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Bitopertin
Catalog No. A15021 -
Bitopertin (R enantiomer)
Catalog No. A15022 -
LY2365109 hydrochloride
Catalog No. A21779 GlyT1 inhibitorLY2365109 hydrochloride is a potent and selective GlyT1 inhibitor, with an IC50 of 15.8 nM for glycine uptake in cells over-expressing hGlyT1a. 了解更多 -
Prasugrel (Effient)
Catalog No. A10748 platelet inhibitorPrasugrel (Effient)是一种新型的血小板抑制剂，用于减少急性冠脉综合征（PCI）患者的血栓性心血管事件（包括支架血栓形成）。 了解更多 -
Clopidogrel
Catalog No. A21206 platelet inhibitorClopidogrel is a well-known and orally active platelet inhibitor that targets P2Y12 receptor. Clopidogrel is used to inhibit blood clots in coronary artery disease, peripheral vascular disease, and cerebrovascular disease. 了解更多 -
Cangrelor Tetrasodium
Catalog No. A17919 P2Y12 receptors inhibitorCangrelor Tetrasodium is a high-affinity, reversible inhibitor of P2Y12 receptors that causes almost complete inhibition of ADP-induced platelet aggregate. It is a modified ATP derivative stable to enzymatic degradation. Unlike clopidogrel (Plavix), which is a prodrug, cangrelor is an active drug not requiring metabolic conversion. 了解更多 -
Clopidogrel thiolactone
Catalog No. A20862 P2Y12 receptor inhibitorClopidogrel thiolactone is a P2Y12 receptor inhibitor, is a potent antiplatelet agent. 了解更多 -
Adiphenine HCl
Catalog No. A11716 -
EVP-6124 (Encenicline)
Catalog No. A15086 nAChR 抑制剂EVP-6124 (Encenicline)是α7神经元烟碱乙酰胆碱受体（nAChRs）的新型部分激动剂；显示对α7nAChRs的选择性，并且不激活或抑制异聚体α4β2nAChRs。 了解更多 -
EVP-6124 hydrochloride
Catalog No. A15087 nAChR 抑制剂EVP-6124 hydrochloride是一种新型的α7神经元烟碱型乙酰胆碱受体（nAChRs）的部分激动剂。EVP-6124对α7nAChRs具有选择性，并且不激活或抑制异源α4β2nAChRs。 了解更多 -
Benzethonium Chloride
Catalog No. A13653 nAChR 抑制剂Benzethonium Chloride是nAChRs的有效抑制剂，可抑制α4β2nAChRs和α7nAChRs，IC50分别为49 nM和122 nM。 了解更多 -
Imidafenacin
Catalog No. A15490 M3 receptors 抑制剂Imidafenacin是一种有效的选择性M3受体抑制剂，Kb为0.317 nM。对M2受体的效力较低（IC50 = 4.13 nM）。 了解更多 -
Anisodamine
Catalog No. A18215 alpha-1 adrenergic receptors / mAChRs inhibitorAnisodamine is an inhibitor of alpha-1 adrenergic receptors and mAChRs isolated from Chinese solanacea plant. 了解更多 -
Darenzepine
Catalog No. A12333 muscarinic receptor inhibitorDarenzepine is a muscarinic receptor inhibitor extracted from patent US 20170095465 A1. 了解更多 -
Galanthamine hydrobromide
Catalog No. A10416 -
Rivastigmine tartrate
Catalog No. A11719 AChE 抑制剂Rivastigmine tartrate是一种双重胆碱酯酶抑制剂(ChEI)。它同时抑制丁酰胆碱酯酶(BChE)和乙酰胆碱酯酶(AChE)。 了解更多 -
Donepezil hydrochloride
Catalog No. A10330 -
Neostigmine bromide (Prostigmin)
Catalog No. A10635 -
Deoxyvasicine HCl
Catalog No. A13925 -
Acotiamide hydrochloride trihydrate
Catalog No. A15782 AChE 抑制剂Acotiamide hydrochloride trihydrate是一种在日本获准用于治疗餐后饱胀，上腹胀气和功能性消化不良引起的早饱的药物。 了解更多 -
Rivastigmine
Catalog No. A14096 -
Tacrine HCl Hydrate
Catalog No. A16970 AChE and BChE 抑制剂Tacrine hydrochloride hydrate是乙酰（AChE）和丁酰胆碱酯酶（BChE）的抑制剂，IC50分别为31 nM和25.6 nM。 了解更多 -
Pitofenone Hydrochloride
Catalog No. A17053 -
Tacrine HCl
Catalog No. A17374 AChE & butyrylcholinesterase inhibitorTacrine is a derivative of aminoacridine that functions as an inhibitor of both acetylcholinesterase (AChE) and butyrylcholinesterase (IC50s = 31 and 26.5 nM, respectively). 了解更多 -
Edrophonium chloride
Catalog No. A17794 acetylcholinesterase inhibitorEdrophonium Chloride, also known as Tensilon, is an acetylcholinesterase inhibitor used in cardiac arrhythmias and in the diagnosis of myasthenia gravis. Edrophonium Chloride has also been used as an antidote to curare principles. 了解更多 -
Galanthamine
Catalog No. A12483 AChE inhibitorGalanthamine is a potent acetylcholinesterase (AChE) inhibitor with an IC50 of 500 nM. 了解更多 -
Acetyllovastatin
Catalog No. A19111 AChE inhibitorAcetyllovastatin, a acetate of Lovastatin, presentes a moderate inhibitory effect against the enzyme acetylcholinesterase with an IC50 of 79 μg/mL. Lovastatin has been found to display antifungal activity, and suppresses proliferation of a number of transformed cell lines. 了解更多 -
(R)-Rivastigmine D6 tartrate
Catalog No. A21454 cholinesterase inhibitor(R)-Rivastigmine D6 (tartrate) is the deuterium labeled (R)-Rivastigmine, which is an cholinesterase inhibitor. 了解更多 -
(+)-Phenserine
Catalog No. A20993 cholinesterase noncompetitive inhibitor(+)-Phenserine is a novel selective cholinesterase noncompetitive inhibitor with an IC50 of 45.3 μM. 了解更多 -
(±)-Huperzine A
Catalog No. A21003 AChE inhibitor(??)-Huperzine A, an active Lycopodium alkaloid extracted from traditional Chinese herb, is a potent, selective and reversible acetylcholinesterase (AChE) inhibitor and has been widely used in China for the treatment of Alzheimer's disease (AD). 了解更多 -
KN-62
Catalog No. A11473 -
CID 2011756
Catalog No. A12416 -
kb NB 142-70
Catalog No. A12423 -
Phenoxybenzamine hydrochloride
Catalog No. A10719 α-adrenergic (AR) 拮抗剂/CaM 抑制剂Phenoxybenzamine hydrochloride是一种细胞可渗透的，非特异性的，不可逆的α-肾上腺素（AR）拮抗剂，也可作为CaM抑制剂。 了解更多 -
CID 755673
Catalog No. A13804 PKD 抑制剂CID755673是一种具有细胞活性的泛PKD1/2/3抑制剂，IC50值分别为180 nM，280nM，以及227 nM。 了解更多 -
KN-93 Phosphate
Catalog No. A14288 CaMKII 抑制剂KN-93 Phosphate是一种有效且特异性的Ca2+/钙调蛋白依赖性蛋白激酶II（CaMKII）抑制剂，Ki为0.37μM，对APK，PKC，MLCK或Ca2+-PDE活性无明显抑制作用。 了解更多 -
K252a
Catalog No. A13897 -
A-484954
Catalog No. A13447 -
KN-92 hydrochloride
Catalog No. A15138 -
KN-92 phosphate
Catalog No. A15139 CaMKII 抑制剂KN-92 phosphate是KN-93的非活性衍生物。KN-93是Ca2+/钙调蛋白依赖性激酶II（CaMKII）的选择性抑制剂，竞争性阻断CaM与激酶的结合（Ki = 370 nM）。 了解更多 -
CID 797718
Catalog No. A13809 PKD1 抑制剂CID797718是CID755673（Adooq目录号A13804）的结构类似物。它是效力降低10倍的PKD1抑制剂，IC50值为7.0+/-0.8 uM。 了解更多 -
CRT-0066101
Catalog No. A16318 PKD 抑制剂CRT-0066101是有效，选择性的蛋白激酶D（PKD）抑制剂；抑制所有PKD同工型（PKD1，PKD3和PKD2的IC50值分别为1、2和2.5 nM）。 了解更多
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