“glucagon receptor”的搜索结果

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  1. Laropiprant (MK0524)

    Catalog No. A11483
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    DP1 抑制剂
    Laropiprant (MK0524)与烟酸合用可降低血液胆固醇。是一种有效的,选择性的 DP receptor 拮抗剂,Ki 值为 0.57 nM,对 TP 受体的 Ki 值为 2.95 nM。 了解更多
  2. MK-2894

    Catalog No. A11497
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    EP4 receptor 拮抗剂
    MK-2894是一种高度有效和选择性的第二代EP4拮抗剂。 了解更多
  3. NS-304 (Selexipag)

    Catalog No. A13880
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    prostacyclin receptor 激动剂
    NS-304 (Selexipag)是一种选择性的前列环素IP1受体激动剂(人和大鼠IP受体的Ki值为260和2100 nM,EP1-4,DP,FP和TP受体的Ki值为> 10μM)。 了解更多
  4. GW627368

    Catalog No. A15525
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    EP4 receptor 拮抗剂
    GW627368是一种新型,有效且选择性的前列腺素EP4受体竞争拮抗剂(Ki = 100 nM),具有额外的人TP受体亲和力(Ki = 150 nM)。 了解更多
  5. MF498

    Catalog No. A15532
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    EP4 receptor 拮抗剂
    MF498是一种新型的选择性E前列腺素类受体4(EP4受体)拮抗剂,对EP4受体具有很强的结合亲和力,Ki为0.7 nM。 了解更多
  6. PF-04418948

    Catalog No. A12894
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    EP2 Receptor 拮抗剂
    PF-04418948是一种有效的选择性前列腺素EP2受体拮抗剂,IC50为16 nM。 了解更多
  7. TG6-10-1

    Catalog No. A15968
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    Prostaglandin E2 receptor 拮抗剂
    TG6-10-1是前列腺素E2受体亚型EP2的有效和选择性拮抗剂。 了解更多
  8. Grapiprant (CJ-023423)

    Catalog No. A15964
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    prostaglandin EP4 receptor 拮抗剂
    Grapiprant (CJ-023423)是一种具有抗痛觉过敏特性的新型,有效且选择性的前列腺素EP4受体拮抗剂。 了解更多
  9. GSK-269984A

    Catalog No. A17096
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    EP1 receptor 拮抗剂
    GSK-269984A是新型的EP1受体拮抗剂。pIC50 值为 7.9。 了解更多
  10. Benorylate

    Catalog No. A17501
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    Prostaglandin Receptor inhibitor
    Benorilate, also known as Win-11450, is an ester of aspirin and paracetamol with analgesic, antipyretic, and anti-inflammatory activity used in the treatment of rheumatoid diseases. Benorilate has less severe side effects than aspirin. 了解更多
  11. Dinoprost tromethamine

    Catalog No. A17505
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    Prostaglandin Receptor inhibitor
    Dinoprost Tromethamine, also known as Dinoprost Trometamol, is a naturally occurring prostaglandin used in medicine to induce labor and as an abortifacient. 了解更多
  12. GSK726701A

    Catalog No. A20101
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    EP4 partial agonist
    GSK726701A is a novel prostaglandin E2 receptor 4 (EP4) partial agonist with a pEC50 of 7.4. 了解更多
  13. (+)-Cloprostenol

    Catalog No. A12979
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    prostaglandin F2α (PGF2α) analogue
    (+)-Cloprostenol is a prostaglandin F2α (PGF2α) analogue, and shows selective agonistic activity at the prostaglandin receptor. 了解更多
  14. CAY10471 Racemate

    Catalog No. A11760
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    Prostaglandin D2 receptor CRTH2 antagonist
    CAY10471 Racemate (TM30089 Racemate) is a potent and highly selective prostaglandin D2 receptor CRTH2 antagonist. 了解更多
  15. Terutroban

    Catalog No. A20884
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    thromboxane-prostaglandin receptor antagonist
    Terutroban is a thromboxane-prostaglandin receptor antagonist. 了解更多
  16. CJ-42794

    Catalog No. A21948
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    EP4 antagonist
    CJ-42794 is a selective prostaglandin E receptor subtype 4 (EP4) antagonist, inhibits [3H]-PGE2 binding to the human EP4 receptor with a mean pKi of 8.5, a binding affinity that was at least 200-fold more selective for the human EP4 receptor than other human EP receptor subtypes (EP1, EP2, and EP3). 了解更多

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