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￥ 0.00 “kinase inhibitor”的搜索结果
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DNA2 inhibitor C5
Catalog No. A19091 DNA2 inhibitorDNA2 inhibitor C5 is a potent, competitive and specific inhibitor of DNA2 nuclease activity with an IC50 of 20 μM. 了解更多 -
B-Raf inhibitor 1 dihydrochloride
Catalog No. A21834 Raf kinase inhibitorB-Raf inhibitor 1 dihydrochloride is a potent Raf kinase inhibitor with Kis of 1 nM, 1 nM, and 0.3 nM for B-RafWT, B-RafV600E, and C-Raf, respectively. 了解更多 -
ITK inhibitor 2
Catalog No. A19096 ITK inhibitorITK inhibitor 2 is a interleukin-2-inducible T-cell kinase (ITK) inhibitor extracted from patent WO2011065402A1, compound 4, with an IC50 of 2 nM. 了解更多 -
Aurora inhibitor 1
Catalog No. A19637 Aurora inhibitorAurora inhibitor 1 is a potent Aurora inhibitor with an IC50 of ?? 4 nM and ??13 nM for Aurora A and Aurora B kinase, respectively. 了解更多 -
GSK-3β inhibitor 1
Catalog No. A19186 GSK-3β inhibitorGSK-3β inhibitor 1 (compound 3a) is a glycogen synthase kinase 3β (GSK-3β) inhibitor and demonstrates high antidiabetic efficacy, with an IC50 of 4.9 nM. 了解更多 -
JAK3 covalent inhibitor-1
Catalog No. A18926 JAK3 covalent 抑制剂JAK3 covalent inhibitor-1 is a potent and selective janus kinase 3 (JAK3) covalent inhibitor with an IC50 of 11 nM and shows 246-fold selectivity vs other JAKs. 了解更多 -
Tyrosine kinase-IN-1
Catalog No. A12486 multi-targeted tyrosine kinase inhibitorTyrosine kinase-IN-1 is a multi-targeted tyrosine kinase inhibitor with IC50s of 4, 20, 4, 2 nM for KDR, Flt-1, FGFR1 and PDGFRα, respectively. 了解更多 -
Tyrosine kinase inhibitor
Catalog No. A15267 Tyrosine kinase 抑制剂Tyrosine kinase inhibitor是一种抑制酪氨酸激酶的药物。酪氨酸激酶是负责通过信号转导级联反应激活许多蛋白质的酶。 了解更多 -
Sodium Channel inhibitor 2
Catalog No. A20453 sodium channel blockerSodium Channel inhibitor 2 is a sodium channel blocker extracted from patent WO 2004011439 A2, compound 3c. 了解更多 -
NAMPT inhibitor-linker 1
Catalog No. A19922 NAMPT inhibitor-linker 1 is a drug-linker conjugates for ADC, composed of an NAMPT inhibitor as a payload, and a linker. 了解更多 -
NAMPT inhibitor-linker 2
Catalog No. A19912 drug-linker conjugates for ADCNAMPT inhibitor-linker 2 is a drug-linker conjugates for ADC, composed of an NAMPT inhibitor as a payload, and a linker. 了解更多 -
Ubiquitin Isopeptidase Inhibitor I, G5
Catalog No. A12293 apoptosis activatorUbiquitin Isopeptidase Inhibitor I, G5 (NSC 144303) is an apoptosome-independent caspase and apoptosis activator with IC50 values of 1.76 and 1.6 μM in E1A and E1A/C9DN cells, respectively. 了解更多 -
Apoptosis Inhibitor (M50054)
Catalog No. A13058 -
PI3K-gamma inhibitor 1
Catalog No. A16275 -
PI3K-alpha inhibitor 1
Catalog No. A16274 PI3Kα 抑制剂PI3K-alpha inhibitor 1 是从专利US/20120088764A1中提取的PI3Kα抑制剂，化合物243，IC50 <0.1uM，PI3Kα抑制剂1还抑制HDAC（0.1uM≤IC50≤1uM）。 了解更多 -
Btk inhibitor 1
Catalog No. A16260 -
c-Met inhibitor 2
Catalog No. A16256 -
PDK1 inhibitor
Catalog No. A16185 PDK1 抑制剂PDK1 inhibitor，强效，ATP竞争性和选择性双重PI3K和PDPK1抑制剂（PDK1和p-T308-PKB抑制的IC50值分别为34 nM和94 nM。 了解更多 -
K+ Channel inhibitor
Catalog No. A16182 -
HIF-2a Translation Inhibitor
Catalog No. A16181 HIF-2a translation 抑制剂HIF-2a Translation Inhibitor（IC50值为5 uM）；独立于HIF-2a mRNA表达或HIF-2a蛋白稳定性，并独立于mTOR活性，降低常氧和低氧状态下HIF-2a蛋白和HIF-2a目标基因的表达。此外，翻译抑制剂76增强了IRP1与HIF-2a IRE（铁反应元件）的结合。 了解更多 -
Cathepsin Inhibitor 1
Catalog No. A11466 Cathepsin 抑制剂Cathepsin Inhibitor 1抑制剂1 是一种Cathepsin (L, L2, S, K, B)的抑制剂，pIC50分别为7.9、6.7、6.0、5.5和5.2。 了解更多 -
PD1-PDL1 inhibitor 2
Catalog No. A15906 -
IRAK-1-4 Inhibitor I
Catalog No. A11462 IRAK-1-4 Inhibitor I是一种苯并咪唑，它破坏IRAK-1和-4的活性，其IC50值分别为300和200 nM。 了解更多 -
Bax inhibitor peptide V5
Catalog No. A15337 Bax 抑制剂Bax inhibitor peptide V5，Bax易位至线粒体的细胞渗透性合成肽抑制剂；由Ku70设计的一种蛋白质，被认为可抑制Bax的线粒体易位。在体外抑制Bax介导的细胞凋亡。 了解更多 -
Bax inhibitor peptide P5
Catalog No. A15336 Bax 抑制剂Bax inhibitor peptide P5，Bax易位至线粒体的细胞渗透性合成肽抑制剂；由Ku70设计的一种蛋白质，被认为可抑制Bax的线粒体易位。在体外抑制Bax介导的细胞凋亡。 了解更多 -
Sodium Channel inhibitor 1
Catalog No. A15243 -
p53 and MDM2 proteins-interaction-inhibitor racemic
Catalog No. A15202 -
mTOR inhibitor (mTOR-IN-1)
Catalog No. A15175 -
Lck inhibitor 2
Catalog No. A15141 Lck 抑制剂Lck inhibitor 2 是酪氨酸激酶的双苯胺基嘧啶抑制剂，包括LCK，BTK，LYN，SYK和TXK。Lck，Btk，Lyn，Btk和Txk的IC50值分别为13nM，9nM，3nM，26nM和2nM。 了解更多 -
DGAT-1 inhibitor 2
Catalog No. A15067 -
c-Met inhibitor 1
Catalog No. A15049 -
CDK9 inhibitor 2
Catalog No. A15039 -
Carboxypeptidase G2 (CPG2) Inhibitor
Catalog No. A15035 -
Caspase-3/7 Inhibitor I
Catalog No. A14919 Caspase-3/7 抑制剂Caspase-3/7 Inhibitor I是caspase-3（Ki = 60 nM）和caspase-7（Ki = 170 nM）的有效，细胞可渗透且可逆的有效抑制剂。 了解更多 -
Elastase Inhibitor, SPCK
Catalog No. A14913 -
Calpain Inhibitor II, ALLM
Catalog No. A14911 Calpain 抑制剂Calpain Inhibitor II, ALLM是钙蛋白酶I，钙蛋白酶II，组织蛋白酶L和组织蛋白酶B的细胞可渗透抑制剂，Ki值分别为120 nM，230 nM，0.6 nM和100 nM。 了解更多 -
PKA inhibitor fragment (6-22) amide
Catalog No. A14868 -
EGFR Inhibitor
Catalog No. A13673 EGFR 抑制剂EGFR inhibitor是一种可透过细胞的4,6-二取代嘧啶化合物，可选择性抑制EGFR激酶，在体外的IC50值为21 nM，可阻断细胞中的受体自身磷酸化。 了解更多 -
K-Ras(G12C) inhibitor 12
Catalog No. A14227 -
PI3k-delta inhibitor 1
Catalog No. A14109 -
K-Ras(G12C) inhibitor 6
Catalog No. A14103 K-Ras(G12C) 抑制剂K-Ras(G12C) inhibitor 6 是致癌性K-Ras（G12C）的不可逆抑制剂，颠覆了天然核苷酸的偏爱性，使GDP优于GTP。 了解更多 -
NSC 42834(JAK2 Inhibitor V, Z3)
Catalog No. A14132 -
HPGDS inhibitor 1
Catalog No. A12258 -
MDM2 Inhibitor
Catalog No. A13582 -
Bozitinib
Catalog No. A18554 c-MET kinase inhibitorBozitinib (PLB-1001) is a highly selective c-MET kinase inhibitor with blood-brain barrier permeability. Bozitinib (PLB-1001) is a ATP-competitive small-molecule inhibitor, binds to the conventional ATP-binding pocket of the tyrosine kinase superfamily. 了解更多 -
Rho-Kinase-IN-1
Catalog No. A20403 ROCK inhibitorRho-Kinase-IN-1 is a Rho kinase (ROCK) inhibitor (Ki values of 30.5 and 3.9 nM for ROCK1 and ROCK2, respectively) extracted from US20090325960A1, compound 1.008. 了解更多
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