微信关注
China
Total item
Cart Subtotal
￥ 0.00 “Akt Inhibitor”的搜索结果
-
RAF mutant-IN-1
Catalog No. A19011 Raf nhibitorRAF mutant-IN-1 is a RAF kinase inhibitor, extracted from patent WO2019107987A1, with IC50 values of 21 nM, 30 nM and 392 nM for C-RAF340D/Y341D, B-RAFV600E and B-RAFWT, respectively. 了解更多 -
VNRX-5133
Catalog No. A18824 -
Mutated EGFR-IN-2
Catalog No. A18565 EGFR 抑制剂Mutated EGFR-IN-2 (compound 91) is a mutant-selective EGFR inhibitor extracted from patent WO2017036263A1, which potently inhibits single-mutant EGFR (T790M) and double-mutant EGFR (including L858R/T790M (IC50=??1nM) and ex19del/T790M), and can suppress activity of single gain-of-function mutant EGFR (including L858R and ex19del) as well. Mutated EGFR-IN-2 shows anti-tumor antivity. 了解更多 -
Licogliflozin
Catalog No. A12828 SGLT1/SGLT2 抑制剂Licogliflozin is a sodium glucose cotransporter (SGLT1 and SGLT2) inhibitor. 了解更多 -
Amsacrine hydrochloride
Catalog No. A17707 antineoplastic agentAmsacrine hydrochloride (m-AMSA hydrochloride; acridinyl anisidide hydrochloride) is an inhibitor of topoisomerase II, and acts as an antineoplastic agent which can intercalates into the DNA of tumor cells. 了解更多 -
Sorafenib N-Oxide
Catalog No. A12005 Raf kinase inhibitorSorafenib N-Oxide is a metabolite of Sorafenib, a potent Raf kinase inhibitor. 了解更多 -
GSK2292767
Catalog No. A16564 PI3Kδ inhibitorGSK2292767 is a potent and selective inhibitor of phosphatidylinositol 3-kinase δ (PI3Kδ; Ki = 79 pM). GSK2292767 is >100-fold selective for PI3Kδ over a panel of 250 kinases. 了解更多 -
IACS-010759
Catalog No. A12006 IACS-10759 is a potent inhibitor of complex I of oxidative phosphorylation (OXPHOS). 了解更多 -
![N-[(4-Aminophenyl)methyl]adenosine](https://www.adooq.cn/media/catalog/product/cache/1/small_image/9df78eab33525d08d6e5fb8d27136e95/a/1/a12659-n-4-aminophenyl-methyl-adenosine_1.gif)
N-[(4-Aminophenyl)methyl]adenosine
Catalog No. A12659 Adenosine receptor inhibitorN-[(4-Aminophenyl)methyl]adenosine is a adenosine receptor inhibitor, with Ki of 29 nM for Rat ecto-5??-Nucleotidase. IC50 value: 29.0 ± 1.7 nM (Ki) Target: Adenosine Receptor 了解更多 -
(S)-SNAP5114
Catalog No. A12834 GABA transport inhibitor(S)-SNAP5114 is a selective GABA transport inhibitor, with IC50 values of 5 μM and 21 μM for hGAT-3 and rGAT-2, respectively. (S)-SNAP5114 is an anticonvulsant drug. 了解更多 -
Osimertinib dimesylate
Catalog No. A18243 EGFR inhibitorOsimertinib dimesylate (AZD-9291 dimesylate) is an irreversible and mutant selective EGFR inhibitor with IC50s of 12 and 1 nM against EGFRL858R and EGFRL858R/T790M, respectively. 了解更多 -
MtbHU-IN-1
Catalog No. A19132 MtbHU inhibitorMtbHU-IN-1 is an inhibitor of Mycobacterium tuberculosis nucleoid-associated protein HU (MtbHU), with a Kd of 98 nM for binding to WT MtbHU. 了解更多 -
MitoTam bromide, hydrobromide
Catalog No. A19142 ETC inhibitorMitoTam bromide, hydrobromide is a tamoxifen derivative, an electron transport chain (ETC) inhibitor, spreduces mitochondrial membrane potential in senescent cells and affects mitochondrial morphology. 了解更多 -
Autotaxin-IN-1
Catalog No. A19164 autotaxin inhibitorAutotaxin-IN-1 is a potent autotaxin inhibitor, which has favorable potency (IC50=2.2 nM), PK properties, and a robust PK/PD relationship. Autotaxin-IN-1 is used in treatment of osteoarthritis pain. 了解更多 -
2-Iminobiotin
Catalog No. A19175 nitric oxide synthases inhibitor2-Iminobiotin (Guanidinobiotin) is a biotin (vitamin H or B7) analog. 2-Iminobiotin is a reversible nitric oxide synthases inhibitor with Kis of 21.8 and 37.5μM for murine iNOS and rat n-cNOS, respectively. 了解更多 -
BACE1-IN-2
Catalog No. A19194 BACE1 inhibitorBACE1-IN-2 is a 1,4-Oxazine β-Secretase 1 (BACE1) inhibitor with an IC50 of 22 nM. 了解更多 -
3'-Azido-3'-deoxy-5-methylcytidine
Catalog No. A19200 XMRV inhibitor3'-Azido-3'-deoxy-5-methylcytidine (CS-92) is a potent xenotropic murine leukemia-related retrovirus (XMRV) inhibitor with a CC50 of 43.5 μM in MCF-7 cells. 了解更多 -
Fulacimstat
Catalog No. A19202 chymase inhibitorFulacimstat is an orally available chymase inhibitor, with IC50s of 4, 3 nM for human and hamster chymase enzyme, respectively. 了解更多 -
Antifungal agent 2
Catalog No. A19213 fungal inhibitorAntifungal agent 2 is a broad-spectrum fungal inhibitor which inhibits growth of pertinent species of Candida, Cryptococcus, and Aspergillus at a concentration as low as 0.5 μg/mL. 了解更多 -
Enarodustat
Catalog No. A19214 prolyl hydroxylase inhibitorEnarodustat is a potent and orally active factor prolyl hydroxylase inhibitor, with an EC50 of 0.22 μM; Enarodustat has entered clinical trial for renal anemia. 了解更多 -
KAN0438757
Catalog No. A19216 PFKFB3 inhibitorKAN0438757 is a potent and selective inhibitor of the metabolic kinase PFKFB3 with an IC50 of 0.19 μM . 了解更多 -
eIF4A3-IN-2
Catalog No. A19219 eIF4A3 inhibitoreIF4A3-IN-2 is a highly selective and noncompetitive eukaryotic initiation factor 4A-3 (eIF4A3) inhibitor with an IC50 of 110 nM. 了解更多 -
Elenbecestat
Catalog No. A19223 BACE-1 inhibitorElenbecestat (E2609) is a potent, orally bioavailable and CNS-penetrant BACE-1 inhibitor for the treatment of Alzheimer's disease (AD). 了解更多
联系我们
United StatesAdooq Bioscience
Toll Free: (866) 930-6790
Fax: +1-323-606-8156
Email: sales@adooq.com
Not your Region? View all Distributors
最近查看过的产品
ADOOQ 产品质量保证
We promise all products to perform as described.