BTK

Catalog No.Inhibitor Name BTKOther
A11020Ibrutinib
****
BLK,Bmx,FGR
A13202AVL-292
****
YES,c-Src,BRK
A13233CNX-774
***
A15558ONO-4059 analogue
**
A16261LFM-A13
*
A12535RN486
**
A11348CGI1746
***
A12706GDC-0834
**
A15008AVL-292 benzenesulfonate
****
YES,c-Src,BRK
A15824ACP-196 (Acalabrutinib)
**
A15976Olmutinib (HM71224)
***
A16262PCI 29732
**
A16263QL47
**

Notes:
1.Hover mouse over " * " to view the IC50 value.(A few compounds have proven potency but without published IC50 data.)
2.For more details about the compound, click on the product name of your interest.
3.The higher the number of " * " is, the more potent the inhibitor or activator is.
4."" refers to compounds which do inhibitory effects on the related isoform, but without specific value.

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  1. MT-802

    Catalog No. A18589
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    BTK degrader
    MT-802 is a potent BTK degrader based on PROTAC technology, with a DC50 of 1 nM. MT-802 has potential to treat C481S mutant chronic lymphocytic leukemia (CLL). 了解更多

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