Cell Metabolism

产品 201 到 250 共 394个

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  1. Safinamide

    Catalog No. A13294
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    MAO-B 抑制剂
    Safinamide是一种高度选择性和可逆的B型单胺氧化酶(MAO-B)抑制剂,可增加新纹状体多巴胺的浓度。 了解更多
  2. RN-1 2HCl

    Catalog No. A14344
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    MAO 抑制剂
    RN-1 2HCl对LSD1的选择性优于单胺氧化酶(MAO)-A和MAO-B(在辣根过氧化物酶偶联测定中,IC50值分别为70 nM,0.51和2.79 μM)。 了解更多
  3. Clorgyline hydrochloride

    Catalog No. A17357
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    monoamine oxidase A inhibitor
    Clorgyline hydrochloride is an irreversible and selective inhibitor of monoamine oxidase A (MAO-A) that is used in scientific research; structurally related to Pargyline. 了解更多
  4. Isocarboxazid

    Catalog No. A17887
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    monoamine oxidase inhibitor
    Isocarboxazid is a non-selective and irreversible inhibitor of monoamine oxidase, with an IC50 of 4.8 μM for rat brain monoamine oxidase in vitro. 了解更多
  5. Rasagiline 13C3 mesylate racemic

    Catalog No. A21350
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    Monoamine oxidase inhibitor
    Rasagiline 13C3 mesylate racemic is the deuterium labeled Rasagiline, which is an irreversible inhibitor of monoamine oxidase. 了解更多
  6. PAT-1251 Hydrochloride

    Catalog No. A21969
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    LOXL2 inhibitor
    PAT-1251 Hydrochloride is a potent, selective and oral lysyl oxidase-like 2 (LOXL2) inhibitor, with IC50s of 0.71 and 1.17 μM for hLOXL2 and hLOXL3, respectively, and also potently inhibits mouse, rat, and dog LOXL2 (IC50s, 0.10, 0.12, and 0.16 μM, respectively). 了解更多
  7. Rasagiline

    Catalog No. A11111
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    MAO B 抑制剂
    Rasagiline是MAO-B(单胺氧化酶-B)的选择性不可逆抑制剂。 了解更多
  8. Hordenine

    Catalog No. A10454
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    MAO-B 抑制剂
    Hordenine是一种苯乙胺生物碱,具有抗菌和抗生素特性。 了解更多
  9. Quercetin (Sophoretin)

    Catalog No. A10766
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    MAO-B 抑制剂
    Quercetin (Sophoretin)抑制许多酶系统,包括酪氨酸蛋白激酶,磷脂酶A2,磷酸二酯酶,线粒体ATPase,PI 3-激酶和蛋白激酶C。 了解更多
  10. Quercetin dihydrate (Sophoretin)

    Catalog No. A10765
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    MAO-B 抑制剂
    Quercetin dihydrate (Sophoretin)抑制许多酶系统,包括酪氨酸蛋白激酶,磷脂酶A2,磷酸二酯酶,线粒体ATPase,PI 3-激酶和蛋白激酶C。 了解更多
  11. Olodaterol

    Catalog No. A15761
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    MAO 抑制剂
    Olodaterol是一种长效的β肾上腺素受体激动剂,由Boehringer-Ingelheim生产,用于吸入治疗慢性阻塞性肺疾病(COPD)患者。 了解更多
  12. Pargyline hydrochloride

    Catalog No. A17288
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    MAO inhibitor
    Pargyline hydrochloride is an irreversible inhibitor of monoamine oxidase (MAO) that is used clinically to treat moderate hypertension. 了解更多
  13. Iproniazid

    Catalog No. A17445
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    MAO inhibitor
    Iproniazid is a non-selective, irreversible monoamine oxidase (MAO) inhibitor (MAOI) that is used as an antidepressive agent. 了解更多
  14. Molindone hydrochloride

    Catalog No. A17647
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    MAO inhibitor
    Molindone HCl is a D2 dopamine receptor antagonist. It also acts as a MAO inhibitor. 了解更多
  15. Minaprine dihydrochloride

    Catalog No. A17722
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    MAO-A inhibitor
    Minaprine is a reversible inhibitor of MAO-A; weakly inhibit acetylcholinesterase; an antidepressant for treatment of depression. 了解更多
  16. Toloxatone

    Catalog No. A18043
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    MAO-A inhibitor
    Toloxatone (MD 69276) is a reversible monoamine oxidase A (MAOA) inhibitor. Antidepressant. 了解更多
  17. Iproniazid phosphate

    Catalog No. A18135
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    MAO inhibitor
    Iproniazid phosphate is an irreversible inhibitor of monoamine oxidase types A and B that is used as an antidepressive agent. It has also been used as an antitubercular agent, but its use is limited by its toxicity. 了解更多
  18. TB5

    Catalog No. A13170
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    hMAO-B inhibitor
    TB5 is a potent, selective and reversible inhibitor of hMAO-B with a Ki value of 0.11??0.01 μM. 了解更多
  19. CX-157

    Catalog No. A12200
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    MAO-A inhibitor
    CX-157 is a reversible inhibitor of monoamine oxidase-A (MAO-A) with an EC50 of 19.3?ng/mL. 了解更多
  20. Salsolidine

    Catalog No. A12969
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    MAO-A inhibitor
    Salsolidine is a tetrahydroisoquinoline alkaloid, acts as a stereoselective competitive MAO A inhibitor. 了解更多
  21. RS 8359

    Catalog No. A21240
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    MAO-A inhibitor
    RS 8359 is a selective and reversible MAO-A inhibitor, with antidepressant activity. 了解更多
  22. Lazabemide

    Catalog No. A21270
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    MAO-B inhibitor
    Lazabemide(Ro 19-6327) is selective, reversible monoamine oxidase B (MAO-B) inhibitor (IC50 values are 0.03 and > 100 μM for MAO-B and MAO-A respectively). 了解更多
  23. Ro 41-1049 hydrochloride

    Catalog No. A21672
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    inhibitor of monoamine oxidase-A (MAO-A)
    Ro 41-1049 hydrochloride is a reversible and selective inhibitor of monoamine oxidase-A (MAO-A). 了解更多
  24. Brofaromine

    Catalog No. A21777
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    MAO inhibitor
    Brofaromine (CGP 11305A) is a monoamine oxidase (MAO) inhibitor with IC50 of 0.2?μM for MAO-A. 了解更多
  25. Apixaban (BMS-562247-01)

    Catalog No. A10082
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    Factor Xa 抑制剂
    Apixaban (BMS-562247-01)是一种抗凝剂,用于预防静脉血栓栓塞和静脉血栓栓塞事件。 了解更多
  26. BMS-740808

    Catalog No. A10158
    Factor Xa 抑制剂
    BMS-740808是凝血因子Xa的高效,选择性,有效和口服生物利用度抑制剂。 了解更多
  27. Rivaroxaban (Xarelto)

    Catalog No. A10800
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    Factor Xa 抑制剂
    Rivaroxaban (Xarelto)是一种Factor Xa的直接抑制剂,无细胞试验中Ki和IC50分别为0.4 nM和0.7 nM。 了解更多
  28. Otamixaban (FXV 673)

    Catalog No. A11517
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    factor Xa 抑制剂
    Otamixaban (FXV 673)是一种静脉内直接因子Xa抑制剂。 了解更多
  29. Razaxaban

    Catalog No. A12870
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    factor Xa 抑制剂
    Razaxaban是凝血因子Xa的选择性,有效和口服生物利用抑制剂。 了解更多
  30. Letaxaban (TAK-442)

    Catalog No. A12871
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    factor Xa 抑制剂
    Letaxaban (TAK-442)是一种有效的,选择性的,口服活性的Xa抑制剂,是一种四氢嘧啶-2(1H)-衍生物。TAK-442在贫血小板的人[半最大抑制浓度(IC(50)):53 nM,TAK-442]和大鼠(IC(50):32 nM,TAK-442)血浆中抑制内源性FXa活性。 了解更多
  31. Betrixaban

    Catalog No. A12518
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    FXa 抑制剂
    Betrixaban是一种抗凝血药,可作为直接Xa因子抑制剂。它具有强大的,口服活性和对因子Xa的高度选择性,由于其低hERG亲和力而从一组相似的化合物中选择。 了解更多
  32. ABT333

    Catalog No. A13878
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    NS5B 抑制剂
    ABT333是NS5B非核苷聚合酶抑制剂。 了解更多
  33. DPC-423

    Catalog No. A14099
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    factor Xa 抑制剂
    DPC423是一种高效且可口服生物利用的吡唑抗血栓形成剂。 了解更多
  34. Edoxaban (tosylate Monohydrate)

    Catalog No. A14317
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    Factor Xa 抑制剂
    Edoxaban (tosylate Monohydrate)是选择性Factor Xa抑制剂,Ki为0.561 nM。 了解更多
  35. 5-R-Rivaroxaban

    Catalog No. A14979
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    Factor Xa 抑制剂
    5-R-Rivaroxaban是利伐沙班的(R)对映异构体。利伐沙班是一种新型的口服直接Xa因子抑制剂,在晚期开发中用于预防和治疗血栓栓塞性疾病。 了解更多
  36. Edoxaban tosylate

    Catalog No. A15076
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    Factor Xa 抑制剂
    Edoxaban tosylate是临床预防卒中的口服Xa(FXa)抑制剂。 了解更多
  37. Fondaparinux Sodium

    Catalog No. A17918
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    factor Xa inhibitor
    Fondaparinux sodium is a factor Xa inhibitor to form the high affinity binding site for the anti-coagulant factor antithrombin III (ATIII). 了解更多
  38. RWJ-445167

    Catalog No. A12154
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    dual inhibitor of thrombin and factor Xa
    RWJ-445167 (3DP-10017) is a dual inhibitor of thrombin and factor Xa with Ki of 4.0 nM and 230 nM, respectively, exhibiting potent antithrombotic activity. 了解更多
  39. Edoxaban

    Catalog No. A18015
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    factor Xa (FXa) inhibitor
    Edoxaban(DU-176) is an oral factor Xa (FXa) inhibitor in clinical development for stroke prevention. 了解更多
  40. BMS-654457

    Catalog No. A21704
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    Factor XIa (FXIa) inhibitor
    BMS-654457 is a small-molecule, reversible inhibitor of factor XIa (FXIa), binding with human and rabbit FXIa with Kis of 0.2 and 0.42 nM, respectively. 了解更多
  41. Nepicastat HCl

    Catalog No. A11172
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    DBH 抑制剂
    Nepicastat HCl是多巴胺β-羟化酶的抑制剂,该酶催化多巴胺向去甲肾上腺素的转化。 了解更多
  42. Tetrahydropapaverine HCl

    Catalog No. A10920
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    Hydroxylase 抑制剂
    Tetrahydropapaverine HCl是TIQs的一种,是Salsolinol和Tetrahydropapaveroline的类似物,对多巴胺神经元具有神经毒性作用。 了解更多
  43. LX 1606 Hippurate

    Catalog No. A10542
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    Hydroxylase 抑制剂
    LX 1606 hippurate是一种口服生物可利用的小分子色氨酸羟化酶(TPH)抑制剂,具有潜在的抗旋转能活性。 了解更多
  44. Nepicastat (free base) (SYN-117)

    Catalog No. A10637
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    dopamine beta-hydroxylase 抑制剂
    Nepicastat (free base) (SYN-117)是多巴胺β-羟化酶的抑制剂,该酶催化多巴胺向去甲肾上腺素的转化。 了解更多
  45. LX 1606 (Telotristat)

    Catalog No. A11785
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    Serotonin synthesis 抑制剂
    LX 1606 (Telotristat)是一种口服生物可利用的小分子色氨酸羟化酶(TPH)抑制剂,具有潜在的抗血清素活性。 了解更多
  46. Ro 61-8048

    Catalog No. A12833
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    Hydroxylase 抑制剂
    Ro 61-8048是有效的竞争性犬尿氨酸3-羟化酶抑制剂(Ki = 4.8 nM,IC50 = 37 nM)。 了解更多
  47. Metyrapone

    Catalog No. A13363
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    Cytochrome P450 抑制剂
    Metyrapone抑制P450介导的ω/ω-1羟化酶活性和CYP11B1。 了解更多
  48. DMOG

    Catalog No. A13998
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    HIF-PH 抑制剂
    DMOG是HIF-PH的细胞渗透性竞争性抑制剂。它可在正常的氧气张力下(0.1至1 mM的浓度)稳定HIF-1α表达。 了解更多
  49. LP-533401

    Catalog No. A14325
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    Tph1 抑制剂
    LP-533401是Tph1的小分子抑制剂。 了解更多
  50. Collagen proline hydroxylase inhibitor

    Catalog No. A11371
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    Collagen proline hydroxylase 抑制剂
    Collagen proline hydroxylase抑制剂是胶原脯氨酸羟化酶抑制剂。 了解更多

产品 201 到 250 共 394个

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