“glucagon receptor”的搜索结果

产品 1 到 50 共 59个

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  1. Ketanserin tartrate

    Catalog No. A13664
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    5HT2A 拮抗剂
    Ketanserin tartrate是一种选择性的5-HT receptor拮抗剂。Ketanserin tartrate 也抑制 hERG 电流 (IhERG),IC50 为 0.11 μM。 了解更多
  2. Ondansetron HCl (GR 38032F)

    Catalog No. A10674
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    5-HT Receptors 拮抗剂
    Ondansetron HCl (GR 38032F)是5-羟色胺5-HT3受体拮抗剂,主要用作止吐药,通常在化疗后用于治疗恶心和呕吐。 了解更多
  3. Masupirdine mesylate

    Catalog No. A21409
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    5-HT6 receptor antagonist
    Masupirdine mesylate (SUVN-502 mesylate) is a potent, selective, orally bioavailable, and brain penetrant 5-HT6 receptor antagonist (Ki of 2.04 nM for human 5-HT6 receptor). 了解更多
  4. Ziprasidone D8

    Catalog No. A21989
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    5-HT / dopamine receptor antagonist
    Ziprasidone D8 is deuterium labeled Ziprasidone, which is a combined 5-HT (serotonin) and dopamine receptor antagonist which exhibits potent effects of antipsychotic activity. 了解更多
  5. Eplivanserin mixture

    Catalog No. A21987
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    serotonin reuptake inhibitor/5-HT2A receptor antagonist
    Eplivanserin mixture is a selective serotonin reuptake inhibitor and a 5-HT2A receptor antagonist, extracted from patent WO 2005/002578 A1. 了解更多
  6. Ritanserin

    Catalog No. A21976
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    5-HT2 receptor antagonist
    Ritanserin (R 55667) is a highly potent, relatively selective, orally active, long acting antagonist of 5-HT2 receptor, with an IC50 of 0.9 nM, less active on Histamine H1, Dopamine D2, Adrenergic α1, Adrenergic α2 receptors. 了解更多
  7. SB-224289 hydrochloride

    Catalog No. A21920
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    5-HT1B receptor antagonist
    SB-224289 hydrochloride is a selective 5-HT1B receptor antagonist, with anxiolytic effect. 了解更多
  8. SB-269970 hydrochloride

    Catalog No. A21889
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    5-HT7 receptor antagonist
    SB269970 hydrochloride (SB-269970A) is a hydrochloride salt form of SB-269970, which is a 5-HT7 receptor antagonist with the pKi of 8.3, exhibits >50-fold selectivity against other receptors. 了解更多
  9. SB 242084

    Catalog No. A21715
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    5-HT2C receptor antagonist
    SB 242084 is a 5-HT2C receptor antagonist(pKi=9.0) that displays 158- and 100-fold selectivity over 5-HT2A and 5-HT2B receptors respectively. 了解更多
  10. SB 242084 hydrochloride

    Catalog No. A21349
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    5-HT2C receptor antagonist
    SB 242084 hydrochloride is a 5-HT2C receptor antagonist(pKi=9.0) that displays 158- and 100-fold selectivity over 5-HT2A and 5-HT2B receptors respectively. 了解更多
  11. RS 127445

    Catalog No. A21256
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    5-HT2B receptor antagonist
    RS 127445 is a novel high affinity, selective 5-HT2B receptor antagonist with pKi of 9.5. 了解更多
  12. Ziprasidone hydrochloride

    Catalog No. A16790
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    5-HT (serotonin)/dopamine receptor antagonist
    Ziprasidone Hcl(CP-88059 Hcl) is a combined 5-HT (serotonin) and dopamine receptor antagonist which exhibits potent effects of antipsychotic activity. 了解更多
  13. WAY-100635 Maleate

    Catalog No. A16787
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    5-HT1A receptor antagonist
    WAY-100635 maleate is a potent and selective 5-hydroxytryptamine 1A (5-HT1A) receptor antagonist with an IC50 value of 0.91 nM and Ki value of 0.39 nM. 了解更多
  14. SB 271046 Hydrochloride

    Catalog No. A11573
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    5-HT6 receptor antagonist
    SB271046 Hydrochloride is a potent, selective and orally active 5-HT6 receptor antagonist with pKi of 8.9. 了解更多
  15. Pancopride

    Catalog No. A12967
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    5-HT3 receptor antagonist
    Pancopride is a new potent and selective 5-HT3 receptor antagonist. 了解更多
  16. Ziprasidone hydrochloride monohydrate

    Catalog No. A11008
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    5-HT (serotonin) and dopamine receptor antagonist
    Ziprasidone hydrochloride monohydrate (CP 88059 hydrochloride monohydrate) is a combined 5-HT (serotonin) and dopamine receptor antagonist which exhibits potent effects of antipsychotic activity. 了解更多
  17. 5-HT4 antagonist 1

    Catalog No. A12268
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    5-HT4 receptor antagonist
    5-HT4 antagonist 1 is a 5-HT4 receptor antagonist with a pKi of 9.6. 了解更多
  18. lumateperone Tosylate

    Catalog No. A12279
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    5-HT2A receptor antagonist
    Lumateperone Tosylate is a 5-HT2A receptor antagonist (Ki = 0.54 nM), a partial agonist of presynaptic D2 receptors and an antagonist of postsynaptic D2 receptors (Ki = 32 nM), and a SERT blocker (Ki = 61 nM). 了解更多
  19. Alosetron (Hydrochloride(1:X))

    Catalog No. A11309
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    Serotonin 5HT3-receptor antagonist
    Alosetron Hydrochloride(1:X) (GR 68755 Hydrochloride(1:X)) is a Serotonin 5HT3-receptor antagonist that is used in treatment of irritable bowel syndrome. 了解更多
  20. Alprenolol hydrochloride

    Catalog No. A17781
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    5-HT1A receptor antagonist
    Alprenolol (hydrochloride) is a non-selective beta blocker as well as 5-HT1A receptor antagonist. 了解更多
  21. Dolasetron Mesylate

    Catalog No. A17729
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    5-HT3 receptor antagonist
    Dolasetron mesylate is a selective 5-HT3 receptor antagonist. 了解更多
  22. Dolasetron

    Catalog No. A17595
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    5-HT3 receptor antagonist
    Dolasetron is a serotonin 5-HT3 receptor antagonist used to treat nausea and vomiting following chemotherapy. Its main effect is to reduce the activity of the vagus nerve, which is a nerve that activates the vomiting center in the medulla oblongata. It does not have much antiemetic effect when symptoms are due to motion sickness. 了解更多
  23. Deramciclane

    Catalog No. A13011
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    5-HT2A and 5-HT2C receptors antagonist
    Deramciclane has a high affinity for 5-HT2A and 5-HT2C receptors; it acts as an antagonist at both receptor subtypes and has inverse agonist properties at the 5-HT2C receptors without direct stimulatory agonist. 了解更多
  24. Pizotifen

    Catalog No. A18107
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    5-HT receptor antagonist
    Pizotifen is a serotonin antagonist which acts mainly at the 5-HT1, 5-HT2A, and 5HT2C receptors with some antihistamine activity. 了解更多
  25. Volinanserin

    Catalog No. A17115
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    5-HT2A receptor 拮抗剂
    Volananserin是高度选择性的5-HT2A受体拮抗剂。 了解更多
  26. Flopropione

    Catalog No. A16550
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    5-HT1A receptor antagonist/COMT inhibitor
    Flopropione是5-HT1A受体拮抗剂,也是儿茶酚-邻甲基转移酶(COMT)抑制剂。 了解更多
  27. Azasetron HCl

    Catalog No. A16417
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    5-HT3 receptor 拮抗剂
    Azasetron HCl是一种选择性的5-HT3受体拮抗剂,IC50为0.33 nM,用于治疗癌症化学疗法引起的恶心和呕吐。 了解更多
  28. GSK163090

    Catalog No. A15838
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    5-HT1A/B/D receptor 拮抗剂
    GSK163090是一种有效的,选择性的,活性的5-HT1A/B/D受体拮抗剂,对于5-HT1A/B/D和多巴胺D2/D3,pKi分别为9.4/8.5/9.7和6.3/6.7。 了解更多
  29. SB271046

    Catalog No. A15438
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    5-HT Receptor 拮抗剂
    SB271046 是一种有效的,选择性的5-HT6受体拮抗剂,pKi为8.9,与其他5-HT受体亚型相比,选择性高200倍。 了解更多
  30. Lerisetron

    Catalog No. A15501
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    5HT3 receptor 拮抗剂
    Lerisetron是具有止吐活性的3型血清素(5-HT3)受体拮抗剂。 了解更多
  31. Ricasetron

    Catalog No. A15499
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    5-HT3 receptor 拮抗剂
    Ricasetron是在5-羟色胺5-HT3受体上充当选择性拮抗剂的药物。 了解更多
  32. Piboserod

    Catalog No. A15542
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    5-HT4 receptor 拮抗剂
    Piboserod是一种选择性的5-HT(4)受体拮抗剂。 了解更多
  33. Alosetron Hydrochloride

    Catalog No. A14989
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    5HT3-receptor 拮抗剂
    Alosetron Hydrochloride是一种5-羟色胺5HT3受体拮抗剂,可用于治疗肠易激综合症。 了解更多
  34. Ziprasidone

    Catalog No. A15286
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    5-HT/dopamine receptor 拮抗剂
    Ziprasidone是5-HT(5-羟色胺)和多巴胺受体拮抗剂的组合,具有抗精神病活性。 了解更多
  35. Clozapine N-oxide

    Catalog No. A15048
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    5-HT1C receptor 拮抗剂
    Clozapine N-oxide是氯氮平的主要代谢产物,在体外可降低SR-2A(5-HT2血清素受体)密度。 了解更多
  36. NAN-190 hydrobromide

    Catalog No. A13417
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    5-HT1A receptor 拮抗剂
    NAN-190 hydrobromide是一种广泛用于科学研究的药物和研究化学品。以前认为它是一种选择性的5-HT1A受体拮抗剂,但后来的发现表明它也能有效地阻断α2肾上腺素能受体。 了解更多
  37. SB 258585 HCl

    Catalog No. A14026
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    5-HT6 serotonin receptor 拮抗剂
    SB 258585 hydrochloride是一种选择性和有效的SR-6拮抗剂。该化合物显示出比其他5-羟色胺受体亚型高160倍的选择性。 了解更多
  38. Tropisetron HCL

    Catalog No. A14375
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    5-HT3 receptor 拮抗剂
    Tropisetron HCL是选择性的5-HT3受体拮抗剂和α7烟碱样受体激动剂,对5-HT3受体的IC50为70.1±0.9 nM。 了解更多
  39. LuAE58054

    Catalog No. A14356
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    5-HT6 receptor 拮抗剂
    LuAE58054是一种有效且选择性的5-HT6受体拮抗剂,Ki 为 0.83 nM。由伦德贝克(Lundbeck)开发,作为增强疗法,用于治疗与阿尔茨海默氏病和精神分裂症相关的认知缺陷。 了解更多
  40. Cyclobenzaprine HCl

    Catalog No. A14255
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    5-HT2 receptor 拮抗剂
    Cyclobenzaprine HCl是一种肌肉松弛剂,可阻止疼痛感。 了解更多
  41. SB-742457

    Catalog No. A14092
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    5-HT6 receptor 拮抗剂
    SB-742457是一种选择性的5-HT6受体拮抗剂,具有认知,记忆和增强学习的作用。 了解更多
  42. Tandospirone

    Catalog No. A13293
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    5-HT Receptor 拮抗剂
    Tandospirone是5HT1A受体的部分激动剂。它以剂量依赖性方式显着降低氟哌啶醇诱导的运动迟缓。 了解更多
  43. PRX-08066

    Catalog No. A13267
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    5-HT2B receptor 拮抗剂
    PRX-08066是一种新型的5-HT受体2B(5-HT2BR)拮抗剂,IC50为3.4 nM,,可减轻单芥子碱诱导的大鼠肺动脉高压和右室肥大。 了解更多
  44. Blonanserin

    Catalog No. A11824
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    D2/5-HT2 receptor 拮抗剂
    Blonanserin是D2/5-HT2受体拮抗剂。 了解更多
  45. N-Desmethylclozapine

    Catalog No. A13762
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    5-HT2C serotonin receptor 拮抗剂
    N-Desmethylclozapine是一种有效的选择性5-HT2C血清素受体拮抗剂。 了解更多
  46. SDZ 205-557 HCl

    Catalog No. A13766
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    5-HT4 Receptor 拮抗剂
    SDZ 205-557 HCl是一种有效的选择性5-HT4 5-羟色胺受体拮抗剂。 了解更多
  47. Tropanserin

    Catalog No. A13767
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    5-HT3 receptor 拮抗剂
    tropanserin充当有效的选择性5-HT3受体拮抗剂。 了解更多
  48. 5-HT1A receptor 拮抗剂
    NAD 299 hydrochloride (Robalzotan)是一种选择性的,高亲和力的5-HT1A受体拮抗剂(体外Ki = 0.6 nM)。 了解更多
  49. Eletriptan

    Catalog No. A13075
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    5-HT1B receptor 激动剂
    Eletriptan是一种选择性5-羟色胺1B/1D(5-HT1B)受体激动剂。 了解更多
  50. Olanzapine (LY170053)

    Catalog No. A10667
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    5-HT Receptors/D2 dopamine receptor 拮抗剂
    Olanzapine (LY170053)对5-HT2血清素和D2多巴胺受体拮抗剂具有高亲和力。 了解更多

产品 1 到 50 共 59个

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