“glucagon receptor”的搜索结果

22 个项目

每页

设置降序顺序
  1. DPI-3290

    Catalog No. A13699
    Quick View
    opioid receptors agonist
    DPI-3290 (Org 41793) is a potent and specific opioid receptors agonist with Ki values of 0.18 nM, 0.46 nM, and 0.62 nM for δ-, μ-, and κ-opioid receptors, respectively. 了解更多
  2. BRL 52537 HCl

    Catalog No. A11210
    Quick View
    Opioid Receptors 激动剂
    BRL 52537 hydrochloride是一种高度选择性和有效的κ阿片类激动剂(Ki = 0.24 nM)。比吗啡强25倍。 了解更多
  3. AR-M 1000390 hydrochloride

    Catalog No. A21911
    Quick View
    δ opioid receptor agonist
    AR-M 1000390 hydrochloride is an exceptionally selective, potent δ opioid receptor agonist with an EC50 of 7.2??0.9 nM for δ agonist potency. 了解更多
  4. GSK1521498 free base (hydrochloride)

    Catalog No. A21792
    Quick View
    μ-opioid receptor (MOR) antagonist
    GSK1521498 free base (hydrochloride) is a potent and selective μ-opioid receptor (MOR) antagonist. 了解更多
  5. CYT-1010 hydrochloride

    Catalog No. A21348
    Quick View
    mu-opioid receptor agonist
    CYT-1010 hydrochloride is a mu-opioid receptor agonist extracted from patent WO2013173730A2, with EC50s of 13.1 nM and 0.0053 nM on beta-arrestin recruitment and inhibition of cAMP production, respectively. 了解更多
  6. JDTic

    Catalog No. A11468
    Quick View
    κ-opioid receptor antagonist
    JDTic is a highly selective antagonist for the κ-opioid receptor; without affecting the μ- or δ-opioid receptors. 了解更多
  7. GSK1521498 free base

    Catalog No. A18994
    Quick View
    μ-opioid receptor antagonist
    GSK1521498 free base is a potent and selective μ-opioid receptor (MOR) antagonist. GSK1521498 free base is being used for the treatment of disorders of compulsive consumption of food, alcohol, and drugs. 了解更多
  8. BTRX-335140

    Catalog No. A18583
    Quick View
    κ opioid receptor antagonist
    BTRX-335140 (CYM-53093) is a potent and selective, orally active κ opioid receptor (KOR) antagonist, has antagonist activity for κOR, μOR and δOR with IC50 values of 0.8 nM, 110 nM, and 6500 nM, respectively. 了解更多
  9. JTC-801

    Catalog No. A11076
    Quick View
    Opioid Receptor 拮抗剂
    JTC-801是nociceptin receptor(也称为ORL-1受体)的选择性拮抗剂。 了解更多
  10. Trimebutine maleate

    Catalog No. A18115
    Quick View
    ?- opioid receptor agonist
    Trimebutine Maleate is a drug with antimuscarinic and weak mu opioid agonist effects. Trimebutine Maleate modulates the calcium and potassium channels, relieves abdominal pain in patients with irritable bowel syndrome. 了解更多
  11. Bevenopran

    Catalog No. A17110
    Quick View
    opioid receptor antagonis
    Bevenopran,也称为CB-5945,ADL-5945,MK-2402,OpRA III,是一种外周选择性μ-和δ-阿片样物质受体拮抗剂。 了解更多
  12. Cebranopadol (GRT-6005)

    Catalog No. A12670
    Quick View
    Opioid Receptor 激动剂
    Cebranopadol是一种有效的伤害感受器/孤儿蛋白FQ肽(NOP)和阿片受体激动剂。作用于人NOP,MOP,KOP 和δ-阿片肽(DOP)受体,Ki/EC50 分别为 0.9 nM/13 nM,0.7 nM/1.2 nM,2.6 nM/17 nM,18 nM/110 nM。 了解更多
  13. TRV130 HCl (Oliceridine)

    Catalog No. A15444
    Quick View
    u-opioid receptor 激动剂
    TRV130 HCl (Oliceridine)是一种新型的μ-opioid 受体(MOR)G蛋白偏向配体。诱导强大的G蛋白信号传导(pEC50 = 8.1),效力和功效与吗啡相似,但β-arrestin募集和受体内在化作用要低得多。 了解更多
  14. Alvimopan monohydrate

    Catalog No. A14992
    Quick View
    ?-opioid receptor 激动剂
    Alvimopan monohydrate是一种外围作用的类阿片受体(PAM-OR,IC50 = 1.7 nM)拮抗剂,可促进术后肠胃的恢复。 了解更多
  15. Alvimopan dihydrate

    Catalog No. A14991
    Quick View
    ?-opioid receptor 激动剂
    Alvimopan dihydrate (LY 246736,ADL 8-2698)是一种外周作用的类阿片受体(PAM-OR,IC50 = 1.7 nM)拮抗剂,可促进术后胃肠道恢复。 了解更多
  16. LY2795050

    Catalog No. A15149
    Quick View
    k-opioid receptor 拮抗剂
    LY2795050是新型选择性κ阿片受体(KOR)拮抗剂(IC50 = 0.72 nM),具有作为PET示踪剂在体内对KOR成像的潜力。 了解更多
  17. ADL5747

    Catalog No. A13479
    δ opioid receptor 激动剂
    ADL5747是一种选择性的非肽类δ opioid激动剂。 了解更多
  18. U-69593

    Catalog No. A14187
    Quick View
    κ1-opioid receptor 激动剂
    U-69593是有效的选择性κ1阿片受体激动剂(EC50 = 80-109 nM)。在体内有活性。抗伤害感受。 了解更多
  19. Nalmefene hydrochloride

    Catalog No. A13843
    Quick View
    dopamine receptor 激动剂
    Nalmefene hydrochloride是opioid receptor拮抗剂。 了解更多
  20. Alvimopan (ADL 8-2698)

    Catalog No. A11292
    Quick View
    Opioid 拮抗剂
    Alvimopan (ADL 8-2698)表现为外周作用的opioid拮抗剂,Alvimopan竞争性结合胃肠道中的mu-opioid receptor。 了解更多
  21. MCOPPB 3HCl

    Catalog No. A10561
    Quick View
    NOP receptor 激动剂
    MCOPPB 3HCl是一种用作伤害感受器受体的有效和选择性激动剂的化合物,pKi为10.07。 了解更多
  22. ADL5859 HCl

    Catalog No. A11072
    Quick View
    Opioid Receptor 激动剂
    ADL5859 HCl是高效的选择性δ阿片受体激动剂,Ki值为0.84 nM,ED50值为20 nM。 了解更多

22 个项目

每页

设置降序顺序
Rewards