COX

Catalog No.Inhibitor Name COXCOX-1COX-2Other
A10193Celecoxib
****
A10461Ibuprofen
*
*
A10474Indomethacin
**
*
A11918Rofecoxib
****
A10304Diclofenac Sodium
***
***
A11695Lornoxicam
****
****
A10623Naproxen Sodium
*
*
A13342Valdecoxib
****
A11693Tolfenamic Acid
***
A16399Amfenac Sodium Monohydrate
**
***
A11694Nimesulide
*
A12520Meclofenamate Sodium
****
***
A16428Carprofen
****
A10636Nepafenac
A10878Sulindac
A10565Meloxicam
A10820Aspirin
A11906Phenacetin
A10736Piroxicam
A10462Ibuprofen Lysine
A11641Pranoprofen
A10090Asaraldehyde
A11692Acemetacin
A13244Bromfenac Sodium

Notes:
1.Hover mouse over " * " to view the IC50 value.(A few compounds have proven potency but without published IC50 data.)
2.For more details about the compound, click on the product name of your interest.
3.The higher the number of " * " is, the more potent the inhibitor or activator is.
4."" refers to compounds which do inhibitory effects on the related isoform, but without specific value.

产品 51 到 60 共 60个

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  1. Radicicol

    Catalog No. A11768
    Hsp90/SRC/COX-2 抑制剂
    Radicicol是Hsp90,SRC和Cox-2的有效抑制剂。 了解更多
  2. Flufenamic acid

    Catalog No. A13333
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    COX 抑制剂
    Flufenamic acid是一种非甾体类抗炎药(NSAID)。抑制钙激活的氯离子通道(CaCC)。也增加通过TRPC6通道的电流,并抑制通过TRPC3和TRPC7通道的电流。 了解更多
  3. Pranoprofen

    Catalog No. A11641
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    COX 抑制剂
    Pranoprofen是一种用于眼科的非甾体类抗炎药。 了解更多
  4. (-)-Epicatechin

    Catalog No. A12043
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    COX-1 抑制剂
    (-)-Epicatechin是绿茶的天然产物。(-)表儿茶素是cox-1的抑制剂。 了解更多
  5. SC 560

    Catalog No. A13023
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    COX-1 抑制剂
    SC 560是一种COX-1选择性抑制剂,IC50 值为9 nM。可以用作研究COX-1衍生的PG在炎症和疼痛中的作用的药理学工具。 了解更多
  6. ATB 346

    Catalog No. A13983
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    COX-2 抑制剂
    ATB-346具有类似于萘普生的抗炎特性,但其胃肠道毒性显着降低。 了解更多
  7. Xanthohumol

    Catalog No. A15919
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    COX 抑制剂
    Xanthohumol是一种来自啤酒花的烯丙基查尔酮,可抑制COX-1和COX-2活性并显示化学预防作用。 了解更多
  8. Etoricoxib

    Catalog No. A13770
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    COX-2 抑制剂
    Etoricoxib特异性结合并抑制环氧合酶2(COX-2),从而抑制花生四烯酸向前列腺素的转化。抑制COX-2可以诱导细胞凋亡并抑制肿瘤细胞的增殖和血管生成。 了解更多
  9. Paradol

    Catalog No. A15205
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    COX-1 抑制剂
    Paradol是几内亚胡椒(Aframomum melegueta)种子的活性风味成分。已发现Paradol具有抗氧化和抗肿瘤的促进作用。 了解更多
  10. Meclofenamate Sodium

    Catalog No. A12520
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    COX 抑制剂
    Meclofenamate Sodium是一种双重COX-1/COX-2抑制剂,IC50为40 nM和50 nM。 了解更多

产品 51 到 60 共 60个

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