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￥ 0.00 “AZ 960”的搜索结果
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INCB054329 Racemate
Catalog No. A21609 -
AZD3839 free base
Catalog No. A21606 BACE1 inhibitorAZD3839 (free base) is a potent and selective BACE1 inhibitor with IC50 of 23.6 uM, about 14-fold selectivity over BACE2, also a β-secretase enzyme inhibitor. 了解更多 -
MethADP sodium salt
Catalog No. A21603 -
Notch inhibitor 1
Catalog No. A21591 Notch inhibitorNotch inhibitor 1 is a potent Notch inhibitor, with IC50s of 7.8 and 8.5 nM for Notch 1 and Notch 3, respectively. Used in the research of cancer. 了解更多 -
IKK 16 hydrochloride
Catalog No. A21588 IKK2/IKK complex/IKK1 inhibitorIKK 16 hydrochloride is a selective IκB kinase (IKK) inhibitor for IKK2, IKK complex and IKK1 with IC50s of 40 nM, 70 nM and 200 nM, respectively. 了解更多 -
cis-Pralsetinib
Catalog No. A21586 RET inhibitorcis-Pralsetinib (cis-BLU-667) is a highly potent and selective inhibitor of rearranged during transfection (RET), with IC50s ranging from 0.3 to 0.4 nM for WT RET and four enzyme variants (V804L, V804M, M918T, CCDC6-RET), and with broad, robust and anti-tumor activity against multiple RET-driven solid tumor types. 了解更多 -
Ipragliflozin L-Proline
Catalog No. A21579 SGLT2 inhibitorIpragliflozin (L-Proline) is a highly potent and selective SGLT2 inhibitor with an IC50 of 2.8 nM; little and NO potency for SGLT1/3/4/5/6. 了解更多 -
LDN-192960
Catalog No. A21546 Haspin/Dual-specificity Tyrosine-regulated Kinase 2 inhibitorLDN-192960 is an inhibitor of Haspin and Dual-specificity Tyrosine-regulated Kinase 2 (DYRK2) with IC50s of 10 nM and 48 nM, respectively. 了解更多 -
Genz-123346
Catalog No. A21536 glucosylceramide synthase inhibitorGenz-123346 is a potent, orally available glucosylceramide synthase inhibitor. 了解更多 -
Taribavirin
Catalog No. A21525 inosine monophosphate dehydrogenase inhibitorTaribavirin is an orally active inosine monophosphate dehydrogenase inhibitor, has activity against a wide range of viruses, especially the hepatitis C virus and influenza virus. 了解更多 -
Sorafenib (D4)
Catalog No. A21495 multikinase inhibitorSorafenib D4 (Bay 43-9006 D4) is the deuterium labeled Sorafenib. Sorafenib is a multikinase inhibitor IC50s of 6 nM, 20 nM, and 22 nM for Raf-1, B-Raf, and VEGFR-3, respectively. 了解更多 -
Docebenone
Catalog No. A21493 5-LO (5-lipoxygenase) inhibitorDocebenone (AA 861) is a potent, selective and orally active 5-LO (5-lipoxygenase) inhibitor. 了解更多 -
Sorafenib (D3)
Catalog No. A21489 multikinase inhibitorSorafenib D3 (Bay 43-9006 D3) is the deuterium labeled Sorafenib. Sorafenib is a multikinase inhibitor IC50s of 6 nM, 20 nM, and 22 nM for Raf-1, B-Raf, and VEGFR-3, respectively. 了解更多 -
Macozinone
Catalog No. A21488 DprE inhibitorMacozinone (PBTZ169) is a bactericidal benzothiazinone and a potent DprE1 (decaprenylphosphoryl-β-d-ribose 2??-oxidase) inhibitor. 了解更多 -
Givinostat hydrochloride
Catalog No. A21487 HDAC inhibitorGivinostat hydrochloride (ITF-2357 hydrochloride) is a HDAC inhibitor with an IC50 of 198 and 157 nM for HDAC1 and HDAC3, respectively. 了解更多 -
MitoTam iodide, hydriodide
Catalog No. A21486 ETC inhibitorMitoTam iodide, hydriodide is a tamoxifen derivative, an electron transport chain (ETC) inhibitor, spreduces mitochondrial membrane potential in senescent cells and affects mitochondrial morphology. 了解更多 -
PF-5006739
Catalog No. A21479 CK1δ/ε inhibitorPF-5006739 is a potent and selective inhibitor of CK1δ/ε with IC50s of 3.9 nM and 17.0 nM, respectively. 了解更多 -
VXc-?486
Catalog No. A21471 -
Delavirdine
Catalog No. A21469 non-nucleoside reverse transcriptase inhibitorDelavirdine(U 90152) is a potent non-nucleoside reverse transcriptase inhibitor (NNRTI). 了解更多 -
Teneligliptin hydrobromide hydrate
Catalog No. A21465 DPP-4 inhibitorTeneligliptin hydrobromide hydrate is a potent chemotype prolylthiazolidine-based DPP-4 inhibitor, which competitively inhibits human plasma, rat plasma, and human recombinant DPP-4 in vitro, with IC50s of approximately 1 nM. 了解更多 -
(R)-Rivastigmine D6 tartrate
Catalog No. A21454 cholinesterase inhibitor(R)-Rivastigmine D6 (tartrate) is the deuterium labeled (R)-Rivastigmine, which is an cholinesterase inhibitor. 了解更多 -
LY-2584702 hydrochloride
Catalog No. A21416 p70S6K inhibitorLY-2584702 hydrochloride is a selective ATP competitive inhibitor of p70S6K with an IC50 of 4 nM. In S6K1 enzyme assay, the IC50 of LY-2584702 is 2 nM. 了解更多 -
Saterinone hydrochloride
Catalog No. A21402 PDE3 inhibitorSaterinone hydrochloride is a phosphodiesterase III (PDE III) inhibitor. 了解更多 -
42-(2-Tetrazolyl)rapamycin
Catalog No. A21394 mTOR inhibitor42-(2-Tetrazolyl)rapamycin is a prodrug compound of a rapamycin analog extracted from patent US 20080171763 A1, Example 1. Rapamycin is a specific mTOR inhibitor. 了解更多 -
LDN-192960 hydrochloride
Catalog No. A21390 DYRK2 inhibitorLDN-192960 hydrochloride is an inhibitor of Haspin and Dual-specificity Tyrosine-regulated Kinase 2 (DYRK2) with IC50s of 10 nM and 48 nM, respectively. 了解更多 -
PF-06821497
Catalog No. A21388 EZH2 inhibitorPF-06821497 (compound 23a) is a potent, selective and orally active Enhancer of Zeste Homolog 2 (EZH2) inhibitor, with a Ki value <0.1 nM against mutant Y641N EZH2. Exhibits robust tumor growth inhibition. 了解更多 -
DHMEQ racemate
Catalog No. A21379 NF-κB inhibitorDHMEQ racemate is a NF-κB inhibitor. DHMEQ racemate is less active than (-)-DHMEQ. 了解更多 -
AZD-5991 S-enantiomer
Catalog No. A21361 Mcl-1 inhibitorAZD-5991 S-enantiomer is the less active enantiomer of AZD-5991. AZD-5991 S-enantiomer is a Mcl-1 inhibitor with an IC50 of 6.3 μM in FRET assay and a Kd of 0.98 μM in surface plasmon resonance (SPR) assay. 了解更多 -
AZD-5991 Racemate
Catalog No. A21357 Mcl-1 inhibitorAZD-5991 Racemate is the racemate of AZD-5991. AZD-5991 Racemate is a Mcl-1 inhibitor with an IC50 of <3 nM in FRET assay. 了解更多 -
β-Secretase Inhibitor IV
Catalog No. A21346 BACE-1 inhibitorβ-Secretase Inhibitor IV is a potent, cell-active BACE-1 inhibitor with IC50s of 15.6 and 16.3nM under BACE-1 concentrations of 2 nM and 100 pM, respectively. 了解更多 -
PF-06424439 methanesulfonate
Catalog No. A21343 DGAT2 inhibitorPF-06424439 methanesulfonate is an oral, potent and selective imidazopyridine diacylglycerol acyltransferase 2 (DGAT2) inhibitor with an IC50 of 14 nM. 了解更多 -
Picoprazole
Catalog No. A21311 H+/K+-ATPase inhibitorPicoprazole is a specific inhibitor of H+/K+-ATPase with IC50 of 3.1??0.4 μM. 了解更多 -
Potassium oxonate
Catalog No. A21302 uricase inhibitorPotassium oxonate is an inhibitor of uricase, inhibits the phosphorylation of 5-FU to 5-fluorouridine-5'-monophosphate catalyzed by pyrimidine phosphoribosyl-transferase in a different manner from allopurinol in cell-free extracts and intact cells in vitro. 了解更多 -
Amicarbazone
Catalog No. A21294 photosynthetic electron transport inhibitorAmicarbazone(BAY-MKH3586; BAY314666) is a potent inhibitor of photosynthetic electron transport via binding to the Qb domain of photosystem II (PSII); herbicide with a broad spectrum of weed control. 了解更多 -
Lazabemide
Catalog No. A21270 MAO-B inhibitorLazabemide(Ro 19-6327) is selective, reversible monoamine oxidase B (MAO-B) inhibitor (IC50 values are 0.03 and > 100 μM for MAO-B and MAO-A respectively). 了解更多 -
Soblidotin
Catalog No. A21227 tubulin polymerization inhibitorSoblidotin (Auristatin PE) is a novel synthetic Dolastatin 10 derivative and inhibitor of tubulin polymerization. 了解更多 -
BMS-906024
Catalog No. A21172 gamma secretase inhibitorBMS-906024 is an oral and selective gamma secretase inhibitor (GSI) that is a small molecule Notch inhibitor. 了解更多 -
PTP1B-IN-3
Catalog No. A21149 PTP1B inhibitorPTP1B-IN-3 is a potent and selective PTP1B inhibitor with IC50s of 120 nM (PTP1B) and 120 nM (TCPTP), respectively. 了解更多
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