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“Akt Inhibitor”的搜索结果

产品 201 到 250 共 5382个

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  1. IMD-0560
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    IMD-0560

    Catalog No. A19224
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    IκB kinase β inhibitor
    IMD-0560 is a novel IκB kinase β inhibitor. 了解更多
  2. SHIN1
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    SHIN1

    Catalog No. A19228
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    SHMT1/2 inhibitor
    SHIN1 (RZ-2994) is a human serine hydroxymethyltransferse 1 and 2 (SHMT1/2) inhibitor with IC50s of 5 and 13 nM, respectively, in an in vitro assay. 了解更多
  3. FT-1518
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    FT-1518

    Catalog No. A19230
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    mTORC1/mTORC2 inhibitor
    FT-1518 is a new generation selective, potent and oral bioavailable mTORC1 and mTORC2 inhibitor, and exhibits antitumor activity. 了解更多
  4. Delgocitinib
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    Delgocitinib

    Catalog No. A19234
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    JAK inhibitor
    Delgocitinib is a novel and specific JAK inhibitor with IC50s of 2.8, 2.6, 13 and 58 nM for JAK1, JAK2, JAK3 and Tyk2, respectively. 了解更多
  5. TC HSD 21
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    TC HSD 21

    Catalog No. A19236
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    17β-HSD3 inhibitor
    TC HSD 21 is a potent 17β-hydroxysteroid dehydrogenase type 3 (17β-HSD3) inhibitor with an IC50 of 14 nM. TC HSD 21 shows excellent selectivity over 17β-HSD isoenzymes and nuclear receptors. 了解更多
  6. SGC-iMLLT
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    SGC-iMLLT

    Catalog No. A19237
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    MLLT1/3-histone interactions inhibitor
    SGC-iMLLT is a first-in-class chemical probe and a potent, selective inhibitor of MLLT1/3-histone interactions with an IC50 of 0.26 μM. 了解更多
  7. PF-06869206
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    PF-06869206

    Catalog No. A19239
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    SLC34A1 inhibitor
    PF-06869206 is an orally bioavailable selective inhibitor of the sodium-phosphate cotransporter NaPi2a (SLC34A1) with an IC50 of 380 nM. 了解更多
  8. CH7057288
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    CH7057288

    Catalog No. A19241
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    TRK inhibitor
    CH7057288 is a potent and selective TRK inhibitor. 了解更多
  9. GNE-955
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    GNE-955

    Catalog No. A19243
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    Pim kinase inhibitor
    GNE-955 is a potent and orally active pan Pim kinase inhibitor with Kis of 0.018, 0.11, 0.08 nM for Pim1, Pim2, Pim3, respectively. 了解更多
  10. Alobresib
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    Alobresib

    Catalog No. A19246
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    BET bromodomain inhibitor
    Alobresib (GS-5829) is a BET bromodomain inhibitor, which represents a highly effective therapeutics agent against recurrent/chemotherapy resistant uterine serous carcinoma (USC) overexpressing c-Myc. 了解更多
  11. JAK1-IN-3
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    JAK1-IN-3

    Catalog No. A19251
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    JAK1 inhibitor
    JAK1-IN-3 is a selective JAK1 inhibitor, with an IC50 of 73 nM, weakly inhibits JAK2, and shows little inhibition on JAK3 (IC50, >14.7, >30 μM, respectively). 了解更多
  12. Selitrectinib
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    Selitrectinib

    Catalog No. A19252
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    TKI inhibitor
    Selitrectinib (LOXO-195) is a next-generation TRK kinase inhibitor (TKI), with IC50s of 0.6 nM, <2.5 nM for TRKA and TRKC respectively. 了解更多
  13. HSK0935
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    HSK0935

    Catalog No. A19253
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    SGLT2 inhibitor
    HSK0935 is a potent, highly selective and orally available SGLT2 inhibitor with an IC50 of 1.3 nM. Antihyperglycemic activities. 了解更多
  14. FT827
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    FT827

    Catalog No. A19256
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    USP7 inhibitor
    FT827 is a selective and covalent ubiquitin-specific protease 7 (USP7) inhibitor (Ki=4.2 ?M). FT827 binds to the USP7 catalytic domain (USP7CD; residues 208-560) with an apparent Kd value of 7.8 ?M. 了解更多
  15. Adavivint
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    Adavivint

    Catalog No. A19257
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    Wnt signaling inhibitor
    Adavivint (SM04690; Lorecivivint) is a potent and selective inhibitor of canonical Wnt signaling, with an EC50 of 19.5 nM via a high-throughput TCF/LEF-reporter assay in SW480 colon cancer cells. 了解更多
  16. AZD3229
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    AZD3229

    Catalog No. A19259
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    pan-KIT mutant inhibitor
    AZD3229 is a potent pan-KIT mutant inhibitor for the treatment of gastrointestinal stromal tumors. 了解更多
  17. MF-094
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    MF-094

    Catalog No. A19260
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    USP30 inhibitor
    MF-094 is a potent and selective USP30 inhibitor with an IC50 of 120 nM. MF-094 increases protein ubiquitination and accelerates mitophagy. 了解更多
  18. PGS-IN-1
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    PGS-IN-1

    Catalog No. A19263
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    PGS inhibitor
    PGS-IN-1 is a potent inhibitor of prostaglandin synthetase (PGS) with an IC50 of 0.28 μM; also inhibits 5-lipoxygenase with an IC50 of 1.05 μM. 了解更多
  19. BB-Cl-Amidine
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    BB-Cl-Amidine

    Catalog No. A19265
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    PAD inhibitor
    BB-Cl-Amidine is a peptidylarginine deminase (PAD) inhibitor. 了解更多
  20. DCPIB
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    DCPIB

    Catalog No. A19268
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    VRAC inhibitor
    DCPIB is a selective, reversible and potent inhibitor of volume-regulated anion channels (VRAC), voltage-dependently activates potassium channels TREK1 and TRAAK, inhibits TRESK, TASK1 and TASK3 (IC50s, 0.14, 0.95, 50.72 μM, respectively). 了解更多
  21. F-1
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    F-1

    Catalog No. A19269
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    ALK and ROS1 dual inhibitor
    F-1 is a potent ALK and ROS1 dual inhibitor, suppresses phospho-ALK and its relative downstream signaling pathways, with IC50s of 2.1 nM, 2.3 nM, 1.3 nM and 3.9 nM for ALKWT, ROS1WT, ALKL1196M and ALKG1202R, respectively. 了解更多
  22. GSK-626616
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    GSK-626616

    Catalog No. A19273
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    DYRK3 inhibitor
    GSK-626616 is a potent, orally bioavailable inhibitor of DYRK3 (IC50=0.7 nM). 了解更多
  23. Trk-IN-4
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    Trk-IN-4

    Catalog No. A19277
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    pan-Trk inhibitor
    Trk-IN-4 (PF-6683324 isomer) is a potent pan-Trk inhibitor in cell-based assays with IC50s of 1.9 nM, 2.6 nM and 1.1 nM for TrkA, TrkB and TrkC, respectively. Anti-hyperalgesic effect. 了解更多
  24. UCN-02
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    UCN-02

    Catalog No. A19279
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    PKC inhibitor
    UCN-02 (7-epi-Hydroxystaurosporine) is a selective protein kinase C (PKC) inhibitor produced by Streptomyces strain N-12, with IC50s of 62 nM and 250 nM for PKC and protein kinase A (PKA), respectively. 了解更多
  25. AZ PFKFB3 26
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    AZ PFKFB3 26

    Catalog No. A19281
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    PFKFB3 inhibitor
    AZ PFKFB3 26 is a potent and selective inhibitor of the metabolic kinase PFKFB3 with an IC50 of 23 nM. AZ PFKFB3 26 inhibits PFKFB1 and PFKFB2 with IC50s of 2.06 and 0.384 μM, respectively. 了解更多
  26. DK419
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    DK419

    Catalog No. A19287
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    Wnt/β-catenin signaling inhibitor
    DK419 is a potent and orally active Wnt/β-catenin signaling inhibitor, with an IC50 of 0.19 μM. DK419 reduces protein lelvels of Axin2, β-catenin, c-Myc, Cyclin D1 and Survivin and induces production of pAMPK. 了解更多
  27. UCT943
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    UCT943

    Catalog No. A19288
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    PI4K inhibitor
    UCT943 is a next-generation Plasmodium falciparum PI4K inhibitor. UCT943 inhibits the P. vivax PI4K (PvPI4K) enzyme with an IC50 of 23 nM. 了解更多
  28. CSF1R-IN-1
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    CSF1R-IN-1

    Catalog No. A19291
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    CSF1R inhibitor
    CSF1R-IN-1 is a CSF1R inhibitor with an with an IC50 of 0.5 nM. 了解更多
  29. PH-002
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    PH-002

    Catalog No. A19297
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    apo inhibitor
    PH-002 is an inhibitor of apolipoprotein (apo) E4 intramolecular domain interaction in neuronal cells that could rescue impairments of mitochondrial motility and neurite outgrowth. 了解更多
  30. Trk-IN-3
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    Trk-IN-3

    Catalog No. A19298
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    pan-Trk inhibitor
    Trk-IN-3 is a potent pan-Trk inhibitor in cell-based assays with IC50s of 8.4 nM, 6.2 nM and 2.2 nM for TrkA, TrkB and TrkC, respectively. Anti-hyperalgesic effect. 了解更多
  31. c-Met-IN-2
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    c-Met-IN-2

    Catalog No. A19302
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    c-Met inhibitor
    c-Met-IN-2 is a potent, selective and orally available c-Met inhibitor, with an IC50 of 0.6 nM, with antitumor activity. 了解更多
  32. Quilseconazole
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    Quilseconazole

    Catalog No. A19305
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    fungal Cyp51 inhibitor
    Quilseconazole (VT-1129) is a potent, orally active fungal Cyp51 (lanosterol 14-α-demethylase) inhibitor, binds tightly to cryptococcal CYP51, but weakly inhibits humans CYP450 enzymes. 了解更多
  33. NIK SMI1
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    NIK SMI1

    Catalog No. A19308
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    NIK inhibitor
    NIK SMI1 is a potent, selective NF-κB inducing kinase (NIK) inhibitor, which inhibits NIK-catalyzed hydrolysis of ATP to ADP with IC50 of 0.23±0.17 nM. 了解更多
  34. Ziritaxestat
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    Ziritaxestat

    Catalog No. A19312
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    ATX inhibitor
    Ziritaxestat (GLPG1690) is a first-in-class autotaxin (ATX) inhibitor, with an IC50 of 131 nM and Ki of 15 nM. 了解更多
  35. Synta66
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    Synta66

    Catalog No. A19314
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    CRAC channel inhibitor
    Synta66 is an inhibitor of store-operated calcium entry channel Orai, which forms the pore of the CRAC channel, and used for the research of neurological disease. 了解更多
  36. PTC596
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    PTC596

    Catalog No. A19320
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    BMI-1 inhibitor
    PTC596 is an orally active and selective B-cell-specific Moloney murine leukemia virus integration site 1 (BMI-1) inhibitor. 了解更多
  37. KU-32
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    KU-32

    Catalog No. A19321
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    Hsp90 inhibitor
    KU-32 is a novel, novobiocin-based Hsp90 inhibitor that can protect against neuronal cell death. 了解更多
  38. BTB-1
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    BTB-1

    Catalog No. A19322
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    Kif18A inhibitor
    BTB-1 is a potent, selective and reversible mitotic motor protein Kif18A inhibitor with an IC50 of 1.69 μM. 了解更多
  39. (+)-JQ1 PA
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    (+)-JQ1 PA

    Catalog No. A19328
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    BET bromodomain inhibitor
    (+)-JQ1 PA is a clickable JQ1 for building PROTACs, which acts as a BET bromodomain inhibitor. 了解更多
  40. AD80
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    AD80

    Catalog No. A19332
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    multikinase inhibitor
    AD80, a multikinase inhibitor, inhibits RET, RAF,SRCand S6K, with greatly reduced mTOR activity. 了解更多
  41. LY 178002
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    LY 178002

    Catalog No. A19333
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    5-lipoxygenase inhibitor
    LY 178002 is a potent inhibitor of 5-lipoxygenase, phospholipase A2, with IC50 of 0.6 μM for 5-1ipoxygenase, inhibits cellular production of LTB4 by human polymorphonuclear leukocytes, and shows relatively weak inhibition on cyclooxygenase. 了解更多
  42. PRN1371
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    PRN1371

    Catalog No. A19340
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    FGFR1-4/CSF1R inhibitor
    PRN1371 is a highly selective and potent FGFR1-4 and CSF1R inhibitor with IC50s of 0.6, 1.3, 4.1, 19.3 and 8.1 nM for FGFR1, FGFR2, FGFR3, FGFR4 and CSF1R, respectively. 了解更多
  43. 2614W94
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    2614W94

    Catalog No. A19341
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    monoamine oxidase-A inhibitor
    2614W94 is a selective, reversible inhibitor of monoamine oxidase-A with a competitive mechanism of inhibition and IC50 of 5 nM and Ki of 1.6 nM with serotonin as substrate. 了解更多
  44. VTX-27
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    VTX-27

    Catalog No. A19347
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    PKCθ inhibitor
    VTX-27 is a selective protein kinase C θ (PKC θ) inhibitor, with Kis of 0.08 nM and 16 nM for PKC θ and PKC δ. 了解更多
  45. Sirt2-IN-1
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    Sirt2-IN-1

    Catalog No. A19348
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    Sirt2 inhibitor
    Sirt2-IN-1 (Compound 9) is a sirtuin 2 (Sirt2) inhibitor with an IC50 of 163 nM. 了解更多
  46. ZEN-3411
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    ZEN-3411

    Catalog No. A19349
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    BET inhibitor
    ZEN-3411 is a BET inhibitor with IC50s of 0.05, 0.05 and 0.06 μM for BRD4(BD1), BRD4(BD2) and BRD4(BD1BD2), respectively. ZEN-3411 can be used to form PROTACs to induce degradation of BRD4. 了解更多
  47. Lodenafil carbonate
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    Lodenafil carbonate

    Catalog No. A19350
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    PDE5 inhibitor
    Lodenafil carbonate, a dimer that acts as a prodrug delivering Lodenafil in vivo, is an orally active phosphodiesterase type 5 (PDE5) inhibitor for the treatment of erectile dysfunction (ED). 了解更多
  48. Ifenprodil glucuronide
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    Ifenprodil glucuronide

    Catalog No. A19353
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    platelet aggregation inhibitor
    Ifenprodil glucuronide is a derivative of Ifenprodil. Ifenprodil is a vasodilator and an inhibitor of platelet aggregation, and Ifenprodil glucuronide has no effect on platelet aggregation and arterial contraction. 了解更多
  49. ML218
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    ML218

    Catalog No. A19355
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    T-type calcium channel inhibitor
    ML218 is a selective T-type calcium channel inhibitor with IC50s of 270 and 310 nM for Cav3.3 and Cav3.2 in electrophysiology assay, respectively. 了解更多
  50. ZEN-3862
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    ZEN-3862

    Catalog No. A19358
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    BET inhibitor
    ZEN-3862 is a BET inhibitor with IC50s of 0.16 and 0.13 μM for BRD4(BD1) and BRD4(BD2) , respectively. ZEN-3862 can be used to form PROTACs to induce degradation of BRD4. 了解更多

产品 201 到 250 共 5382个

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