“ADM Hydrochloride”的搜索结果

产品 51 到 100 共 147个

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  1. Maprotiline hydrochloride

    Catalog No. A10555
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    noradrenalin re-uptake 抑制剂
    Maprotiline hydrochloride是选择性去甲肾上腺素再摄取抑制剂。 了解更多
  2. ICI 118,551 hydrochloride

    Catalog No. A13225
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    β2 adrenergic 拮抗剂
    ICI 118,551 hydrochloride是选择性的β2 adrenergic receptor 拮抗剂,结合 β2,β1 和 β3 肾上腺素能受体的Ki 值分别为 0.7,49.5 和 611 nM。 了解更多
  3. ent Naxagolide Hydrochloride

    Catalog No. A13089
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    dopamine D2-receptor 激动剂
    ent Naxagolide Hydrochloride是一种多巴胺D2受体激动剂,用于治疗锥体外系疾病。该化合物是抗帕金森病药物。 了解更多
  4. Olopatadine hydrochloride

    Catalog No. A10671
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    Olopatadine hydrochloride是一种双重作用的组胺H1受体拮抗剂和肥大细胞稳定剂。 了解更多
  5. Tamsulosin hydrochloride

    Catalog No. A12846
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    Tamsulosin hydrochloride是前列腺素α1A肾上腺素受体的拮抗剂。 了解更多
  6. Sibutramine hydrochloride

    Catalog No. A12397
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    SNR 抑制剂
    Sibutramine hydrochloride是5-HT和去甲肾上腺素再摄取抑制剂(SNRI)。 了解更多
  7. Nalfurafine hydrochloride

    Catalog No. A12579
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    opioid κ-selective 激动剂
    Nalfurafine hydrochloride是一种κ-opioid激动剂。 了解更多
  8. Phenoxybenzamine hydrochloride

    Catalog No. A10719
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    α-adrenergic (AR) 拮抗剂/CaM 抑制剂
    Phenoxybenzamine hydrochloride是一种细胞可渗透的,非特异性的,不可逆的α-肾上腺素(AR)拮抗剂,也可作为CaM抑制剂。 了解更多
  9. Granisetron Hydrochloride

    Catalog No. A10437
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    5-HT3 receptor 拮抗剂
    Granisetron Hydrochloride是血清素5-ht3受体拮抗剂。 了解更多
  10. Dopamine hydrochloride

    Catalog No. A10331
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    Dopamine hydrochloride (abbreviated as DA)是儿茶酚胺家族中的一种简单的有机化学物质,是一种单胺类神经递质,一种由神经细胞释放以向其他神经细胞发送信号的化学物质。 了解更多
  11. Clonidine hydrochloride

    Catalog No. A10232
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    Alpha adrenergic 激动剂
    Clonidine hydrochloride被归类为中枢作用的α肾上腺素能激动剂。Clonidine主要作为咪唑啉受体激动剂。 了解更多
  12. Detomidine hydrochloride

    Catalog No. A10298
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    Adrenergic Receptor 激动剂
    Detomidine hydrochloride是具有镇痛作用的镇静剂。α2-肾上腺素能激动剂产生剂量依赖性的镇静和镇痛作用,并通过激活α2儿茶酚胺受体介导,从而引起负反馈反应,从而减少兴奋性神经递质的产生。 了解更多
  13. Ro 10-5824 dihydrochloride

    Catalog No. A21986
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    dopamine D4 receptor partial agonist
    Ro 10-5824 dihydrochloride is a selective dopamine D4 receptor partial agonist, with Ki of 5.2 nM. 了解更多
  14. Vofopitant dihydrochloride

    Catalog No. A21543
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    NK1 receptor antagonist
    Vofopitant dihydrochloride (GR 205171A) is a potent, selective and orally available tachykinin neurokinin 1(NK1) receptor antagonist. 了解更多
  15. JNJ-37822681 dihydrochloride

    Catalog No. A21470
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    dopamine D2 receptor antagonist
    JNJ-37822681 dihydrochloride is a potent, specific, centrally active, fast-dissociating dopamine D2 receptor antagonist with a moderate binding affinity for the dopamine D2L receptor (Ki =158 nM), which has potential for the treatment of schizophrenia and bipolar disorder. 了解更多
  16. PF429242 dihydrochloride

    Catalog No. A21386
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    S1P inhibitor
    PF429242 dihydrochloride is a reversible and competitive S1P inhibitor with an IC50 of 175 nM. 了解更多
  17. SB-277011 dihydrochloride

    Catalog No. A21353
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    dopamine D3 receptor antagonist
    SB-277011 dihydrochloride (SB-277011A dihydrochloride) is a potent, selective, orally bioavailable and brain penetrate dopamine D3 receptor antagonist, with pKis of 8.0, 6.0, <5.2 and 5.9 for D3, D2, 5-HT1B, and 5-HT1D receptors, respectively. 了解更多
  18. Lesopitron dihydrochloride

    Catalog No. A12950
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    5-HT1A receptor agonist
    Lesopitron dihydrochloride is a full and selective 5-HT1A receptor agonist with IC50 of 125 nM in rat hippocampal membranes. 了解更多
  19. MT-DADMe-ImmA

    Catalog No. A13651
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    human 5'-methylthioadenosine phosphorylase inhibitor
    MT-DADMe-ImmA is an inhibitor of human 5'-methylthioadenosine phosphorylase (MTAP) with a Ki of 90 pM. 了解更多
  20. KAG-308

    Catalog No. A18389
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    EP4 激动剂
    KAG-308, a newly-identified EP4-selective agonist shows efficacy for treating ulcerative colitis and can bring about lower risk of colorectal carcinogenesis by oral administration. 了解更多
  21. Levocetirizine Dihydrochloride

    Catalog No. A17440
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    L-isomer of cetirizine and histamine H1 receptor antagonist
    Levocetirizine dihydrochloride is a L-isomer of cetirizine and histamine H1 receptor antagonist. It incrases levels of CD4+ CD25+ T cells and decreases levels of eosinophils, decreasing allergy symptoms. 了解更多
  22. Buspirone HCl

    Catalog No. A15687
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    5HT(1A) receptor 激动剂
    Buspirone hydrochloride是一种具有5-D(2)多巴胺能作用的血清素能(5HT(1A)受体激动剂)抗焦虑药,用于焦虑症。 了解更多
  23. Buclizine HCl

    Catalog No. A15666
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    Buclizine hydrochloride是哌嗪衍生物家族的抗组胺药和抗胆碱能药。 了解更多
  24. Bavisant dihydrochloride hydrate

    Catalog No. A15016
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    H3 receptor 拮抗剂
    Bavisant dihydrochloride hydrate是人类H3受体的高度选择性口服活性拮抗剂。 了解更多
  25. Bavisant dihydrochloride

    Catalog No. A15015
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    H3 receptor 拮抗剂
    Bavisant dihydrochloride是一种人类H3受体的高选择性,口服活性拮抗剂。 了解更多
  26. Dexpramipexole dihydrochloride

    Catalog No. A15066
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    dopamine 激动剂
    Dexpramipexole dihydrochloride是一种神经保护剂和弱非麦角灵多巴胺激动剂。 了解更多
  27. SB 258585 HCl

    Catalog No. A14026
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    5-HT6 serotonin receptor 拮抗剂
    SB 258585 hydrochloride是一种选择性和有效的SR-6拮抗剂。该化合物显示出比其他5-羟色胺受体亚型高160倍的选择性。 了解更多
  28. Medetomidine HCl

    Catalog No. A13775
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    adrenergic alpha-2 receptor 激动剂
    Medetomidine Hydrochloride是一种肾上腺素α2-受体激动剂,Ki为1.08 nM,比作用于α1-adrenoceptor选择性高1620倍。由于其镇痛和镇静作用而被用于兽医学。 了解更多
  29. (+) PD 128907

    Catalog No. A14376
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    Dopamine receptor 激动剂
    (+)-PD 128907 hydrochloride是一种有效的D3DR(多巴胺受体)激动剂(Ki = 2.3 nM)。 了解更多
  30. Atipamezole HCl

    Catalog No. A13902
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    α2 adrenergic receptor 拮抗剂
    Atipamezole hydrochloride是一种选择性α2肾上腺素受体拮抗剂(α2A、α2B、α2C、α1A和α1B受体的Ki值分别为1.1、1.0、0.89、1300和6500nm)。已经被证明是大脑的渗透剂。 了解更多
  31. SB 399885 HCl

    Catalog No. A14102
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    5-HT6 拮抗剂
    SB 399885 hydrochloride是一种有效的,脑渗透剂和口服活性的SR-6拮抗剂。它对SR-6的选择性比其他血清素受体高200倍(对于人类重组,天然大鼠和天然人类SR-6受体,pKi值分别为9.11、8.81和9.02)。 了解更多
  32. GBR 12783 dihydrochloride

    Catalog No. A13128
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    dopamine uptake 抑制剂
    GBR 12783 dihydrochloride是一种非常有效的选择性多巴胺摄取抑制剂(抑制大鼠纹状体突触体中[3H]-多巴胺摄取的IC50为1.8 nM)。 了解更多
  33. cis-(Z)-Flupentixol dihydrochloride

    Catalog No. A12347
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    Dopamine receptor 拮抗剂
    cis-(Z)-Flupentixol dihydrochloride是多巴胺受体拮抗剂、抗精神病药物、抗精神病药物。 了解更多
  34. Pramipexole dihydrochloride

    Catalog No. A12536
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    Pramipexole dihydrochloride是对D3受体表现出选择性的多巴胺受体激动剂。 了解更多
  35. Fexofenadine HCl

    Catalog No. A11859
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    COX 抑制剂/histamine H1 receptor 激动剂
    Fexofenadine Hydrochloride是一种抗组胺药,可抑制Cox-1,Cox-2,并且是组胺H1受体激动剂,IC50为246 nM。 了解更多
  36. Nebivolol HCl

    Catalog No. A10630
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    Nebivolol hydrochloride是β1-肾上腺素受体的高度选择性拮抗剂(Ki = 0.88 nM,β2-肾上腺素受体Ki = 48 nM)。 了解更多
  37. Ropinirole HCl

    Catalog No. A11916
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    Ropinirole Hydrochloride是一种多巴胺受体激动剂。 了解更多
  38. Cetirizine Dihydrochloride

    Catalog No. A10195
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    Cetirizine Dihydrochloride是第二代抗组胺药,是羟嗪的主要代谢产物,是用于治疗过敏,花粉症,血管性水肿和荨麻疹的消旋选择性H1受体反向激动剂。 了解更多
  39. GBR-12935 2HCl

    Catalog No. A11937
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    DAT and SLC6A2 抑制剂
    GBR-12935 dihydrochloride是一种有效的选择性多巴胺再摄取抑制剂。 了解更多
  40. Duloxetine HCl

    Catalog No. A11717
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    Duloxetine Hydrochloride是一种5-羟色胺和去甲肾上腺素再摄取抑制剂(SNRI),Ki为 4.6 nM。用于治疗压力性尿失禁和抑郁症。 了解更多
  41. Pramipexole dihydrochloride monohyrate

    Catalog No. A10747
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    Dopamine Receptor 激动剂
    Pramipexole dihydrochloride monohyrate是非麦角灵类的多巴胺激动剂,适用于治疗早期帕金森氏病(PD)和不安腿综合征(RLS)。 了解更多
  42. Vanoxerine 2HCl (GBR-12909)

    Catalog No. A10725
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    dopamine re-uptake 抑制剂
    Vanoxerine 2HCl (GBR-12909)是哌嗪衍生物,是一种有效的、选择性的多巴胺摄取(dopamine uptake)抑制剂。 了解更多
  43. Naftopidil 2HCl

    Catalog No. A10619
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    5-HT1A and α1-adrenergic receptor 拮抗剂
    Naftopidil 2HCl是选择性5-HT1A和α1-肾上腺素能受体拮抗剂,IC50分别为0.1μM和0.2μM。 了解更多
  44. BRL-15572 dihydrochloride

    Catalog No. A11178
    5-HT1D receptor 拮抗剂
    BRL-15572是一种选择性的h5-HT1D拮抗剂,相对于h5-HT1B表现出60倍的选择性,对一系列其他受体类型的亲和力很小或没有亲和力。 了解更多
  45. MCOPPB 3HCl

    Catalog No. A10561
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    NOP receptor 激动剂
    MCOPPB 3HCl是一种用作伤害感受器受体的有效和选择性激动剂的化合物,pKi为10.07。 了解更多
  46. CGS 21680 HCl

    Catalog No. A16441
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    Adenosine A2 receptor 激动剂
    CGS 21680 HCl是腺苷A2受体激动剂,IC50为22 nM,比A1受体高140倍。 了解更多
  47. Octopamine hydrochloride

    Catalog No. A13419
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    Octopamine hydrochloride是一种无脊椎生物胺神经递质,与去甲肾上腺素相关,是肾上腺素受体激动剂。 了解更多
  48. Tetrahydrozoline Hydrochloride

    Catalog No. A13080
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    Adrenergic Receptor 激动剂
    Tetrahydrozoline Hydrochloride是一种引起结膜血管收缩的α激动剂。 了解更多
  49. Trazodone HCl

    Catalog No. A11703
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    Trazodone HCl 是一种抗抑郁药,属于5-羟色胺受体拮抗剂和再摄取抑制剂。 了解更多
  50. Azelastine HCl (Allergodil)

    Catalog No. A10117
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    Azelastine HCl (Allergodil)是有效的第二代选择性组胺拮抗剂(组胺-H1-受体拮抗剂)。 了解更多

产品 51 到 100 共 147个

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