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Lu AE58054 (Idalopirdine)
Catalog No. A12521 -
Tandospirone
Catalog No. A13293 5-HT Receptor 拮抗剂Tandospirone是5HT1A受体的部分激动剂。它以剂量依赖性方式显着降低氟哌啶醇诱导的运动迟缓。 了解更多 -
SB-742457
Catalog No. A14092 -
SB 399885 HCl
Catalog No. A14102 5-HT6 拮抗剂SB 399885 hydrochloride是一种有效的，脑渗透剂和口服活性的SR-6拮抗剂。它对SR-6的选择性比其他血清素受体高200倍（对于人类重组，天然大鼠和天然人类SR-6受体，pKi值分别为9.11、8.81和9.02）。 了解更多 -
Cyclobenzaprine HCl
Catalog No. A14255 -
Tropisetron HCL
Catalog No. A14375 5-HT3 receptor 拮抗剂Tropisetron HCL是选择性的5-HT3受体拮抗剂和α7烟碱样受体激动剂，对5-HT3受体的IC50为70.1±0.9 nM。 了解更多 -
NAN-190 hydrobromide
Catalog No. A13417 5-HT1A receptor 拮抗剂NAN-190 hydrobromide是一种广泛用于科学研究的药物和研究化学品。以前认为它是一种选择性的5-HT1A受体拮抗剂，但后来的发现表明它也能有效地阻断α2肾上腺素能受体。 了解更多 -
Clozapine N-oxide
Catalog No. A15048 5-HT1C receptor 拮抗剂Clozapine N-oxide是氯氮平的主要代谢产物，在体外可降低SR-2A（5-HT2血清素受体）密度。 了解更多 -
Ziprasidone
Catalog No. A15286 5-HT/dopamine receptor 拮抗剂Ziprasidone是5-HT（5-羟色胺）和多巴胺受体拮抗剂的组合，具有抗精神病活性。 了解更多 -
Alosetron Hydrochloride
Catalog No. A14989 -
Cyproheptadine hydrochloride
Catalog No. A16169 -
Azasetron HCl
Catalog No. A16417 5-HT3 receptor 拮抗剂Azasetron HCl是一种选择性的5-HT3受体拮抗剂，IC50为0.33 nM，用于治疗癌症化学疗法引起的恶心和呕吐。 了解更多 -
LY 334370 hydrochloride
Catalog No. A17027 5-HT1F 激动剂LY 334370 hydrochloride是一种选择性的5-HT1F受体激动剂（Ki值为1.87、16.4，> 100 (IC50)）。CAS：199673-74-0（LY 334370盐酸盐）；182563-08-2（LY 334370游离碱） 了解更多 -
Volinanserin
Catalog No. A17115 -
Dolasetron
Catalog No. A17595 5-HT3 receptor antagonistDolasetron is a serotonin 5-HT3 receptor antagonist used to treat nausea and vomiting following chemotherapy. Its main effect is to reduce the activity of the vagus nerve, which is a nerve that activates the vomiting center in the medulla oblongata. It does not have much antiemetic effect when symptoms are due to motion sickness. 了解更多 -
Dolasetron Mesylate
Catalog No. A17729 5-HT3 receptor antagonistDolasetron mesylate is a selective 5-HT3 receptor antagonist. 了解更多 -
Alprenolol hydrochloride
Catalog No. A17781 5-HT1A receptor antagonistAlprenolol (hydrochloride) is a non-selective beta blocker as well as 5-HT1A receptor antagonist. 了解更多 -
Alosetron (Hydrochloride(1:X))
Catalog No. A11309 Serotonin 5HT3-receptor antagonistAlosetron Hydrochloride(1:X) (GR 68755 Hydrochloride(1:X)) is a Serotonin 5HT3-receptor antagonist that is used in treatment of irritable bowel syndrome. 了解更多 -
Silodosin (Rapaflo)
Catalog No. A10843 α1-adrenoceptor 拮抗剂Silodosin (Rapaflo)是具有高尿嘧啶选择性的α1-肾上腺素受体拮抗剂。它几乎不引起体位性低血压（与其他α1阻滞剂相反）。 了解更多 -
Phenoxybenzamine hydrochloride
Catalog No. A10719 α-adrenergic (AR) 拮抗剂/CaM 抑制剂Phenoxybenzamine hydrochloride是一种细胞可渗透的，非特异性的，不可逆的α-肾上腺素（AR）拮抗剂，也可作为CaM抑制剂。 了解更多 -
Tamsulosin
Catalog No. A12657 -
ICI 118,551 hydrochloride
Catalog No. A13225 β2 adrenergic 拮抗剂ICI 118,551 hydrochloride是选择性的β2 adrenergic receptor 拮抗剂,结合 β2，β1 和 β3 肾上腺素能受体的Ki 值分别为 0.7，49.5 和 611 nM。 了解更多 -
Diprophylline
Catalog No. A11971 -
Labetalol HCl
Catalog No. A14239 alpha1/beta adrenergic receptors 拮抗剂Labetalol HCl是选择性α1-肾上腺素能受体和非选择性β-肾上腺素能受体的双重拮抗剂。 了解更多 -
Atipamezole HCl
Catalog No. A13902 α2 adrenergic receptor 拮抗剂Atipamezole hydrochloride是一种选择性α2肾上腺素受体拮抗剂（α2A、α2B、α2C、α1A和α1B受体的Ki值分别为1.1、1.0、0.89、1300和6500nm）。已经被证明是大脑的渗透剂。 了解更多 -
Celiprolol HCl
Catalog No. A13623 adrenergic receptor 拮抗剂Celiprolol HCl是一种b1肾上腺素能受体拮抗剂和b2肾上腺素能受体局部激动剂，在体外显示其ED50值为40-50 uM可使人的动脉和静脉松弛。 了解更多 -
BRL 44408 maleate
Catalog No. A13399 -
HEAT hydrochloride (BE 2254)
Catalog No. A13408 Adrenergic α1 Receptor 拮抗剂HEAT hydrochloride (BE 2254)是一种选择性很强的α1-肾上腺素受体拮抗剂，是3-[125I]-衍生物的前体。肾上腺素受体或肾上腺素能受体是参与多种交感神经系统过程的G蛋白偶联受体。 了解更多 -
Idazoxan Hydrochloride
Catalog No. A13409 α2- adrenoceptor 拮抗剂 / I2 imidazoline receptor 激动剂Idazoxan hydrochloride 是α2-AR肾上腺素受体拮抗剂和潜在I2咪唑啉受体激动剂。还显示I1咪唑啉受体拮抗剂活性。(I1、I2和α的公钥基础设施值分别为5.90、7.22、8.01、7.43和7.7)。 了解更多 -
Rauwolscine
Catalog No. A13426 -
S-(-)-Atenolol
Catalog No. A13427 -
(S)-Timolol maleate
Catalog No. A13429 -
Tamsulosin hydrochloride
Catalog No. A14936 -
Acebutolol HCl
Catalog No. A16387 -
Urapidil
Catalog No. A17074 -
Nifenalol HCl
Catalog No. A17246 beta-adrenergic receptor antagonistNifenalol, also known as INPEA, is a new beta-adrenergic receptor antagonist. 了解更多 -
Metipranolol hydrochloride
Catalog No. A18064 β-adrenergic receptor antagonistMetipranolol (hydrochloride) is a non-selective β-adrenergic receptor (β-AR) antagonist. Formulations containing metipranolol have been used in the treatment of elevated IOP in patients with ocular hypertension or glaucoma. 了解更多 -
Atenolol
Catalog No. A21962 -
Chlorcyclizine hydrochloride
Catalog No. A18025 histamine H1 antagonistChlorcyclizine hydrochloride is a histamine H1 antagonist. 了解更多 -
Toreforant
Catalog No. A21058 histamine H4 receptor (H4R) antagonistToreforant is a potent and selective histamine H4 receptor (H4R) antagonist, with a Ki at the human receptor of 8.4 nM. 了解更多 -
PF-03654746
Catalog No. A21429 histamine H3 receptor antagonistPF-03654746 is a potent and selective histamine H3 receptor antagonist with high brain penetration. 了解更多
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- CXCR (19)
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- Endothelin Receptors (17)
- LPA Receptor (11)
- Prostanoid Receptors (14)
- Adenosine Receptors (27)
- Cannabinoid Receptors (8)
- Neurotensin Receptors (1)
- Orexin Receptors (18)
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- Neurokinin Receptors (19)
- Protease-Activated Receptors (PAR) (1)
- S1P Receptor (4)
- CGRP Receptor (7)
- Sigma receptor (5)
- cAMP (1)
- Imidazoline Receptor (2)
- CCK (6)
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