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靶点信息
Akt1 | Akt2 | Akt3 | ||
58 nM | 210 nM | 2119 nM |
In vitro | DMSO | 19 mg/mL (34.44 mM) | |
Water | Insoluble | ||
Ethanol | Insoluble | ||
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations. |
Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
---|---|---|---|
0.1 mM | 18.13 mL | 90.65 mL | 181.29 mL |
0.5 mM | 3.63 mL | 18.13 mL | 36.26 mL |
1 mM | 1.81 mL | 9.06 mL | 18.13 mL |
5 mM | 0.36 mL | 1.81 mL | 3.63 mL |
*The above data is based on the productmolecular weight 551.6 . Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.
目录号 | A11286 |
---|---|
作用机制 | Inhibitor (抑制剂) |
M. Wt | 551.6 |
Formula | C34H29N7O |
Purity | >99% |
Storage | Store lyophilized at -20ºC, keep desiccated. |
CAS No. | 612847-09-3 |
SMILES | C1CN(CCC1N2C3=CC=CC=C3NC2=O)CC4=CC=C(C=C4)C5=NC6=CC7=C(C=C6N=C5C8=CC=CC=C8)N=CN7 |
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Product Questions
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