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Kainic acid monohydrate
Catalog No. A13485 Kainate receptor 激动剂Kainic acid monohydrate是海藻酸酯类离子型谷氨酸受体激动剂。可在体内诱发癫痫发作和神经退行性变，也已用于在啮齿动物中诱发实验性癫痫和检查兴奋性诱发的神经元凋亡机制。 了解更多 -
HEAT hydrochloride (BE 2254)
Catalog No. A13408 Adrenergic α1 Receptor 拮抗剂HEAT hydrochloride (BE 2254)是一种选择性很强的α1-肾上腺素受体拮抗剂，是3-[125I]-衍生物的前体。肾上腺素受体或肾上腺素能受体是参与多种交感神经系统过程的G蛋白偶联受体。 了解更多 -
Idazoxan Hydrochloride
Catalog No. A13409 α2- adrenoceptor 拮抗剂 / I2 imidazoline receptor 激动剂Idazoxan hydrochloride 是α2-AR肾上腺素受体拮抗剂和潜在I2咪唑啉受体激动剂。还显示I1咪唑啉受体拮抗剂活性。(I1、I2和α的公钥基础设施值分别为5.90、7.22、8.01、7.43和7.7)。 了解更多 -
Moxonidine Hydrochloride
Catalog No. A13416 imidazoline receptor 1 激动剂Moxonidine Hydrochloride (BDF5895)是咪唑啉1型受体（I1-R）选择性激动剂，为降压剂。 了解更多 -
NAN-190 hydrobromide
Catalog No. A13417 5-HT1A receptor 拮抗剂NAN-190 hydrobromide是一种广泛用于科学研究的药物和研究化学品。以前认为它是一种选择性的5-HT1A受体拮抗剂，但后来的发现表明它也能有效地阻断α2肾上腺素能受体。 了解更多 -
Rauwolscine
Catalog No. A13426 -
Tulobuterol
Catalog No. A13432 -
Xylazine HCl
Catalog No. A13434 -
Tamsulosin hydrochloride
Catalog No. A14936 -
Cariprazine hydrochloride
Catalog No. A15036 D3/D2 Dopamine Receptor 拮抗剂Cariprazine hydrochloride是一种新型的抗精神病药物，对多巴胺D3（Ki = 0.09 nM）和D2（Ki = 0.5 nM）受体具有高选择性和亲和力，对5-羟色胺5-HT（1A）受体具有中等亲和力。 了解更多 -
Cetirizine
Catalog No. A15041 -
Clemizole hydrochloride
Catalog No. A15047 H1 histamine receptor 拮抗剂Clemizole hydrochloride是H1组胺受体的拮抗剂，对NS4B RNA结合的IC50值为8 mM。 了解更多 -
Clozapine N-oxide
Catalog No. A15048 5-HT1C receptor 拮抗剂Clozapine N-oxide是氯氮平的主要代谢产物，在体外可降低SR-2A（5-HT2血清素受体）密度。 了解更多 -
Ebrotidine
Catalog No. A15075 -
Metoclopramide
Catalog No. A15161 -
Otenabant
Catalog No. A15200 -
rac-Rotigotine Hydrochloride
Catalog No. A15217 -
Reparixin L-lysine salt
Catalog No. A15219 CXCL8 receptor 抑制剂Reparixin L-lysine salt是CXCL8受体的抑制剂，也抑制CXCR1和CXCR2的活化，已显示在各种损伤模型中减弱了炎症反应。 了解更多 -
SB-408124 HCl
Catalog No. A15231 OX Receptor 拮抗剂SB408124 Hydrochloride是OX1受体的非肽拮抗剂，全细胞和膜的Ki分别为57 nM和27 nM。表现出比OX2受体高50倍的选择性。 了解更多 -
Talnetant hydrochloride
Catalog No. A15255 NK3 receptor 拮抗剂Talnetant Hydrochloride是一种有效且选择性的NK3受体拮抗剂（ki = 1.4 nM，hNK-3-CHO）；对hNK-3受体的选择性是对hNK-2受体的100倍，在浓度高达100 uM时对hNK-1没有亲和力。 了解更多 -
Ziprasidone
Catalog No. A15286 5-HT/dopamine receptor 拮抗剂Ziprasidone是5-HT（5-羟色胺）和多巴胺受体拮抗剂的组合，具有抗精神病活性。 了解更多 -
Alosetron Hydrochloride
Catalog No. A14989 -
Alvimopan dihydrate
Catalog No. A14991 ?-opioid receptor 激动剂Alvimopan dihydrate (LY 246736,ADL 8-2698)是一种外周作用的类阿片受体（PAM-OR，IC50 = 1.7 nM）拮抗剂，可促进术后胃肠道恢复。 了解更多 -
Alvimopan monohydrate
Catalog No. A14992 ?-opioid receptor 激动剂Alvimopan monohydrate是一种外围作用的类阿片受体（PAM-OR，IC50 = 1.7 nM）拮抗剂，可促进术后肠胃的恢复。 了解更多 -
Atrasentan HCl
Catalog No. A15007 Endothelin 拮抗剂 receptorAtrasentan hydrochloride是一种开发用于治疗前列腺癌的内皮素拮抗剂受体（IC50 = 0.0551 nM，ETA）。 了解更多 -
Bavisant dihydrochloride
Catalog No. A15015 -
Bavisant dihydrochloride hydrate
Catalog No. A15016 -
MF498
Catalog No. A15532 -
Ricasetron
Catalog No. A15499 -
Lerisetron
Catalog No. A15501 -
Macitentan
Catalog No. A11492 Endothelin receptor 拮抗剂Macitentan是一种口服活性非肽双重ETA/ETB(内皮素) receptor双重拮抗剂，IC50为0.5 nM/391 nM。用于治疗特发性肺纤维化(IPF)和肺动脉高压(PAH)。 了解更多 -
SB271046
Catalog No. A15438 -
TRV130 HCl (Oliceridine)
Catalog No. A15444 u-opioid receptor 激动剂TRV130 HCl (Oliceridine)是一种新型的μ-opioid 受体（MOR）G蛋白偏向配体。诱导强大的G蛋白信号传导（pEC50 = 8.1），效力和功效与吗啡相似，但β-arrestin募集和受体内在化作用要低得多。 了解更多 -
SCH 23390 HCl
Catalog No. A13066 -
Pimavanserin (ACP-103)
Catalog No. A14434 5-HT2A receptor 激动剂Pimavanserin (ACP-103)是一种有效的选择性5-HT2A受体反向激动剂，在基于细胞的功能测定中，平均pIC50为8.7。 了解更多 -
CBiPES HCl
Catalog No. A15811 -
Preladenant
Catalog No. A13504
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