多 -
NVP-AAM077 Tetrasodium Hydrate (PEAQX)
Catalog No. A14071 -
CVT 6883
Catalog No. A13745 -
2-Hydroxysaclofen
Catalog No. A13696 -
VU 0361737
Catalog No. A12467 mGlu4 receptors modulatorVU 0361737是mGluR-4的选择性正变构调节剂（人和大鼠受体的EC50值分别为240和110 nM）。 了解更多 -
Bisoprolol
Catalog No. A13406 Bisoprolol是心脏选择性β1-adrenergic receptor阻滞剂，用于阻止心肌梗死、心力衰竭、心绞痛和轻中度高血压。 了解更多 -
LY 255283
Catalog No. A13090 -
Oxybutynin
Catalog No. A10684 Oxybutynin (Ditropan)是一种抗胆碱能药物，是一种竞争性的muscarinic acetylcholine receptorM1，M2，和M3拮抗剂，用于缓解尿道和膀胱疾病。 了解更多 -
Ondansetron HCl (GR 38032F)
Catalog No. A10674 5-HT Receptors 拮抗剂Ondansetron HCl (GR 38032F)是5-羟色胺5-HT3受体拮抗剂，主要用作止吐药，通常在化疗后用于治疗恶心和呕吐。 了解更多 -
Anamorelin
Catalog No. A12346 Anamorelin是一种新型 ghrelin receptor激动剂，FLIPR 检测中，EC50 为 0.74 nM，用于治疗与恶病质/厌食症相关的非小肺癌。 了解更多 -
Chlormezanone (Trancopal)
Catalog No. A10201 Chlormezanone (Trancopal)是一种非苯二氮卓类药物，用于治疗焦虑症。已经建议将其用于治疗肌肉痉挛。氯甲酮与中央苯并二氮杂receptor受体结合，后者与GABA受体发生变构作用。这增强了抑制性神经递质GABA的作用，增强了对网状激活系统的抑制作用，并阻断了在刺激网状通路后发生的皮质和边缘觉醒。 了解更多 -
Calcitriol (Rocaltrol)
Catalog No. A10173 Calcitriol (Rocaltrol)作为vitamin D的激素活性形式，是一种非选择性vitamin D receptor的激活剂，对vitamin D receptor的结合亲和力(IC50=0.4 nM)。 了解更多 -
BRL 52537 HCl
Catalog No. A11210 Opioid Receptors 激动剂BRL 52537 hydrochloride是一种高度选择性和有效的κ阿片类激动剂（Ki = 0.24 nM）。比吗啡强25倍。 了解更多 -
GW3965 HCl
Catalog No. A11204 -
A2A receptor antagonist 1
Catalog No. A12567 adenosine A2A/A1 receptor antagonistA2A receptor antagonist 1 (CPI-444 analog) is an antagonist of both adenosine A2A receptor and A1 receptor with Kis of 4 and 264 nM, respectively. 了解更多 -
Sigma-1 receptor antagonist 2
Catalog No. A18504 sigma 1 receptor antagonistSigma-1 receptor antagonist 2 is a potent and selective sigma 1 receptor (??1 R) antagonist with Kis of 3.88 and 1288 nM for ??1 and ??2 receptor, respectively. 了解更多 -
S1p receptor agonist 1
Catalog No. A20461 S1P receptor agonistS1p receptor agonist 1 is an S1P receptor agonist extracted from patent WO 2015039587 A1, compound example 2. 了解更多 -
Sigma-2 receptor antagonist 1
Catalog No. A20310 sigma-2 (??-2) receptor antagonistSigma-2 receptor antagonist 1 is a sigma-2 (??-2) receptor antagonist. 了解更多 -
Interferon receptor inducer-1
Catalog No. A19877 IFN receptor inducerInterferon receptor inducer-1 (compound 6) is an interferon (IFN) receptor inducer. Used accordingly in the treatment of a disorder in which the induction of interferon is involved. 了解更多 -
Y1 receptor antagonist 1
Catalog No. A19763 neuropeptide Y1 receptor antagonistY1 receptor antagonist 1 (H 409-22 isomer) is a neuropeptide Y1 receptor antagonist. 了解更多 -
Glucagon receptor antagonists-1
Catalog No. A11428 glucagon receptor antagonistGlucagon receptor antagonists-1 is a highly potent glucagon receptor antagonist. 了解更多 -
Glucocorticoid receptor agonist
Catalog No. A11431 Glucocorticoid receptor agonistGlucocorticoid receptor agonist is a potent Glucocorticoid receptor agonist. 了解更多 -
Sigma-1 receptor antagonist 3
Catalog No. A18501 Sigma-1 receptor antagonistSigma-1 receptor antagonist 3 (compound135) is a potent and selective Sigma-1 (??1) receptor antagonist with a Ki of 1.14 nM. 了解更多 -
H4 Receptor antagonist 1
Catalog No. A18929 histamine H4 receptor inverse agonistH4 Receptor antagonist 1 is a potent and selective histamine H4 receptor inverse agonist, with an IC50 of 19 nM. 了解更多 -
Glucagon receptor antagonists-3
Catalog No. A11430 Glucagon receptor antagonistGlucagon receptor antagonists-3 is a highly potent glucagon receptor antagonist. 了解更多 -
Glucagon receptor antagonists-2
Catalog No. A11429 Glucagon receptor antagonistGlucagon receptor antagonists-2 is a highly potent glucagon receptor antagonist. 了解更多 -
GLP-1 receptor agonist 1
Catalog No. A19885 GLP-1 receptor agonistGLP-1 receptor agonist 1 is a glucagon-like peptide-1 (GLP-1) receptor agonist extracted from patent WO2018056453A1, Compound 67. 了解更多 -
GLP-1 receptor agonist 2
Catalog No. A19722 GLP-1R agonistGLP-1 receptor agonist 2 is a glucagon-like peptide-1 receptor (GLP-1R) agonist. 了解更多 -
Orexin 2 Receptor Agonist
Catalog No. A15982 -
Calcium-Sensing Receptor Antagonists I
Catalog No. A15034 Calcium-Sensing Receptor 拮抗剂Calcium-Sensing Receptor Antagonists I 是钙敏感甲状旁腺激素受体的拮抗剂。 了解更多 -
TGR5-Receptor-Agonist
Catalog No. A13732 TGR5(GPCR19) 激动剂TGR5 Receptor Agonist是一种有效的TGR5（GPCR19）激动剂，在U2-OS细胞分析（pEC50 = 6.8）和黑素细胞（pEC50 = 7.5）中显示出增强的效力。 了解更多 -
Toll-Like Receptor 7 Ligand II
Catalog No. A12683 TLR7 LigandToll-Like Receptor 7 Ligand II是一种细胞可渗透的羟基腺嘌呤化合物，可作为强效且高度特异性的TLR7（toll样受体7）激动剂，对TLR2/3/5/8/9没有任何可检测的活性。它在刺激体外培养物中产生TLR7依赖性细胞因子方面比R848效力高10倍。 了解更多 -
ML-335
Catalog No. A22244 OPRM1(μ-opioid receptor)-OPRD1(δ-opioid receptor) heterodimerization agonistML335 (CYM 51010, CID-23723457) is an agonist for OPRM1(μ-opioid receptor)-OPRD1(δ-opioid receptor) heterodimerization with EC50 of 403 nM demonstrating selectivity over the individual OPRM1 and OPRD1 receptors and the serotonin HT5A receptor with EC50 of 14.9 μM, 1.1 μM, and >40 μM, respectively. 了解更多
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