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Etamicastat
Catalog No. A21132 DβH inhibitorEtamicastat (BIA 5-453) is a potent and reversible peripheral dopamine-β-hydroxylase (DβH) inhibitor. 了解更多 -
Risarestat
Catalog No. A21112 aldose reductase inhibitorRisarestat (CT-112), an aldose reductase inhibitor, is developed for the treatment of diabetic complications 了解更多 -
FR 167653 free base
Catalog No. A21110 p38 MAPK inhibitorFR 167653 free base, an orally active and selective p38 MAPK inhibitor, is a potent suppressor of TNF-α and IL-1β production via specific inhibition of p38 MAPK activity. 了解更多 -
Centanafadine
Catalog No. A21099 dual NE/DA transporter inhibitorCentanafadine is dual norepinephrine (NE)/dopamine (DA) transporter inhibitor, also inhibits serotonin transporter, with IC50s of 6 nM, 38 nM and 83 nM for human NE, DA and serotonin transporter , respectively. 了解更多 -
Solenopsin
Catalog No. A21087 ATP-competitive AKT inhibitorSolenopsin is an ATP-competitive AKT inhibitor with IC50 value of 10 μM . 了解更多 -
Gepotidacin
Catalog No. A21086 topoisomerase II inhibitorGepotidacin (GSK2140944) is a novel triazaacenaphthylene bacterial type II topoisomerase inhibitor. 了解更多 -
Relebactam
Catalog No. A21071 diazabicyclooctane inhibitorRelebactam is a diazabicyclooctane inhibitor with activity against a wide spectrum of β-lactamases, including class A (extended-spectrum β-lactamases [ESBLs] and KPC) and class C (AmpC) enzymes. 了解更多 -
Indirubin Derivative E804
Catalog No. A21052 IGF1R inhibitorE 804 is a potent inhibitor of Insulin-like Growth Factor 1 Receptor (IGF1R), with an IC50 of 0.65 μM for IGF1R. 了解更多 -
CAL-130 Racemate
Catalog No. A20942 PI3Kδ inhibitorCAL-130 Racemate is the racemate of CAL-130. CAL-130 Racemate is a PI3Kδ inhibitor. 了解更多 -
KU 59403
Catalog No. A20928 -
Forodesine
Catalog No. A20903 PNP inhibitorForodesine(BCX-1777 freebase; Immucillin-H) is an orally bioavailable PNP inhibitor with picomolar potency; induces apoptosis, mainly in T cells. 了解更多 -
Targapremir-210
Catalog No. A20886 miR-210 inhibitorTargapremir-210 is a potent miR-210 inhibitor with an IC50 of 200 nM in MDA-MB-231 cells. Targapremir-210 binds to the Dicer site of the miR-210 hairpin precursor. This interaction inhibits production of the mature miRNA. 了解更多 -
Tegoprazan
Catalog No. A20873 gastric H+/K+-ATPase inhibitorTegoprazan, a potassium-competitive acid blocker, is a potent, oral active and highly selective inhibitor of gastric H+/K+-ATPase that could control gastric acid secretion and motility, with IC50 values ranging from 0.29-0.52 μM for porcine, canine, and human H+/K+-ATPases in vitro. 了解更多 -
Lansoprazole sodium
Catalog No. A18306 proton pump inhibitorLansoprazole sodium(AG-1749) is a proton pump inhibitor which prevents the stomach from producing acid. 了解更多 -
Ixazomib citrate
Catalog No. A18017 20S proteasome inhibitorIxazomib citrate (MLN9708) is a reversible inhibitor of the chymotrypsin-like proteolytic β5 site of the 20S proteasome with an IC50 of 3.4 nM and a Ki of 0.93 nM. 了解更多 -
Isocarboxazid
Catalog No. A17887 monoamine oxidase inhibitorIsocarboxazid is a non-selective and irreversible inhibitor of monoamine oxidase, with an IC50 of 4.8 μM for rat brain monoamine oxidase in vitro. 了解更多 -
Dapagliflozin ((2S)-1,2-propanediol, hydrate)
Catalog No. A17687 SGLT2 inhibitorDapagliflozin ((2S)-1,2-propanediol, hydrate), a new type of drug used to treat diabetes mellitus (DM), is a competitive sodium/glucose cotransporter 2 (SGLT2) inhibitor, which results in excretion of glucose into the urine. 了解更多 -
Lenvatinib mesylate
Catalog No. A17567 multi-targeted tyrosine kinase inhibitorLenvatinib mesylate (E7080 mesylate), an oral, multi-targeted tyrosine kinase inhibitor that inhibits VEGFR1-3, FGFR1-4, PDGFR, KIT, and RET, shows potent antitumor activities. 了解更多 -
Grazoprevir
Catalog No. A17303 Hepatitis C virus NS3/4a protease inhibitorGrazoprevir (MK-5172) is a selective inhibitor of Hepatitis C virus NS3/4a protease with broad activity across genotypes and resistant variants, with Kis of 0.01 nM (gt1b), 0.01 nM (gt1a), 0.08 nM (gt2a), 0.15 nM (gt2b), 0.90 nM (gt3a), respectively. 了解更多 -
Lomitapide mesylate
Catalog No. A16600 MTP inhibitorLomitapide mesylate(AEGR-733; BMS-201038) is an inhibitor of microsomal triglyceride-transfer protein (MTP) wtih in vitro IC50 of 8 nM. 了解更多 -
Diethylcarbamazine citrate
Catalog No. A16506 arachidonic acid metabolism inhibitorDiethylcarbamazine citrate is an inhibitor of arachidonic acid metabolism in filarial microfilaria; is highly specific for several parasites and does not contain any toxic metallic elements. 了解更多 -
(R)-Lansoprazole
Catalog No. A16496 proton pump inhibitor(R)-Lansoprazole is a proton pump inhibitor which prevents the stomach from producing acid. 了解更多 -
Retaspimycin
Catalog No. A15221 Hsp90 inhibitorRetaspimycin is a potent and water-soluble inhibitor of Hsp90, with EC50s of 119 nM for both Hsp90 and Grp9. 了解更多 -
Nav1.7-IN-3
Catalog No. A13626 voltage-gated sodium channel Nav1.7 inhibitorNav1.7-IN-3 is a selective, orally bioavailable voltage-gated sodium channel Nav1.7 inhibitor with an IC50 of 8 nM. Pain relief. Limited CNS penetration. 了解更多 -
Mericitabine
Catalog No. A11539 HCV NS5B polymerase inhibitorMericitabine (RG 7128; R-7128) is a nucleoside inhibitor of the HCV NS5B polymerase that acts as an RNA chain terminator and prevents elongation of RNA transcripts during replication. 了解更多 -
Pim1/AKK1-IN-1
Catalog No. A11476 multi-kinase inhibitorPim1/AKK1-IN-1 is a potent multi-kinase inhibitor with Kd values of 35 nM/53 nM/75 nM/380 nM for Pim1/AKK1/MST2/LKB1 respectively, and also inhibits MPSK1 and TNIK. 了解更多 -
IRAK inhibitor 2
Catalog No. A11456 interleukin-1 receptor associated kinase inhibitorIRAK inhibitor 2 is interleukin-1 receptor associated kinase inhibitor . 了解更多 -
IRAK inhibitor 1
Catalog No. A11455 IRAK-4 inhibitorIRAK inhibitor 1 is a potent IRAK-4 inhibitor with IC50 of 216 nM, is poorly active against JNK-1 and JNK-2 with IC50 of 3.801 μM, and >10 μM, respectively. 了解更多 -
EMD638683 S-Form
Catalog No. A11399 SGK1 inhibitorEMD638683 S-Form is the S-form of EMD638683. EMD638683 is a highly selective SGK1 inhibitor with IC50 of 3 μM. 了解更多 -
EMD638683 R-Form
Catalog No. A11398 SGK1 inhibitorEMD638683 R-Form is the R-form of EMD638683. EMD638683 is a highly selective SGK1 inhibitor with IC50 of 3 μM. 了解更多 -
Cenisertib
Catalog No. A11262 multi-kinase inhibitorCenisertib (AS-703569) is a multi-kinase inhibitor that blocks the activity of Aurora-kinase-A/B, ABL1, AKT, STAT5 and FLT3. 了解更多 -
Imidaprilate
Catalog No. A20003 ACE inhibitorImidaprilate is an active metabolite of TA-6366, acts as a potent angiotensin converting enzyme (ACE) inhibitor, with an IC50 of 2.6 nM, and is used in the research of hypertensive disease. 了解更多 -
CHMFL-ABL/KIT-155
Catalog No. A12421 ABL/c-KIT dual kinase inhibitorCHMFL-ABL/KIT-155 (CHMFL-ABL-KIT-155; compound 34) is a highly potent and orally active type II ABL/c-KIT dual kinase inhibitor. 了解更多 -
eIF4A3-IN-1
Catalog No. A12956 eIF4A3 inhibitoreIF4A3-IN-1 (compound 53a) is a selective eukaryotic initiation factor 4A3 (eIF4A3) inhibitor (IC50=0.26 μM; Kd=0.043 μM). 了解更多 -
P-gp inhibitor 1
Catalog No. A13384 P-gp inhibitorP-gp inhibitor 1 is a novel inhibitor reversing P-glycoprotein-mediated multidrug resistance. 了解更多 -
c-met-IN-1
Catalog No. A12488 c-Met inhibitorc-met-IN-1 (compound 16) is a potent and selective c-Met inhibitor, with IC50 of 1.1 nM, with antitumor activity. 了解更多 -
KRas G12C inhibitor 4
Catalog No. A12972 KRas G12C inhibitorKRas G12C inhibitor 1 is a compound that inhibits KRas G12C, extracted from patent US 20180072723 A1. 了解更多
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