“ADM Hydrochloride”的搜索结果

产品 1 到 50 共 695个

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  1. Berberine HCl

    Catalog No. A10126
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    Berberine hydrochloride被发现具有对心血管系统的多种有益作用和显着的抗炎活性。 小ber碱可有效降低LPS刺激的巨噬细胞的细胞内超氧化物水平。 小碱对细胞氧化还原的这种恢复是通过其对gp91phox表达的选择性抑制和SOD活性的增强而介导的。 了解更多
  2. Thioridazine hydrochloride

    Catalog No. A11119
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    Thioridazine hydrochloride是一种多巴胺受体拮抗剂,具有抗精神病活性。 最近还报道了硫代哒嗪能够成功杀死人类癌症干细胞。 了解更多
  3. Memantine hydrochloride

    Catalog No. A11708
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    NMDA receptor 拮抗剂
    Memantine hydrochloride是nmda受体的拮抗剂,与离子通道位点结合。它还是CYP2B6和CYP2D6抑制剂,作用于重组CYP2B6和CYP2D6,Ki分别为0.51 nM和94.9 μM。它被用于治疗帕金森综合征。 了解更多
  4. Amiloride hydrochloride dihydrate

    Catalog No. A11728
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    Amiloride hydrochloride dihydrate是一种强效上皮钠通道阻滞剂和选择性低阈值(t型)钙通道蛋白抑制剂(kd=30μm)。 了解更多
  5. Benidipine hydrochloride

    Catalog No. A11730
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    Benidipine hydrochloride是一种长效的T型钙通道阻滞剂,对高血压糖尿病患者的血压和肾功能有影响。 了解更多
  6. Chlorpromazine hydrochloride

    Catalog No. A10206
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    Chlorpromazine hydrochloride是典型的抗精神病药类别的多巴胺拮抗剂,具有治疗精神分裂症的其他抗肾上腺素能,抗5-羟色胺能,抗胆碱能和抗组胺能特性。 了解更多
  7. Clomipramine HCl

    Catalog No. A10231
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    5-HT Receptor 激动剂
    Clomipramine HCl是下列转运蛋白的阻滞剂:5-羟色胺转运蛋白 (SERT)(Ki = 0.14 nM),去甲肾上腺素转运蛋白(NET)(Ki = 54 nM),多巴胺转运蛋白(DAT)(Ki = 3,020 nM),甘氨酸转运蛋白(GlyT/LeuT)。 了解更多
  8. Dobutamine hydrochloride

    Catalog No. A10325
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    Adrenoceptors 激动剂
    Dobutamine hydrochloride是一种直接作用剂,其主要活性来自刺激心脏的β1肾上腺素能受体,增加收缩力和心输出量。 了解更多
  9. Roxatidine acetate hydrochloride

    Catalog No. A11921
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    Roxatidine acetate hydrochloride是一种用于溃疡治疗的组胺H2受体拮抗剂。 了解更多
  10. Hydralazine hydrochloride

    Catalog No. A10455
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    Hydralazine hydrochloride是肼屈嗪的盐酸盐(安普索林),是一种直接作用的平滑肌松弛剂,IC50为1.9 mM。 了解更多
  11. Lincomycin hydrochloride (U-10149A)

    Catalog No. A10532
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    Lincomycin hydrochloride是Lincomycin的一水盐,是从林肯链霉菌中分离的林肯酰胺抗生素,据报道其抑制细菌蛋白质合成并依赖于浓度。 了解更多
  12. Phenformin hydrochloride

    Catalog No. A10717
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    Phenformin hydrochloride是双胍类药物中苯乙双胍的盐酸盐,具有抗糖尿病活性。 了解更多
  13. Oxymetazoline hydrochloride

    Catalog No. A10686
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    alpha-1 adrenergic 激动剂
    Oxymetazoline是一种选择性的α-1激动剂和部分α-2激动剂局部减充血剂,以盐酸羟甲唑啉的形式使用。 了解更多
  14. 5-Aminolevulinic acid hydrochloride

    Catalog No. A10016
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    5-Aminolevulinic acid hydrochloride是天然存在的氨基酸。四吡咯的前体在叶绿素和血红素生物合成中的作用。 了解更多
  15. Sinomenine hydrochloride

    Catalog No. A12221
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    Sinomenine hydrochloride增强人肝癌细胞中依赖COX-2途径的抗转铁蛋白受体抗体的抑制作用。 了解更多
  16. Guvacine hydrochloride

    Catalog No. A13613
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    GABA uptake 抑制剂
    Guvacine hydrochloride可抑制GABA的摄取(hGABA T-1,rGABA T-2,hGABA T-3和hBGT-1的IC50值分别为14、58、119和1870 uM)。 了解更多
  17. Chitosamine hydrochloride

    Catalog No. A14821
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    Chitosamine hydrochloride从天然几丁质中提取。 了解更多
  18. Tamsulosin hydrochloride

    Catalog No. A14936
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    α1 receptor 拮抗剂
    Tamsulosin hydrochloride是一种选择性的α1受体拮抗剂,是用于良性前列腺增生的药物。 了解更多
  19. DPPI 1c hydrochloride

    Catalog No. A15298
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    DPP-4 抑制剂
    DPPI 1c hydrochloride是一种双氰基吡咯烷化合物,可作为CD26(DPP 4)的缓慢结合和定点活性抑制剂,IC50 = 106 nM,对DPP II,DPP III,DPP VIII,DPP IX,FAP几乎没有活性,甚至浓度高达30μM的APP。 了解更多
  20. NSC 146109 hydrochloride

    Catalog No. A15349
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    p53 activator
    NSC 146109 hydrochloride是激活p53依赖性转录的细胞渗透性,基因型选择性抗肿瘤剂。 了解更多
  21. RETRA hydrochloride

    Catalog No. A15351
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    mutant p53 Reactivator
    RETRA hydrochloride是一种抗肿瘤剂,在体内外均以突变的p53和p73依赖性方式抑制肿瘤细胞的生长。 了解更多
  22. UNC 926 hydrochloride

    Catalog No. A15367
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    MBT Domain (L3MBTL1) 抑制剂
    UNC 926 hydrochloride是甲基赖氨酸阅读器域抑制剂。 了解更多
  23. Asenapine HCl

    Catalog No. A15002
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    adrenergic receptor/5-HT receptor 抑制剂
    Asenapine hydrochloride抑制肾上腺素能受体(α1,α2A,α2B,α2C)的Ki为0.25-1.2 nM,还抑制5-HT受体(1A,1B,2A,2B,2C,5A,6、7),Ki为0.03- 4.0 nM。 了解更多
  24. Atrasentan HCl

    Catalog No. A15007
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    Endothelin 拮抗剂 receptor
    Atrasentan hydrochloride是一种开发用于治疗前列腺癌的内皮素拮抗剂受体(IC50 = 0.0551 nM,ETA)。 了解更多
  25. Finafloxacin hydrochloride

    Catalog No. A15472
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    Finafloxacin hydrochloride是氟喹诺酮化合物。 了解更多
  26. SCH 23390 HCl

    Catalog No. A13066
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    D1/D5 receptor 拮抗剂
    SCH 23390 HCl是一种有效的多巴胺受体拮抗剂(D1和D5受体亚型的Ki值分别为0.2 nM和0.3 nM)。 了解更多
  27. CBiPES HCl

    Catalog No. A15811
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    mGlu2 receptor modulator
    CBiPES HCl是mGluR-2的选择性正变构调节剂,IC50值为98.2 nM。 了解更多
  28. Benzocaine hydrochloride

    Catalog No. A16130
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    Benzocaine hydrochloride是一种表面麻醉剂,通过阻止脉冲沿神经纤维和神经末梢的传递而起作用。 了解更多
  29. Lidocaine hydrochloride

    Catalog No. A16132
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    Histamine H1-receptor 激动剂
    Lidocaine hydrochloride是用作抗心律不齐药物的局部麻醉药和心脏抑制剂。 了解更多
  30. Tiagabine hydrochloride

    Catalog No. A16135
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    GABA reuptake 抑制剂
    Tiagabine hydrochloride是一种抗惊厥药。该药物还用于治疗惊恐症,还有其他一些抗惊厥药。 了解更多
  31. Azasetron HCl

    Catalog No. A16417
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    5-HT3 receptor 拮抗剂
    Azasetron HCl是一种选择性的5-HT3受体拮抗剂,IC50为0.33 nM,用于治疗癌症化学疗法引起的恶心和呕吐。 了解更多
  32. Rimonabant hydrochloride

    Catalog No. A11548
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    CB1 receptor inverse 激动剂
    Rimonabant hydrochloride是CB1受体反向激动剂。 了解更多
  33. Tacrine HCl Hydrate

    Catalog No. A16970
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    AChE and BChE 抑制剂
    Tacrine hydrochloride hydrate是乙酰(AChE)和丁酰胆碱酯酶(BChE)的抑制剂,IC50分别为31 nM和25.6 nM。 了解更多
  34. Robenidine Hydrochloride

    Catalog No. A16991
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    Antibiotic
    Robenidine Hydrochloride是一种用于控制球虫病的抗生素,球虫病是一种破坏家禽的原生动物感染。 了解更多
  35. Melitracen hydrochloride

    Catalog No. A17494
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    dopamine D1/2 receptor antagonist
    Melitracen HCl ia potential dopamine D1/2 receptor antagonist used to treat depression. It is often co-administered with flupenthixol as a treatment for trigeminal neuralgia. It does not effect cardiovascular function. 了解更多
  36. Lincomycin Hydrochloride Monohydrate

    Catalog No. A17584
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    Antibacterial agent
    Lincomycin hydrochloride is a peptidyl transferase and protein translation inhibitor used to treat bacterial infections. It also inhibits growth of plasmodium. 了解更多
  37. Nefazodone hydrochloride

    Catalog No. A17622
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    5-HT2 receptors inhibitor
    Nefazodone HCl is an inhibitor of 5-HT2 receptors, SERT, NET, and hERG K+ channels used to treat mood disorders. It decreases immobility time in the forced swim test. 了解更多
  38. Rimantadine Hydrochloride

    Catalog No. A17649
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    antiviral drug
    Rimantadine is an orally administered antiviral drug used to treat, and in rare cases prevent, influenzavirus A infection. 了解更多
  39. Amiodarone hydrochloride

    Catalog No. A11798
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    Amiodarone hydrochloride is an antiarrhythmic drug for inhibition of ATP-sensitive potassium channel with IC50 of 19.1 μM. 了解更多
  40. Nicardipine hydrochloride

    Catalog No. A16634
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    calcium channel blocker
    Nicardipine hydrochloride (YC-93) is a calcium channel blocker with an IC50 of 1 μM for blocking cardiac calcium channels. 了解更多
  41. Caroverine HCl

    Catalog No. A22495
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    Caroverine hydrochloride is a potent, competitive and reversible antagonist of NMDA and AMPA glutamate receptor. Caroverine hydrochloride is also an antioxidant and calcium-blocking agent that exhibits vasorelaxant action. Caroverine hydrochloride can be used for the research of inner ear tinnitus. 了解更多
  42. Benzamidine hydrochloride

    Catalog No. A22323
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    trypsin-like serine proteases inhibitor
    Benzamidine hydrochloride is an reversible competitive inhibitor of trypsin-like serine proteases, with Kis of 97 ?M, 21 ?M, 20 ?M and 110 ?M for uPA, trypsin, tryptase and factor Xa, respectively. 了解更多
  43. Bendamustine HCl (SDX-105)

    Catalog No. A10124
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    Bendamustine Hydrochloride (SDX-105)是一种小分子双功能DNA烷基化剂,结合了氮芥菜碱功能和嘌呤类似物结构。苯达莫司汀具有致密的破坏DNA的功能,使其与用作抗增殖剂的其他化合物区分开来,这些功能被认为可通过多种不同途径(包括凋亡和有丝分裂灾难)促进细胞死亡。 了解更多
  44. Nepicastat HCl

    Catalog No. A11172
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    DBH 抑制剂
    Nepicastat HCl是多巴胺β-羟化酶的抑制剂,该酶催化多巴胺向去甲肾上腺素的转化。 了解更多
  45. Pazopanib HCl (GW786034)

    Catalog No. A10699
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    VEGFR/PDGFR/FGFR 抑制剂
    Pazopanib HCl (GW786034)是VEGFR-1,VEGFR-2,VEGFR-3,PDGFR-a/β和c-kit的有效且选择性的多靶点酪氨酸激酶抑制剂,可阻止肿瘤生长并抑制血管生成。 了解更多
  46. SKF 89976A HCl

    Catalog No. A10849
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    GABA uptake 抑制剂
    SKF 89976A HCl是一种有效的GABA吸收抑制剂,hGAT-1,rGAT-2,hGAT-3和hBGT-1的IC50分别为0.13、550、944和7210μM。 了解更多
  47. Tetrahydropapaverine HCl

    Catalog No. A10920
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    Hydroxylase 抑制剂
    Tetrahydropapaverine HCl是TIQs的一种,是Salsolinol和Tetrahydropapaveroline的类似物,对多巴胺神经元具有神经毒性作用。 了解更多
  48. BRL 52537 HCl

    Catalog No. A11210
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    Opioid Receptors 激动剂
    BRL 52537 hydrochloride是一种高度选择性和有效的κ阿片类激动剂(Ki = 0.24 nM)。比吗啡强25倍。 了解更多
  49. Rotigotine HCl

    Catalog No. A11118
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    Dopamine Receptor 激动剂
    Rotigotine hydrochloride是一种多巴胺D2和D3受体激动剂。D2和D3的Ki值分别为13和0.71 nM。 了解更多
  50. MK 3207 HCl

    Catalog No. A10598
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    CGRP Receptor 拮抗剂
    MK 3207 hydrochloride是一种有效的CGRP受体拮抗剂,IC50为0.12 nM。 了解更多

产品 1 到 50 共 695个

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