“glucagon receptor”的搜索结果

产品 51 到 100 共 279个

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  1. Maropitant

    Catalog No. A21473
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    NK1 receptor antagonist
    Maropitant is a neurokinin (NK1) receptor antagonist. 了解更多
  2. (±)-Ibipinabant

    Catalog No. A21439
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    CB-1 receptor antagonist
    (±)-Ibipinabant ((±)-SLV319) is the racemate of SLV319. (±)-Ibipinabant ((±)-SLV319) is a potent and selective cannabinoid-1 (CB-1) receptor antagonist with an IC50 of 22 nM. 了解更多
  3. PF-03654746 Tosylate

    Catalog No. A21434
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    histamine H3 receptor antagonist
    PF-03654746 Tosylate is a potent and selective histamine H3 receptor antagonist with high brain penetration. 了解更多
  4. PF-03654746

    Catalog No. A21429
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    histamine H3 receptor antagonist
    PF-03654746 is a potent and selective histamine H3 receptor antagonist with high brain penetration. 了解更多
  5. RG7713

    Catalog No. A21380
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    Brain-Penetrant Vasopressin 1a (V1a) receptor antagonist
    RG7713 (RO5028442) is a highly potent and selective Brain-Penetrant Vasopressin 1a (V1a) receptor antagonist with Kis of 1 nM (hV1a) and 39 nM (mV1a). 了解更多
  6. SB-277011 dihydrochloride

    Catalog No. A21353
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    dopamine D3 receptor antagonist
    SB-277011 dihydrochloride (SB-277011A dihydrochloride) is a potent, selective, orally bioavailable and brain penetrate dopamine D3 receptor antagonist, with pKis of 8.0, 6.0, <5.2 and 5.9 for D3, D2, 5-HT1B, and 5-HT1D receptors, respectively. 了解更多
  7. SB 242084 hydrochloride

    Catalog No. A21349
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    5-HT2C receptor antagonist
    SB 242084 hydrochloride is a 5-HT2C receptor antagonist(pKi=9.0) that displays 158- and 100-fold selectivity over 5-HT2A and 5-HT2B receptors respectively. 了解更多
  8. Darusentan

    Catalog No. A21280
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    endothelin A (ETA) receptor antagonist
    Darusentan is a selective endothelin A (ETA) receptor antagonist. 了解更多
  9. Lixivaptan

    Catalog No. A21279
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    vasopressin receptor V2 antagonist
    Lixivaptan (VPA-985, WAY-VPA 985) is an orally active and selective vasopressin receptor V2 antagonist, with IC50 values of 1.2 and 2.3 nM for human and rat V2, respectively. 了解更多
  10. RS 127445

    Catalog No. A21256
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    5-HT2B receptor antagonist
    RS 127445 is a novel high affinity, selective 5-HT2B receptor antagonist with pKi of 9.5. 了解更多
  11. Mavoglurant

    Catalog No. A21223
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    mGlu5 receptor antagonist
    Mavoglurant is a structurally novel, non-competitive mGlu5 receptor antagonist, has an IC50 of 30 nM in a functional assay with human mGluR5. 了解更多
  12. LAS101057

    Catalog No. A21203
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    A2B receptor antagonist
    LAS101057 is a potent, selective, and orally efficacious A2B receptor antagonist. 了解更多
  13. Tezosentan

    Catalog No. A21118
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    endothelin (ET) receptor antagonist
    Tezosentan (RO 610612) is an endothelin (ET) receptor antagonist, with pA2s of 9.5, 7.7 for ETA and ETB receptors, respectively. 了解更多
  14. Terutroban

    Catalog No. A20884
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    thromboxane-prostaglandin receptor antagonist
    Terutroban is a thromboxane-prostaglandin receptor antagonist. 了解更多
  15. Sparsentan

    Catalog No. A20879
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    angiotensin II and endothelin A receptor antagonist
    Sparsentan (RE-021) is a highly potent dual angiotensin II and endothelin A receptor antagonist with Kis of 0.8 and 9.3 nM, respectively. 了解更多
  16. Haloperidol hydrochloride

    Catalog No. A18304
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    dopamine D2 receptor antagonist
    Haloperidol hydrochloride is a potent dopamine D2 receptor antagonist, widely used as an antipsychotic. 了解更多
  17. Ziprasidone hydrochloride

    Catalog No. A16790
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    5-HT (serotonin)/dopamine receptor antagonist
    Ziprasidone Hcl(CP-88059 Hcl) is a combined 5-HT (serotonin) and dopamine receptor antagonist which exhibits potent effects of antipsychotic activity. 了解更多
  18. WAY-100635 Maleate

    Catalog No. A16787
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    5-HT1A receptor antagonist
    WAY-100635 maleate is a potent and selective 5-hydroxytryptamine 1A (5-HT1A) receptor antagonist with an IC50 value of 0.91 nM and Ki value of 0.39 nM. 了解更多
  19. SB-334867 free base

    Catalog No. A16695
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    orexin OX1 receptor antagonist
    SB-334867 free base is a selective non-peptide orexin OX1 receptor antagonist with a pKb value of 7.2. 了解更多
  20. SB 271046 Hydrochloride

    Catalog No. A11573
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    5-HT6 receptor antagonist
    SB271046 Hydrochloride is a potent, selective and orally active 5-HT6 receptor antagonist with pKi of 8.9. 了解更多
  21. JDTic

    Catalog No. A11468
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    κ-opioid receptor antagonist
    JDTic is a highly selective antagonist for the κ-opioid receptor; without affecting the μ- or δ-opioid receptors. 了解更多
  22. CP-96486

    Catalog No. A12471
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    LTD4/PAF receptor antagonist
    CP-96486 is a potent and orally active leukotriene D4 (LTD4)/platelet activating factor (PAF) receptor antagonist with Kis of 20 and 24 nM, respectively. 了解更多
  23. Pancopride

    Catalog No. A12967
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    5-HT3 receptor antagonist
    Pancopride is a new potent and selective 5-HT3 receptor antagonist. 了解更多
  24. Foropafant

    Catalog No. A13388
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    PAF receptor antagonist
    Foropafant (SR27417) highly potent, competitive, selective and orally active antagonist of platelet-activating factor (PAF) receptor. 了解更多
  25. Ziprasidone hydrochloride monohydrate

    Catalog No. A11008
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    5-HT (serotonin) and dopamine receptor antagonist
    Ziprasidone hydrochloride monohydrate (CP 88059 hydrochloride monohydrate) is a combined 5-HT (serotonin) and dopamine receptor antagonist which exhibits potent effects of antipsychotic activity. 了解更多
  26. TY-52156

    Catalog No. A12265
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    S1P3 receptor antagonist
    TY-52156 is a potent and selective S1P3 receptor antagonist with a Ki value of 110 nM. 了解更多
  27. 5-HT4 antagonist 1

    Catalog No. A12268
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    5-HT4 receptor antagonist
    5-HT4 antagonist 1 is a 5-HT4 receptor antagonist with a pKi of 9.6. 了解更多
  28. lumateperone Tosylate

    Catalog No. A12279
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    5-HT2A receptor antagonist
    Lumateperone Tosylate is a 5-HT2A receptor antagonist (Ki = 0.54 nM), a partial agonist of presynaptic D2 receptors and an antagonist of postsynaptic D2 receptors (Ki = 32 nM), and a SERT blocker (Ki = 61 nM). 了解更多
  29. Veralipride

    Catalog No. A13132
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    D2 receptor antagonist
    Veralipride is a D2 receptor antagonist. It is an alternative antidopaminergic treatment for menopausal symptoms. 了解更多
  30. GSK598809

    Catalog No. A13695
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    dopamine D3 Receptor (DRD3) antagonist
    GSK598809 is a potent and selective dopamine D3 Receptor (DRD3) antagonist, with a pKi of 8.9. 了解更多
  31. Mozavaptan

    Catalog No. A16622
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    nonpeptide vasopressin V2 receptor antagonist
    Mozavaptan (OPC31260) is a orally effective, nonpeptide vasopressin V2 receptor antagonist with an IC50 of 14 nM. 了解更多
  32. CAY10471 Racemate

    Catalog No. A11760
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    Prostaglandin D2 receptor CRTH2 antagonist
    CAY10471 Racemate (TM30089 Racemate) is a potent and highly selective prostaglandin D2 receptor CRTH2 antagonist. 了解更多
  33. GSK1059865

    Catalog No. A12401
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    orexin 1 receptor antagonist
    GSK1059865 is a potent orexin 1 receptor antagonist. 了解更多
  34. ST3932

    Catalog No. A12880
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    Adenosine A2A receptor antagonist
    ST3932 is a metabolite of ST1535, acts as an antagonist of adenosine A2A receptor, with Kis of 8 nM and 33 nM for A2A and A1 receptors, respectively. 了解更多
  35. GSK1521498 free base

    Catalog No. A18994
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    μ-opioid receptor antagonist
    GSK1521498 free base is a potent and selective μ-opioid receptor (MOR) antagonist. GSK1521498 free base is being used for the treatment of disorders of compulsive consumption of food, alcohol, and drugs. 了解更多
  36. BAY-545

    Catalog No. A20116
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    A2B adenosine receptor antagonist
    BAY-545 is a potent and selective A2B adenosine receptor antagonist, with an IC50 of 59 nM. 了解更多
  37. Alosetron (Hydrochloride(1:X))

    Catalog No. A11309
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    Serotonin 5HT3-receptor antagonist
    Alosetron Hydrochloride(1:X) (GR 68755 Hydrochloride(1:X)) is a Serotonin 5HT3-receptor antagonist that is used in treatment of irritable bowel syndrome. 了解更多
  38. Dexloxiglumide

    Catalog No. A18541
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    CCKA receptor antagonist
    Dexloxiglumide is a selective cholecystokinin type A (CCKA) receptor antagonist. Dexloxiglumide, the active enantiomer of Loxiglumide, inhibits smooth muscle cell contractions induced by cholecystokinin-octapeptide (CCK-8). 了解更多
  39. SHR1653

    Catalog No. A18575
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    Oxytocin receptor antagonist
    SHR1653 is a highly potent, selective and brain penetrated oxytocin receptor (OTR) antagonist, with an IC50 of 15 nM for hOTR. 了解更多
  40. BTRX-335140

    Catalog No. A18583
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    κ opioid receptor antagonist
    BTRX-335140 (CYM-53093) is a potent and selective, orally active κ opioid receptor (KOR) antagonist, has antagonist activity for κOR, μOR and δOR with IC50 values of 0.8 nM, 110 nM, and 6500 nM, respectively. 了解更多
  41. ASP6432

    Catalog No. A18759
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    LPA1 receptor antagonist
    ASP6432 is a potent and selective Type 1 Lysophosphatidic Acid (LPA1) receptor antagonist. 了解更多
  42. A-381393

    Catalog No. A18784
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    Dopamine D4 receptor antagonist
    A-381393 is a potent and selective agonist of the dopamine D4 receptor. 了解更多
  43. Metipranolol hydrochloride

    Catalog No. A18064
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    β-adrenergic receptor antagonist
    Metipranolol (hydrochloride) is a non-selective β-adrenergic receptor (β-AR) antagonist. Formulations containing metipranolol have been used in the treatment of elevated IOP in patients with ocular hypertension or glaucoma. 了解更多
  44. Mebhydrolin napadisylate

    Catalog No. A17997
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    histamine H1-receptor antagonist
    Diazoline is a histamine H1-receptor antagonist. 了解更多
  45. Alprenolol hydrochloride

    Catalog No. A17781
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    5-HT1A receptor antagonist
    Alprenolol (hydrochloride) is a non-selective beta blocker as well as 5-HT1A receptor antagonist. 了解更多
  46. Acrivastine

    Catalog No. A17746
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    Histamine 1 receptor antagonist
    Acrivastine (BW825C) is a short acting histamine 1 receptor antagonist for the treatment of allergic rhinitis. 了解更多
  47. Dolasetron Mesylate

    Catalog No. A17729
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    5-HT3 receptor antagonist
    Dolasetron mesylate is a selective 5-HT3 receptor antagonist. 了解更多
  48. Hydroxyzine pamoate

    Catalog No. A17712
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    Histamine H1 receptor antagonist
    Hydroxyzine pamoate is an histamine H1 receptor antagonist that is effective in the treatment of chronic urticaria, dermatitis, and histamine-mediated pruritus. Unlike its major metabolite CETIRIZINE, it does cause drowsiness. 了解更多
  49. Dolasetron

    Catalog No. A17595
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    5-HT3 receptor antagonist
    Dolasetron is a serotonin 5-HT3 receptor antagonist used to treat nausea and vomiting following chemotherapy. Its main effect is to reduce the activity of the vagus nerve, which is a nerve that activates the vomiting center in the medulla oblongata. It does not have much antiemetic effect when symptoms are due to motion sickness. 了解更多
  50. Melitracen hydrochloride

    Catalog No. A17494
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    dopamine D1/2 receptor antagonist
    Melitracen HCl ia potential dopamine D1/2 receptor antagonist used to treat depression. It is often co-administered with flupenthixol as a treatment for trigeminal neuralgia. It does not effect cardiovascular function. 了解更多

产品 51 到 100 共 279个

每页
页面:
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  2. 2
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