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￥ 0.00 “kinase inhibit”的搜索结果
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Vacuolin-1
Catalog No. A22213 cell-permeable lysosomal exocytosis inhibitorVacuolin-1 is a potent and cell-permeable lysosomal exocytosis inhibitor. 了解更多 -
Theliatinib
Catalog No. A22215 EGFR inhibitorTheliatinib (HMPL-309) is a potent, ATP-competitive, orally active and highly selective EGFR inhibitor with a Ki of 0.05 nM and an IC50 of 3 nM. 了解更多 -
Ticlopidine
Catalog No. A22216 inhibitor of platelet aggregationTiclopidine (Yuclid, Ticlopidinum, Ticlopidina) is an orally active inhibitor of platelet aggregation induced by adenosine diphosphate (ADP). 了解更多 -
S29434
Catalog No. A22217 inhibitor of quinone reductase 2 (QR2)S29434 (NMDPEF) is a potent, competitive, selective and cell-permeable inhibitor of quinone reductase 2 (QR2), with IC50s ranging from 5 to 16 nM for human QR2 at different organizational levels, and has good selectivity for QR2 over QR1. 了解更多 -
GC376 sodium
Catalog No. A22221 -
LMPTP INHIBITOR 1 dihydrochloride
Catalog No. A22227 LMPTP inhibitorLMPTP INHIBITOR 1 (dihydrochloride) is a selective inhibitor of low molecular weight protein tyrosine phosphatase (LMPTP), with an IC50 of 0.8 μM LMPTP-A. 了解更多 -
KN-93 phosphate
Catalog No. A22229 membrane-permeant synthetic inhibitorKN-93 phosphate is a novel membrane-permeant synthetic inhibitor of purified neuronal CaMK-II, with Ki of 370 nM. 了解更多 -
Enocitabine
Catalog No. A22234 DNA replication inhibitorEnocitabine is a nucleoside analog, and is a potent DNA replication inhibitor, and a DNA chain terminator. 了解更多 -
Cl-amidine TFA
Catalog No. A22235 peptidylarginine deminase (PAD) inhibitorCl-amidine TFA is an orally active peptidylarginine deminase (PAD) inhibitor, with IC50 values of 0.8 μM, 6.2 μM and 5.9 μM for PAD1, PAD3, and PAD4, respectively. 了解更多 -
Taletrectinib
Catalog No. A22237 ROS1/NTRK inhibitorTaletrectinib (DS-6051b) is a potent, orally active, and new-generation selective ROS1/NTRK inhibitor. 了解更多 -
LY-3475070
Catalog No. A22239 CD73 InhibitorLY-3475070 is a potent and selective CD73 Inhibitor with IC50 of 28 nM. 了解更多 -
Mobocertinib succinate
Catalog No. A22240 EGFR/HER2 oncogenic mutants inhibitorMobocertinib succinate (TAK-788 succinate) is a potent and orally active inhibitor of EGFR and HER2 oncogenic mutants, including exon 20 insertions, with selectivity over WT EGFR. Antitumor activity. 了解更多 -
TSPC (HUN86320)
Catalog No. A22250 inhibitor for GA perceptionTSPC is an inhibitor for GA perception by in vitro and in planta evaluations. 了解更多 -
Propachlor
Catalog No. A22260 LDH1A1 inhibitorPropachlor is a specific ALDH1A1 inhibitor. It is sometimes used as an herbicide. 了解更多 -
Iso-H7 dihydrochloride
Catalog No. A22368 inhibitor of phosphokinase CIso-H7 dihydrochloride is an inhibitor of phosphokinase C. 了解更多 -
SAR-020106
Catalog No. A22371 CHK1 inhibitorSAR-020106 is an ATP-competitive, potent, and selective CHK1 inhibitor with an IC50 of 13.3 nM for human CHK1. 了解更多 -
Nemiralisib
Catalog No. A22373 PI3Kδ inhibitorNemiralisib (GSK2269557 free base) is a potent and highly selective PI3Kδ inhibitor with a pKi of 9.9. 了解更多 -
Tirabrutinib hydrochloride
Catalog No. A22375 BTK inhibitorTirabrutinib (ONO-4059) hydrochloride is a selective and novel inhibitor of BTK with IC50 2.2 nm, Tirabrutinib binds to BTK within B cells, thereby preventing B-cell receptor signaling and impeding B-cell development. 了解更多 -
Miransertib hydrochloride
Catalog No. A22376 Akt inhibitorMiransertib hydrochloride (ARQ-092 hydrochloride) is a potent, orally active, selective and allosteric Akt inhibitor with IC50s of 2.7 nM, 14 nM and 8.1 nM for Akt1, Akt2, Akt3, respectively. 了解更多 -
PF-06273340
Catalog No. A22377 pan-Trk inhibitorPF-06273340 is a highly potent, kinases elective, well-tolerated pan-Trk inhibitor with IC50 values of 6, 4, 3 nM for TrkA, TrkB, Trk C, respectively. 了解更多 -
VPS34 inhibitor 1 (Compound 19)
Catalog No. A22378 VPS34 inhibitorVPS34 inhibitor 1 (Compound 19, PIK-III analogue) is a potent and selective inhibitor of VPS34 with an IC50 of 15 nM. 了解更多 -
UK-371804 HCl
Catalog No. A22379 uPA inhibitorUK-371804 is a potent and selective urokinase-type plasmogen activator (uPA) inhibitor with excellent enzyme potency (Ki=10 nM) and selectivity profile (4000-fold versus tPA and 2700-fold versus plasmin). 了解更多 -
Selective PI3Kδ Inhibitor 1 (compound 7n)
Catalog No. A22381 PI3Kδ inhibitorSelective PI3Kδ Inhibitor 1 (compound 7n) is an inhibitor of PI3Kδ with an IC50 of 0.9 nM and >1000-fold selectivity against other class I PI3K isoforms [PI3K α/γ/β=3670/1460/21300 nM]. 了解更多 -
Gambogenic acid
Catalog No. A22383 EZH2 inhibitorGambogenic acid is an active ingredient in gamboge, with anticancer activity. Gambogenic acid acts as an effective inhibitor of EZH2, specifically and covalently binds to Cys668 within the EZH2-SET domain, and induces EZH2 ubiquitination. 了解更多 -
Cyasterone
Catalog No. A22387 EGFR inhibitorCyasterone, a natural EGFR inhibitor, mainly isolated from Ajuga decumbens Thunb (Labiatae). 了解更多 -
ZM323881 hydrochloride
Catalog No. A22392 VEGFR2 inhibitorZM323881 hydrochloride is a potent and selective VEGFR2 inhibitor with an IC50 of less than 2 nM. 了解更多 -
2,3-Butanedione-2-monoxime
Catalog No. A22395 inhibitor of skeletal muscle myosin-II2,3-Butanedione monoxime (BDM, Diacetyl monoxime, Diacetylmonoxime) is the well-characterized, low-affinity, non-competitive inhibitor of skeletal muscle myosin-II and inhibits skeletal and cardiac muscle contraction. 了解更多 -
Norcantharidin
Catalog No. A22396 dual inhibitor for c-Met and EGFRNorcantharidin (Endothall anhydride) is a synthetic anticancer compound which is a dual inhibitor for c-Met and EGFR in human colon cancers. 了解更多 -
2,5-Dihydroxybenzoic acid
Catalog No. A22397 inhibitor of fibroblast growth factors2,5-Dihydroxybenzoic acid is a derivative of benzoic and a powerful inhibitor of fibroblast growth factors. 了解更多 -
Ginsenoside Re
Catalog No. A22398 antiinflammation agentGinsenoside Re (Ginsenoside B2) is an extract from Panax notoginseng. Ginsenoside Re decreases the β-amyloid protein (Aβ). Ginsenoside Re plays a role in antiinflammation through inhibition of JNK and NF-κB. 了解更多 -
Stylopine
Catalog No. A22400 -
Liensinine
Catalog No. A22404 autophagy/mitophagy inhibitorLiensinine is an autophagy/mitophagy inhibitor. Liensinine, a major isoquinoline alkaloid, extracted from the seed embryo of Nelumbo nucifera Gaertn, has a wide range of biological activities, including anti-arrhythmias, anti-hypertension, anti-pulmonary fibrosis, relaxation on vascular smooth muscle, etc. 了解更多 -
(E/Z)-BCI
Catalog No. A22405 dual-specificity phosphatase 6 (DUSP6) inhibitor(E/Z)-BCI (NSC 150117) is a dual-specificity phosphatase 6 (DUSP6) inhibitor with anti-inflammatory activities. (E/Z)-BCI attenuates LPS-induced inflammatory mediators and ROS production in macrophage cells via activating the Nrf2 signaling axis and inhibiting the NF-κB pathway. 了解更多
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